Degradation of Natural <i>Undaria pinnatifida</i> into Unsaturated Guluronic Acid Oligosaccharides by a Single Alginate Lyase

Here, we report on a bifunctional alginate lyase (Vnalg7) expressed in <i>Pichia pastoris</i>, which can degrade natural <i>Undaria pinnatifida</i> into unsaturated guluronic acid di- and trisaccharide without pretreatment. The enzyme activity of Vnalg7 (3620.00 U/mL-culture)...

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Main Authors: Hui Wang, Jiaqi Wen, Nuraliya Ablimit, Kun Deng, Wenzhuo Wang, Wei Jiang
Format: Article
Language:English
Published: MDPI AG 2024-10-01
Series:Marine Drugs
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Online Access:https://www.mdpi.com/1660-3397/22/10/453
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author Hui Wang
Jiaqi Wen
Nuraliya Ablimit
Kun Deng
Wenzhuo Wang
Wei Jiang
author_facet Hui Wang
Jiaqi Wen
Nuraliya Ablimit
Kun Deng
Wenzhuo Wang
Wei Jiang
author_sort Hui Wang
collection DOAJ
description Here, we report on a bifunctional alginate lyase (Vnalg7) expressed in <i>Pichia pastoris</i>, which can degrade natural <i>Undaria pinnatifida</i> into unsaturated guluronic acid di- and trisaccharide without pretreatment. The enzyme activity of Vnalg7 (3620.00 U/mL-culture) was 15.81-fold higher than that of the original <i>alg</i> (228.90 U/mL-culture), following engineering modification. The degradation rate reached 52.75%, and reducing sugar reached 30.30 mg/mL after combining Vnalg7 (200.00 U/mL-culture) and 14% (<i>w</i>/<i>v</i>) <i>U. pinnatifida</i> for 6 h. Analysis of the action mode indicated that Vnalg7 could degrade many substrates to produce a variety of unsaturated alginate oligosaccharides (AOSs), and the minimal substrate was tetrasaccharide. Site-directed mutagenesis showed that Glu<sup>238</sup>, Glu<sup>241</sup>, Glu<sup>312</sup>, Arg<sup>236</sup>, His<sup>307</sup>, Lys<sup>414</sup>, and Tyr<sup>418</sup> are essential catalytic sites, while Glu<sup>334</sup>, Glu<sup>344</sup>, and Asp<sup>311</sup> play auxiliary roles. Mechanism analysis revealed the enzymatic degradation pattern of Vnalg7, which mainly recognizes and attacks the third glycosidic linkage from the reducing end of oligosaccharide substrate. Our findings provide a novel alginate lyase tool and a sustainable and commercial production strategy for value-added biomolecules using seaweeds.
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publishDate 2024-10-01
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spelling doaj-art-9bbef1d1a6b64da9b1ee0539b46c08812025-08-20T02:10:56ZengMDPI AGMarine Drugs1660-33972024-10-01221045310.3390/md22100453Degradation of Natural <i>Undaria pinnatifida</i> into Unsaturated Guluronic Acid Oligosaccharides by a Single Alginate LyaseHui Wang0Jiaqi Wen1Nuraliya Ablimit2Kun Deng3Wenzhuo Wang4Wei Jiang5State Key Laboratory of Animal Biotech Breeding, College of Biological Sciences, China Agricultural University, Yuan Ming Yuan West Road No. 2, Haidian District, Beijing 100193, ChinaState Key Laboratory of Animal Biotech Breeding, College of Biological Sciences, China Agricultural University, Yuan Ming Yuan West Road No. 2, Haidian District, Beijing 100193, ChinaState Key Laboratory of Animal Biotech Breeding, College of Biological Sciences, China Agricultural University, Yuan Ming Yuan West Road No. 2, Haidian District, Beijing 100193, ChinaState Key Laboratory of Animal Biotech Breeding, College of Biological Sciences, China Agricultural University, Yuan Ming Yuan West Road No. 2, Haidian District, Beijing 100193, ChinaState Key Laboratory of Animal Biotech Breeding, College of Biological Sciences, China Agricultural University, Yuan Ming Yuan West Road No. 2, Haidian District, Beijing 100193, ChinaState Key Laboratory of Animal Biotech Breeding, College of Biological Sciences, China Agricultural University, Yuan Ming Yuan West Road No. 2, Haidian District, Beijing 100193, ChinaHere, we report on a bifunctional alginate lyase (Vnalg7) expressed in <i>Pichia pastoris</i>, which can degrade natural <i>Undaria pinnatifida</i> into unsaturated guluronic acid di- and trisaccharide without pretreatment. The enzyme activity of Vnalg7 (3620.00 U/mL-culture) was 15.81-fold higher than that of the original <i>alg</i> (228.90 U/mL-culture), following engineering modification. The degradation rate reached 52.75%, and reducing sugar reached 30.30 mg/mL after combining Vnalg7 (200.00 U/mL-culture) and 14% (<i>w</i>/<i>v</i>) <i>U. pinnatifida</i> for 6 h. Analysis of the action mode indicated that Vnalg7 could degrade many substrates to produce a variety of unsaturated alginate oligosaccharides (AOSs), and the minimal substrate was tetrasaccharide. Site-directed mutagenesis showed that Glu<sup>238</sup>, Glu<sup>241</sup>, Glu<sup>312</sup>, Arg<sup>236</sup>, His<sup>307</sup>, Lys<sup>414</sup>, and Tyr<sup>418</sup> are essential catalytic sites, while Glu<sup>334</sup>, Glu<sup>344</sup>, and Asp<sup>311</sup> play auxiliary roles. Mechanism analysis revealed the enzymatic degradation pattern of Vnalg7, which mainly recognizes and attacks the third glycosidic linkage from the reducing end of oligosaccharide substrate. Our findings provide a novel alginate lyase tool and a sustainable and commercial production strategy for value-added biomolecules using seaweeds.https://www.mdpi.com/1660-3397/22/10/453alginate lyaseaction modealginate oligosaccharidecatalytic mechanism<i>Undaria pinnatifida</i>
spellingShingle Hui Wang
Jiaqi Wen
Nuraliya Ablimit
Kun Deng
Wenzhuo Wang
Wei Jiang
Degradation of Natural <i>Undaria pinnatifida</i> into Unsaturated Guluronic Acid Oligosaccharides by a Single Alginate Lyase
Marine Drugs
alginate lyase
action mode
alginate oligosaccharide
catalytic mechanism
<i>Undaria pinnatifida</i>
title Degradation of Natural <i>Undaria pinnatifida</i> into Unsaturated Guluronic Acid Oligosaccharides by a Single Alginate Lyase
title_full Degradation of Natural <i>Undaria pinnatifida</i> into Unsaturated Guluronic Acid Oligosaccharides by a Single Alginate Lyase
title_fullStr Degradation of Natural <i>Undaria pinnatifida</i> into Unsaturated Guluronic Acid Oligosaccharides by a Single Alginate Lyase
title_full_unstemmed Degradation of Natural <i>Undaria pinnatifida</i> into Unsaturated Guluronic Acid Oligosaccharides by a Single Alginate Lyase
title_short Degradation of Natural <i>Undaria pinnatifida</i> into Unsaturated Guluronic Acid Oligosaccharides by a Single Alginate Lyase
title_sort degradation of natural i undaria pinnatifida i into unsaturated guluronic acid oligosaccharides by a single alginate lyase
topic alginate lyase
action mode
alginate oligosaccharide
catalytic mechanism
<i>Undaria pinnatifida</i>
url https://www.mdpi.com/1660-3397/22/10/453
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