Identification of Homeobox Transcription Factors in a Dimorphic Fungus <i>Talaromyces marneffei</i> and Protein-Protein Interaction Prediction of RfeB

<i>Talaromyces marneffei</i> is a thermally dimorphic fungus that can cause life-threatening systemic mycoses, particularly in immunocompromised individuals. Fungal homeobox transcription factors control various developmental processes, including the regulation of sexual reproduction, mo...

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Main Authors: Monsicha Pongpom, Nopawit Khamto, Panwarit Sukantamala, Thitisuda Kalawil, Tanaporn Wangsanut
Format: Article
Language:English
Published: MDPI AG 2024-09-01
Series:Journal of Fungi
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Online Access:https://www.mdpi.com/2309-608X/10/10/687
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author Monsicha Pongpom
Nopawit Khamto
Panwarit Sukantamala
Thitisuda Kalawil
Tanaporn Wangsanut
author_facet Monsicha Pongpom
Nopawit Khamto
Panwarit Sukantamala
Thitisuda Kalawil
Tanaporn Wangsanut
author_sort Monsicha Pongpom
collection DOAJ
description <i>Talaromyces marneffei</i> is a thermally dimorphic fungus that can cause life-threatening systemic mycoses, particularly in immunocompromised individuals. Fungal homeobox transcription factors control various developmental processes, including the regulation of sexual reproduction, morphology, metabolism, and virulence. However, the function of homeobox proteins in <i>T. marneffei</i> has not been fully explored. Here, we searched the <i>T. marneffei</i> genome for the total homeobox transcription factors and predicted their biological relevance by performing gene expression analysis in different cell types, including conidia, mycelia, yeasts, and during phase transition. RfeB is selected for further computational analysis since (i) its transcripts were differentially expressed in different phases of <i>T. marneffei</i>, and (ii) this protein contains the highly conserved protein-protein interaction region (IR), which could be important for pathobiology and have therapeutic application. To assess the structure-function of the IR region, in silico alanine substitutions were performed at three-conserved IR residues (Asp276, Glu279, and Gln282) of RfeB, generating a triple RfeB mutated protein. Using 3D modeling and molecular dynamics simulations, we compared the protein complex formation of wild-type and mutated RfeB proteins with the putative partner candidate TmSwi5. Our results demonstrated that the mutated RfeB protein exhibited increased free binding energy, elevated protein compactness, and a reduced number of atomic contacts, suggesting disrupted protein stability and interaction. Notably, our model revealed that the IR residues primarily stabilized the RfeB binding sites located in the central region (CR). This computational approach for protein mutagenesis could provide a foundation for future experimental studies on the functional characterization of RfeB and other homeodomain-containing proteins in <i>T. marneffei</i>.
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spelling doaj-art-9e198481b66f43dcae7c92fcfa616b622025-08-20T02:10:54ZengMDPI AGJournal of Fungi2309-608X2024-09-01101068710.3390/jof10100687Identification of Homeobox Transcription Factors in a Dimorphic Fungus <i>Talaromyces marneffei</i> and Protein-Protein Interaction Prediction of RfeBMonsicha Pongpom0Nopawit Khamto1Panwarit Sukantamala2Thitisuda Kalawil3Tanaporn Wangsanut4Department of Microbiology, Faculty of Medicine, Chiang Mai University, Chiang Mai 50200, ThailandDepartment of Chemistry, Faculty of Science, Chiang Mai University, Chiang Mai 50200, ThailandFaculty of Dentistry, Chiang Mai University, Chiang Mai 50200, ThailandDepartment of Microbiology, Faculty of Medicine, Chiang Mai University, Chiang Mai 50200, ThailandDepartment of Microbiology, Faculty of Medicine, Chiang Mai University, Chiang Mai 50200, Thailand<i>Talaromyces marneffei</i> is a thermally dimorphic fungus that can cause life-threatening systemic mycoses, particularly in immunocompromised individuals. Fungal homeobox transcription factors control various developmental processes, including the regulation of sexual reproduction, morphology, metabolism, and virulence. However, the function of homeobox proteins in <i>T. marneffei</i> has not been fully explored. Here, we searched the <i>T. marneffei</i> genome for the total homeobox transcription factors and predicted their biological relevance by performing gene expression analysis in different cell types, including conidia, mycelia, yeasts, and during phase transition. RfeB is selected for further computational analysis since (i) its transcripts were differentially expressed in different phases of <i>T. marneffei</i>, and (ii) this protein contains the highly conserved protein-protein interaction region (IR), which could be important for pathobiology and have therapeutic application. To assess the structure-function of the IR region, in silico alanine substitutions were performed at three-conserved IR residues (Asp276, Glu279, and Gln282) of RfeB, generating a triple RfeB mutated protein. Using 3D modeling and molecular dynamics simulations, we compared the protein complex formation of wild-type and mutated RfeB proteins with the putative partner candidate TmSwi5. Our results demonstrated that the mutated RfeB protein exhibited increased free binding energy, elevated protein compactness, and a reduced number of atomic contacts, suggesting disrupted protein stability and interaction. Notably, our model revealed that the IR residues primarily stabilized the RfeB binding sites located in the central region (CR). This computational approach for protein mutagenesis could provide a foundation for future experimental studies on the functional characterization of RfeB and other homeodomain-containing proteins in <i>T. marneffei</i>.https://www.mdpi.com/2309-608X/10/10/687Hox proteinhomeoboxhomeodomainmolecular dynamics<i>Talaromyces marneffei</i>morphogenesis
spellingShingle Monsicha Pongpom
Nopawit Khamto
Panwarit Sukantamala
Thitisuda Kalawil
Tanaporn Wangsanut
Identification of Homeobox Transcription Factors in a Dimorphic Fungus <i>Talaromyces marneffei</i> and Protein-Protein Interaction Prediction of RfeB
Journal of Fungi
Hox protein
homeobox
homeodomain
molecular dynamics
<i>Talaromyces marneffei</i>
morphogenesis
title Identification of Homeobox Transcription Factors in a Dimorphic Fungus <i>Talaromyces marneffei</i> and Protein-Protein Interaction Prediction of RfeB
title_full Identification of Homeobox Transcription Factors in a Dimorphic Fungus <i>Talaromyces marneffei</i> and Protein-Protein Interaction Prediction of RfeB
title_fullStr Identification of Homeobox Transcription Factors in a Dimorphic Fungus <i>Talaromyces marneffei</i> and Protein-Protein Interaction Prediction of RfeB
title_full_unstemmed Identification of Homeobox Transcription Factors in a Dimorphic Fungus <i>Talaromyces marneffei</i> and Protein-Protein Interaction Prediction of RfeB
title_short Identification of Homeobox Transcription Factors in a Dimorphic Fungus <i>Talaromyces marneffei</i> and Protein-Protein Interaction Prediction of RfeB
title_sort identification of homeobox transcription factors in a dimorphic fungus i talaromyces marneffei i and protein protein interaction prediction of rfeb
topic Hox protein
homeobox
homeodomain
molecular dynamics
<i>Talaromyces marneffei</i>
morphogenesis
url https://www.mdpi.com/2309-608X/10/10/687
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