Optimizing drug design by merging generative AI with a physics-based active learning framework

Abstract Machine learning is transforming drug discovery, with generative models (GMs) gaining attention for their ability to design molecules with specific properties. However, GMs often struggle with target engagement, synthetic accessibility, or generalization. To address these, we developed a GM...

Full description

Saved in:
Bibliographic Details
Main Authors: Isaac Filella-Merce, Alexis Molina, Lucía Díaz, Marek Orzechowski, Yamina A. Berchiche, Yang Ming Zhu, Júlia Vilalta-Mor, Laura Malo, Ajay S. Yekkirala, Soumya Ray, Victor Guallar
Format: Article
Language:English
Published: Nature Portfolio 2025-08-01
Series:Communications Chemistry
Online Access:https://doi.org/10.1038/s42004-025-01635-7
Tags: Add Tag
No Tags, Be the first to tag this record!