Synthesis, Experimental and Computational Evaluation of SERAAK1 as a 5-HT<sub>2A</sub> Receptor Ligand

Synthesis, Experimental and Computational Evaluation of SERAAK1 as a 5-HT<sub>2A</sub> Receptor Ligand

Many drug discovery efforts have identified potentially promising molecules; however, a common limitation of these reports is the lack of further experimental confirmation of pharmacokinetic properties and behavioral effects of discovered compounds. In this study, we aim to address this limitation....

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Bibliographic Details
Main Authors:	Agata Zięba, Ewa Kędzierska, Michał K. Jastrzębski, Tadeusz Karcz, Agnieszka Olejarz-Maciej, Agata Sumara, Tuomo Laitinen, Tomasz M. Wróbel, Emilia Fornal, Marián Castro, Agnieszka A. Kaczor
Format:	Article
Language:	English
Published:	MDPI AG 2025-05-01
Series:	Molecules
Subjects:	5-HT<sub>2A</sub> receptor ADMET antidepressants antipsychotics in vivo studies molecular modeling
Online Access:	https://www.mdpi.com/1420-3049/30/10/2165
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