Analysis of Factors That Regulate HIV-1 Fusion in Reverse

Based on observations that HIV-1 envelope (Env) proteins on the surfaces of cells have the capacity to fuse with neighboring cells or enveloped viruses that express CD4 receptors and CXCR4 co-receptors, we tested factors that affect the capacities of lentiviral vectors pseudotyped with CD4 and CXCR4...

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Main Authors: Ayna Alfadhli, Robin Lid Barklis, Fikadu G. Tafesse, Eric Barklis
Format: Article
Language:English
Published: MDPI AG 2025-03-01
Series:Viruses
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Online Access:https://www.mdpi.com/1999-4915/17/4/472
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author Ayna Alfadhli
Robin Lid Barklis
Fikadu G. Tafesse
Eric Barklis
author_facet Ayna Alfadhli
Robin Lid Barklis
Fikadu G. Tafesse
Eric Barklis
author_sort Ayna Alfadhli
collection DOAJ
description Based on observations that HIV-1 envelope (Env) proteins on the surfaces of cells have the capacity to fuse with neighboring cells or enveloped viruses that express CD4 receptors and CXCR4 co-receptors, we tested factors that affect the capacities of lentiviral vectors pseudotyped with CD4 and CXCR4 variants to infect Env-expressing cells. The process, which we refer to as fusion in reverse, involves the binding and activation of cellular Env proteins to fuse membranes with lentiviruses carrying CD4 and CXCR4 proteins. We have found that infection via fusion in reverse depends on cell surface Env levels, is inhibitable by an HIV-1-specific fusion inhibitor, and preferentially requires lentiviral pseudotyping with a glycosylphosphatidylinositol (GPI)-anchored CD4 variant and a cytoplasmic tail-truncated CXCR4 protein. We have demonstrated that latently HIV-1-infected cells can be specifically infected using this mechanism, and that activation of latently infected cells increases infection efficiency. The fusion in reverse approach allowed us to characterize how alteration of CD4 plus CXCR4 lipid membranes affected Env protein activities. In particular, we found that perturbation of membrane cholesterol levels did not affect Env activity. In contrast, viruses assembled in cells deficient for long-chain sphingolipids showed increased infectivities, while viruses that incorporated a lipid scramblase were non-infectious. Our results yield new insights into factors that influence envelope protein functions.
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spelling doaj-art-9398d089135e473b938f933de6820b132025-08-20T03:13:33ZengMDPI AGViruses1999-49152025-03-0117447210.3390/v17040472Analysis of Factors That Regulate HIV-1 Fusion in ReverseAyna Alfadhli0Robin Lid Barklis1Fikadu G. Tafesse2Eric Barklis3Department of Molecular Microbiology and Immunology, Oregon Health and Science University, Portland, OR 97239, USADepartment of Molecular Microbiology and Immunology, Oregon Health and Science University, Portland, OR 97239, USADepartment of Molecular Microbiology and Immunology, Oregon Health and Science University, Portland, OR 97239, USADepartment of Molecular Microbiology and Immunology, Oregon Health and Science University, Portland, OR 97239, USABased on observations that HIV-1 envelope (Env) proteins on the surfaces of cells have the capacity to fuse with neighboring cells or enveloped viruses that express CD4 receptors and CXCR4 co-receptors, we tested factors that affect the capacities of lentiviral vectors pseudotyped with CD4 and CXCR4 variants to infect Env-expressing cells. The process, which we refer to as fusion in reverse, involves the binding and activation of cellular Env proteins to fuse membranes with lentiviruses carrying CD4 and CXCR4 proteins. We have found that infection via fusion in reverse depends on cell surface Env levels, is inhibitable by an HIV-1-specific fusion inhibitor, and preferentially requires lentiviral pseudotyping with a glycosylphosphatidylinositol (GPI)-anchored CD4 variant and a cytoplasmic tail-truncated CXCR4 protein. We have demonstrated that latently HIV-1-infected cells can be specifically infected using this mechanism, and that activation of latently infected cells increases infection efficiency. The fusion in reverse approach allowed us to characterize how alteration of CD4 plus CXCR4 lipid membranes affected Env protein activities. In particular, we found that perturbation of membrane cholesterol levels did not affect Env activity. In contrast, viruses assembled in cells deficient for long-chain sphingolipids showed increased infectivities, while viruses that incorporated a lipid scramblase were non-infectious. Our results yield new insights into factors that influence envelope protein functions.https://www.mdpi.com/1999-4915/17/4/472HIV-1fusionlipidmembranes
spellingShingle Ayna Alfadhli
Robin Lid Barklis
Fikadu G. Tafesse
Eric Barklis
Analysis of Factors That Regulate HIV-1 Fusion in Reverse
Viruses
HIV-1
fusion
lipid
membranes
title Analysis of Factors That Regulate HIV-1 Fusion in Reverse
title_full Analysis of Factors That Regulate HIV-1 Fusion in Reverse
title_fullStr Analysis of Factors That Regulate HIV-1 Fusion in Reverse
title_full_unstemmed Analysis of Factors That Regulate HIV-1 Fusion in Reverse
title_short Analysis of Factors That Regulate HIV-1 Fusion in Reverse
title_sort analysis of factors that regulate hiv 1 fusion in reverse
topic HIV-1
fusion
lipid
membranes
url https://www.mdpi.com/1999-4915/17/4/472
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