Antidepressant activity of flavones from traditional Chinese medicine: a meta-analysis

Context Flavones, the key active components in Traditional Chinese Medicine (TCM), have demonstrated antidepressant activity. Given the numerous animal studies conducted, a systematic analysis is essential to provide a valuable reference for future research.Object This study investigated the antidep...

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Main Authors: Qing Wang, Youyuan Lu, Xue Mi, Caiyan Yang, Wei Ma, Changbo Xia, Hanqing Wang
Format: Article
Language:English
Published: Taylor & Francis Group 2025-12-01
Series:Pharmaceutical Biology
Subjects:
Online Access:https://www.tandfonline.com/doi/10.1080/13880209.2025.2467374
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author Qing Wang
Youyuan Lu
Xue Mi
Caiyan Yang
Wei Ma
Changbo Xia
Hanqing Wang
author_facet Qing Wang
Youyuan Lu
Xue Mi
Caiyan Yang
Wei Ma
Changbo Xia
Hanqing Wang
author_sort Qing Wang
collection DOAJ
description Context Flavones, the key active components in Traditional Chinese Medicine (TCM), have demonstrated antidepressant activity. Given the numerous animal studies conducted, a systematic analysis is essential to provide a valuable reference for future research.Object This study investigated the antidepressant activity of flavones based on animal models and summarized the underlying mechanisms.Methods We systematically searched 7 bibliographic Databases as of August 12, 2023, such as Web of Science, PubMed, China National Knowledge Infrastructure, etc. The meta-analysis was performed using either the random or fixed-effect model, supplemented by trial sequential analysis (TSA). The Grading of Recommendations, Assessment, Development and Evaluations (GRADE) approach was used to assess the quality of evidence.Results A total of 25 studies involving 458 mice were included, identifying five flavones (baicalin, baicalein, apigenin, luteolin, vitexin) with antidepressant activity. Compared to the control group, flavones significantly reduced immobility time in forced swimming and tail suspension tests. Flavones also decreased serum and hippocampal levels of interleukin (IL)-1β and tumor necrosis factor-alpha (TNF-α), reduced nuclear factor kappa B (NF-κB) levels, and increased brain-derived neurotrophic factor (BDNF) levels. Relative to the positive group, flavones raised IL-6, sucrose preference rate, and corticosterone (CORT) levels, with no significant differences in other factors. The TSA showed the efficacy of flavones for treating depression with adequate ‘information size’ for the primary outcome.Conclusions The results demonstrate that flavones exert protective effects against depression in mice, primarily by stimulating neurotrophic factors and modulating inflammatory pathways. These findings emphasize their potential as promising candidates for the development of novel antidepressant therapies.
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spelling doaj-art-8535bc17ac45407595b7ed9cc4fa94b42025-08-20T02:30:27ZengTaylor & Francis GroupPharmaceutical Biology1388-02091744-51162025-12-0163115616910.1080/13880209.2025.2467374Antidepressant activity of flavones from traditional Chinese medicine: a meta-analysisQing Wang0Youyuan Lu1Xue Mi2Caiyan Yang3Wei Ma4Changbo Xia5Hanqing Wang6College of Pharmacy, Ningxia Medical University, Yinchuan, ChinaCollege of Pharmacy, Ningxia Medical University, Yinchuan, ChinaCollege of Pharmacy, Ningxia Medical University, Yinchuan, ChinaDepartment of Pharmacy, The First People’s Hospital of Yinchuan, Yinchuan, ChinaDepartment of Pharmacy, The First People’s Hospital of Yinchuan, Yinchuan, ChinaDepartment of Pharmacy, Central’s Hospital of Xinxiang, Xinxiang, ChinaCollege of Pharmacy, Ningxia Medical University, Yinchuan, ChinaContext Flavones, the key active components in Traditional Chinese Medicine (TCM), have demonstrated antidepressant activity. Given the numerous animal studies conducted, a systematic analysis is essential to provide a valuable reference for future research.Object This study investigated the antidepressant activity of flavones based on animal models and summarized the underlying mechanisms.Methods We systematically searched 7 bibliographic Databases as of August 12, 2023, such as Web of Science, PubMed, China National Knowledge Infrastructure, etc. The meta-analysis was performed using either the random or fixed-effect model, supplemented by trial sequential analysis (TSA). The Grading of Recommendations, Assessment, Development and Evaluations (GRADE) approach was used to assess the quality of evidence.Results A total of 25 studies involving 458 mice were included, identifying five flavones (baicalin, baicalein, apigenin, luteolin, vitexin) with antidepressant activity. Compared to the control group, flavones significantly reduced immobility time in forced swimming and tail suspension tests. Flavones also decreased serum and hippocampal levels of interleukin (IL)-1β and tumor necrosis factor-alpha (TNF-α), reduced nuclear factor kappa B (NF-κB) levels, and increased brain-derived neurotrophic factor (BDNF) levels. Relative to the positive group, flavones raised IL-6, sucrose preference rate, and corticosterone (CORT) levels, with no significant differences in other factors. The TSA showed the efficacy of flavones for treating depression with adequate ‘information size’ for the primary outcome.Conclusions The results demonstrate that flavones exert protective effects against depression in mice, primarily by stimulating neurotrophic factors and modulating inflammatory pathways. These findings emphasize their potential as promising candidates for the development of novel antidepressant therapies.https://www.tandfonline.com/doi/10.1080/13880209.2025.2467374Depressionflavonesanimal studiesmeta-analysismechanisms
spellingShingle Qing Wang
Youyuan Lu
Xue Mi
Caiyan Yang
Wei Ma
Changbo Xia
Hanqing Wang
Antidepressant activity of flavones from traditional Chinese medicine: a meta-analysis
Pharmaceutical Biology
Depression
flavones
animal studies
meta-analysis
mechanisms
title Antidepressant activity of flavones from traditional Chinese medicine: a meta-analysis
title_full Antidepressant activity of flavones from traditional Chinese medicine: a meta-analysis
title_fullStr Antidepressant activity of flavones from traditional Chinese medicine: a meta-analysis
title_full_unstemmed Antidepressant activity of flavones from traditional Chinese medicine: a meta-analysis
title_short Antidepressant activity of flavones from traditional Chinese medicine: a meta-analysis
title_sort antidepressant activity of flavones from traditional chinese medicine a meta analysis
topic Depression
flavones
animal studies
meta-analysis
mechanisms
url https://www.tandfonline.com/doi/10.1080/13880209.2025.2467374
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