Synthesis of aryl hydrazone derivatives for α-naphthalide and benzothiazolide

    Three series of new N-(α–naphthyl-2-(aryl hydrazono)-3-oxo butanamide, N-(6-chloro) benzothiazol-2-yl)-2-(aryl hydrazono)-3- oxo butanamide and N-(6-methyl) benzothiazol-2-yl)-2-(aryl hydrazono)-3- oxo butanamide were synthesized in two steps derived from α-naphthyl amine, 2-aminobenzothiazole....

Full description

Saved in:
Bibliographic Details
Main Authors: Luma S. Ahamed, Zena G. Al-Rekabi
Format: Article
Language:English
Published: University of Baghdad, College of Science for Women 2024-10-01
Series:مجلة بغداد للعلوم
Subjects:
Online Access:https://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/11923
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849410872895602688
author Luma S. Ahamed
Zena G. Al-Rekabi
author_facet Luma S. Ahamed
Zena G. Al-Rekabi
author_sort Luma S. Ahamed
collection DOAJ
description     Three series of new N-(α–naphthyl-2-(aryl hydrazono)-3-oxo butanamide, N-(6-chloro) benzothiazol-2-yl)-2-(aryl hydrazono)-3- oxo butanamide and N-(6-methyl) benzothiazol-2-yl)-2-(aryl hydrazono)-3- oxo butanamide were synthesized in two steps derived from α-naphthyl amine, 2-aminobenzothiazole. : The first step was involved the reaction of different fused aromatic amines (α-naphthyl amine, 6-chloro-2-aminobenzothiazole and 6-methyl-2- aminobenzothiazole) with methyl acetoacetate at (160-170) 0C by using modern method to provide greatly improved yields. In the second step arenediazonium chloride was added to [3-oxo-butanamide derivatives] in basic solution at (0-5) 0C to get ten new dyes of aryl hydrazono derivatives. These synthesized compounds were characterized by FT-IR, 13C-NMR, 1H-NMR, UV-Visible spectroscopy, and by measuring their melting points, and solubility.
format Article
id doaj-art-96551840b540454da63ca277dafbfd0f
institution Kabale University
issn 2078-8665
2411-7986
language English
publishDate 2024-10-01
publisher University of Baghdad, College of Science for Women
record_format Article
series مجلة بغداد للعلوم
spelling doaj-art-96551840b540454da63ca277dafbfd0f2025-08-20T03:34:57ZengUniversity of Baghdad, College of Science for Womenمجلة بغداد للعلوم2078-86652411-79862024-10-017110.21123/bsj.2010.11923Synthesis of aryl hydrazone derivatives for α-naphthalide and benzothiazolide Luma S. AhamedZena G. Al-Rekabi     Three series of new N-(α–naphthyl-2-(aryl hydrazono)-3-oxo butanamide, N-(6-chloro) benzothiazol-2-yl)-2-(aryl hydrazono)-3- oxo butanamide and N-(6-methyl) benzothiazol-2-yl)-2-(aryl hydrazono)-3- oxo butanamide were synthesized in two steps derived from α-naphthyl amine, 2-aminobenzothiazole. : The first step was involved the reaction of different fused aromatic amines (α-naphthyl amine, 6-chloro-2-aminobenzothiazole and 6-methyl-2- aminobenzothiazole) with methyl acetoacetate at (160-170) 0C by using modern method to provide greatly improved yields. In the second step arenediazonium chloride was added to [3-oxo-butanamide derivatives] in basic solution at (0-5) 0C to get ten new dyes of aryl hydrazono derivatives. These synthesized compounds were characterized by FT-IR, 13C-NMR, 1H-NMR, UV-Visible spectroscopy, and by measuring their melting points, and solubility. https://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/11923benzothiazolide, Synthesis, aryl hydrazone, α-naphthalide
spellingShingle Luma S. Ahamed
Zena G. Al-Rekabi
Synthesis of aryl hydrazone derivatives for α-naphthalide and benzothiazolide
مجلة بغداد للعلوم
benzothiazolide, Synthesis, aryl hydrazone, α-naphthalide
title Synthesis of aryl hydrazone derivatives for α-naphthalide and benzothiazolide
title_full Synthesis of aryl hydrazone derivatives for α-naphthalide and benzothiazolide
title_fullStr Synthesis of aryl hydrazone derivatives for α-naphthalide and benzothiazolide
title_full_unstemmed Synthesis of aryl hydrazone derivatives for α-naphthalide and benzothiazolide
title_short Synthesis of aryl hydrazone derivatives for α-naphthalide and benzothiazolide
title_sort synthesis of aryl hydrazone derivatives for α naphthalide and benzothiazolide
topic benzothiazolide, Synthesis, aryl hydrazone, α-naphthalide
url https://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/11923
work_keys_str_mv AT lumasahamed synthesisofarylhydrazonederivativesforanaphthalideandbenzothiazolide
AT zenagalrekabi synthesisofarylhydrazonederivativesforanaphthalideandbenzothiazolide