Conformational Study of n,n’-(Alkane-1,n-diyl)bis(2-phenyl-3,5-dihydro-4<i>H</i>-imidazol-4-one)s with Different Spacer Length

In this study, we investigated the conformational abilities of n,n’-(Alkanediyl)-bis(2-phenyl-3,5-dihydro-4<i>H</i>-imidazol-4-one)s (<b>1</b>) to gain insight into their biological potential as a platform for the generation of various QACs. Among the conformers of <b>1...

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Main Authors: Anastasia A. Lobankova, Vyacheslav S. Grinev, Alevtina Yu. Yegorova
Format: Article
Language:English
Published: MDPI AG 2023-11-01
Series:Chemistry Proceedings
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Online Access:https://www.mdpi.com/2673-4583/14/1/6
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author Anastasia A. Lobankova
Vyacheslav S. Grinev
Alevtina Yu. Yegorova
author_facet Anastasia A. Lobankova
Vyacheslav S. Grinev
Alevtina Yu. Yegorova
author_sort Anastasia A. Lobankova
collection DOAJ
description In this study, we investigated the conformational abilities of n,n’-(Alkanediyl)-bis(2-phenyl-3,5-dihydro-4<i>H</i>-imidazol-4-one)s (<b>1</b>) to gain insight into their biological potential as a platform for the generation of various QACs. Among the conformers of <b>1</b>, due to the flexibility of the polymethylene fragment, the phenyl rings can take on different mutual arrangements, while there is a clear tendency for the formation of π–π interactions. From the point of view of the reactivity to alkylating agents, a preliminary conclusion can be drawn about the favorable mutual arrangement of imidazolone rings located at a sufficient distance to carry out both mono- and bisalkylation to obtain bis-QAC.
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issn 2673-4583
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publishDate 2023-11-01
publisher MDPI AG
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series Chemistry Proceedings
spelling doaj-art-9e4ff838d16f49659e0c393fb03705c22025-08-20T02:00:29ZengMDPI AGChemistry Proceedings2673-45832023-11-01141610.3390/ecsoc-27-16053Conformational Study of n,n’-(Alkane-1,n-diyl)bis(2-phenyl-3,5-dihydro-4<i>H</i>-imidazol-4-one)s with Different Spacer LengthAnastasia A. Lobankova0Vyacheslav S. Grinev1Alevtina Yu. Yegorova2Institute of Chemistry, N.G. Chernyshevsky Saratov National Research State University, 83 Ulitsa Astrakhanskaya, 410012 Saratov, RussiaInstitute of Chemistry, N.G. Chernyshevsky Saratov National Research State University, 83 Ulitsa Astrakhanskaya, 410012 Saratov, RussiaInstitute of Chemistry, N.G. Chernyshevsky Saratov National Research State University, 83 Ulitsa Astrakhanskaya, 410012 Saratov, RussiaIn this study, we investigated the conformational abilities of n,n’-(Alkanediyl)-bis(2-phenyl-3,5-dihydro-4<i>H</i>-imidazol-4-one)s (<b>1</b>) to gain insight into their biological potential as a platform for the generation of various QACs. Among the conformers of <b>1</b>, due to the flexibility of the polymethylene fragment, the phenyl rings can take on different mutual arrangements, while there is a clear tendency for the formation of π–π interactions. From the point of view of the reactivity to alkylating agents, a preliminary conclusion can be drawn about the favorable mutual arrangement of imidazolone rings located at a sufficient distance to carry out both mono- and bisalkylation to obtain bis-QAC.https://www.mdpi.com/2673-4583/14/1/6bis-imidazolonesquantum chemical calculationsconformational studyquaternary ammonium compound precursors
spellingShingle Anastasia A. Lobankova
Vyacheslav S. Grinev
Alevtina Yu. Yegorova
Conformational Study of n,n’-(Alkane-1,n-diyl)bis(2-phenyl-3,5-dihydro-4<i>H</i>-imidazol-4-one)s with Different Spacer Length
Chemistry Proceedings
bis-imidazolones
quantum chemical calculations
conformational study
quaternary ammonium compound precursors
title Conformational Study of n,n’-(Alkane-1,n-diyl)bis(2-phenyl-3,5-dihydro-4<i>H</i>-imidazol-4-one)s with Different Spacer Length
title_full Conformational Study of n,n’-(Alkane-1,n-diyl)bis(2-phenyl-3,5-dihydro-4<i>H</i>-imidazol-4-one)s with Different Spacer Length
title_fullStr Conformational Study of n,n’-(Alkane-1,n-diyl)bis(2-phenyl-3,5-dihydro-4<i>H</i>-imidazol-4-one)s with Different Spacer Length
title_full_unstemmed Conformational Study of n,n’-(Alkane-1,n-diyl)bis(2-phenyl-3,5-dihydro-4<i>H</i>-imidazol-4-one)s with Different Spacer Length
title_short Conformational Study of n,n’-(Alkane-1,n-diyl)bis(2-phenyl-3,5-dihydro-4<i>H</i>-imidazol-4-one)s with Different Spacer Length
title_sort conformational study of n n alkane 1 n diyl bis 2 phenyl 3 5 dihydro 4 i h i imidazol 4 one s with different spacer length
topic bis-imidazolones
quantum chemical calculations
conformational study
quaternary ammonium compound precursors
url https://www.mdpi.com/2673-4583/14/1/6
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