Low nanomolar affinity to major grass pollen allergen Phl p 5 as achieved in an unmutated human antibody-lineage ancestor

BackgroundGroup 5 allergens, such as Phl p 5 of timothy grass, are major contributors to grass pollen allergy. Antibody 212597 specific for this allergen was recently isolated by single cell sequencing of bone marrow B cells of a grass pollen-allergic subject. This antibody, although subjected only...

Full description

Saved in:
Bibliographic Details
Main Authors: Mattias Essén, Eric Franciskovic, Céleste Sele, Magdalena Godzwon, Mats Ohlin
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-07-01
Series:Frontiers in Immunology
Subjects:
Online Access:https://www.frontiersin.org/articles/10.3389/fimmu.2025.1600778/full
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850107054945992704
author Mattias Essén
Eric Franciskovic
Céleste Sele
Magdalena Godzwon
Mats Ohlin
Mats Ohlin
author_facet Mattias Essén
Eric Franciskovic
Céleste Sele
Magdalena Godzwon
Mats Ohlin
Mats Ohlin
author_sort Mattias Essén
collection DOAJ
description BackgroundGroup 5 allergens, such as Phl p 5 of timothy grass, are major contributors to grass pollen allergy. Antibody 212597 specific for this allergen was recently isolated by single cell sequencing of bone marrow B cells of a grass pollen-allergic subject. This antibody, although subjected only to a low level of hypermutation resulting in six amino acid substitution across the heavy and light chain variable domains, has achieved sub-nM affinity for the allergen, suggesting that antibodies specific for this major group of allergens can be of high affinity even at the naïve, unmutated stage. The present study was designed to assess affinity and biophysical characters of the antibody, its inferred unmutated ancestor, and other intermediate and allelic variants thereof.MethodsSite-directed mutagenesis was used to revert substitutions of antibody 212579. Mutants, including its inferred unmutated common ancestor were characterized with respect to allergen affinity, thermostability, and hydrodynamic radius.ResultsWe demonstrate that even the antibody’s inferred unmutated common ancestor shows high affinity for the allergen in the low-nM range. Glutamate at heavy chain position 38, a residue unique to allele IGHV3-48*03, the germline gene origin of the heavy chain of antibody 212579, was critical for high affinity binding. Substitution to serine as found in other alleles of IGHV3–48 reduced the affinity about 20-fold. A substitution, N40HT in the heavy/light chain variable domain interface, introduced into the antibody through somatic hypermutation, did not impact its affinity for the allergen but reduced its thermal stability and increased its hydrodynamic radius.ConclusionUnmutated, high affinity (low-nM) antibodies specific for a major allergen (Phl p 5) can be generated directly in naïve B cells and are, given an appropriate rearrangement, imprinted into the repertoire through rearrangements involving immunoglobulin germline gene alleles IGHV3-48*03 and IGKV3-20*01. This specificity depends on an allele-unique residue encoded by the immunoglobulin germline repertoire. Substitutions in the heavy/light chain variable domain interface, such as N40HT in a heavy chain variable domain, might negatively impact biophysical properties of the antibody and should be considered as targets for further evolution or reversion if they negatively impact an antibody’s developability properties.
format Article
id doaj-art-9d5ec11a1be6460b932a34234e0e6992
institution OA Journals
issn 1664-3224
language English
publishDate 2025-07-01
publisher Frontiers Media S.A.
record_format Article
series Frontiers in Immunology
spelling doaj-art-9d5ec11a1be6460b932a34234e0e69922025-08-20T02:38:41ZengFrontiers Media S.A.Frontiers in Immunology1664-32242025-07-011610.3389/fimmu.2025.16007781600778Low nanomolar affinity to major grass pollen allergen Phl p 5 as achieved in an unmutated human antibody-lineage ancestorMattias Essén0Eric Franciskovic1Céleste Sele2Magdalena Godzwon3Mats Ohlin4Mats Ohlin5Department of Immunotechnology, Lund University, Lund, SwedenDepartment of Immunotechnology, Lund University, Lund, SwedenLund Protein Production Platform LP3, Department of Biology, Lund University, Lund, SwedenDepartment of Immunotechnology, Lund University, Lund, SwedenDepartment of Immunotechnology, Lund University, Lund, SwedenSciLifeLab, Lund University, Lund, SwedenBackgroundGroup 5 allergens, such as Phl p 5 of timothy grass, are major contributors to grass pollen allergy. Antibody 212597 specific for this allergen was recently isolated by single cell sequencing of bone marrow B cells of a grass pollen-allergic subject. This antibody, although subjected only to a low level of hypermutation resulting in six amino acid substitution across the heavy and light chain variable domains, has achieved sub-nM affinity for the allergen, suggesting that antibodies specific for this major group of allergens can be of high affinity even at the naïve, unmutated stage. The present study was designed to assess affinity and biophysical characters of the antibody, its inferred unmutated ancestor, and other intermediate and allelic variants thereof.MethodsSite-directed mutagenesis was used to revert substitutions of antibody 212579. Mutants, including its inferred unmutated common ancestor were characterized with respect to allergen affinity, thermostability, and hydrodynamic radius.ResultsWe demonstrate that even the antibody’s inferred unmutated common ancestor shows high affinity for the allergen in the low-nM range. Glutamate at heavy chain position 38, a residue unique to allele IGHV3-48*03, the germline gene origin of the heavy chain of antibody 212579, was critical for high affinity binding. Substitution to serine as found in other alleles of IGHV3–48 reduced the affinity about 20-fold. A substitution, N40HT in the heavy/light chain variable domain interface, introduced into the antibody through somatic hypermutation, did not impact its affinity for the allergen but reduced its thermal stability and increased its hydrodynamic radius.ConclusionUnmutated, high affinity (low-nM) antibodies specific for a major allergen (Phl p 5) can be generated directly in naïve B cells and are, given an appropriate rearrangement, imprinted into the repertoire through rearrangements involving immunoglobulin germline gene alleles IGHV3-48*03 and IGKV3-20*01. This specificity depends on an allele-unique residue encoded by the immunoglobulin germline repertoire. Substitutions in the heavy/light chain variable domain interface, such as N40HT in a heavy chain variable domain, might negatively impact biophysical properties of the antibody and should be considered as targets for further evolution or reversion if they negatively impact an antibody’s developability properties.https://www.frontiersin.org/articles/10.3389/fimmu.2025.1600778/fullaffinityantibodyantibody repertoireIgEimmunoglobulin germline gene allelemolecular evolution
spellingShingle Mattias Essén
Eric Franciskovic
Céleste Sele
Magdalena Godzwon
Mats Ohlin
Mats Ohlin
Low nanomolar affinity to major grass pollen allergen Phl p 5 as achieved in an unmutated human antibody-lineage ancestor
Frontiers in Immunology
affinity
antibody
antibody repertoire
IgE
immunoglobulin germline gene allele
molecular evolution
title Low nanomolar affinity to major grass pollen allergen Phl p 5 as achieved in an unmutated human antibody-lineage ancestor
title_full Low nanomolar affinity to major grass pollen allergen Phl p 5 as achieved in an unmutated human antibody-lineage ancestor
title_fullStr Low nanomolar affinity to major grass pollen allergen Phl p 5 as achieved in an unmutated human antibody-lineage ancestor
title_full_unstemmed Low nanomolar affinity to major grass pollen allergen Phl p 5 as achieved in an unmutated human antibody-lineage ancestor
title_short Low nanomolar affinity to major grass pollen allergen Phl p 5 as achieved in an unmutated human antibody-lineage ancestor
title_sort low nanomolar affinity to major grass pollen allergen phl p 5 as achieved in an unmutated human antibody lineage ancestor
topic affinity
antibody
antibody repertoire
IgE
immunoglobulin germline gene allele
molecular evolution
url https://www.frontiersin.org/articles/10.3389/fimmu.2025.1600778/full
work_keys_str_mv AT mattiasessen lownanomolaraffinitytomajorgrasspollenallergenphlp5asachievedinanunmutatedhumanantibodylineageancestor
AT ericfranciskovic lownanomolaraffinitytomajorgrasspollenallergenphlp5asachievedinanunmutatedhumanantibodylineageancestor
AT celestesele lownanomolaraffinitytomajorgrasspollenallergenphlp5asachievedinanunmutatedhumanantibodylineageancestor
AT magdalenagodzwon lownanomolaraffinitytomajorgrasspollenallergenphlp5asachievedinanunmutatedhumanantibodylineageancestor
AT matsohlin lownanomolaraffinitytomajorgrasspollenallergenphlp5asachievedinanunmutatedhumanantibodylineageancestor
AT matsohlin lownanomolaraffinitytomajorgrasspollenallergenphlp5asachievedinanunmutatedhumanantibodylineageancestor