Sensitivity of Aspergillus nidulans to the cellulose synthase inhibitor dichlobenil: insights from wall-related genes' expression and ultrastructural hyphal morphologies.

The fungal cell wall constitutes an important target for the development of antifungal drugs, because of its central role in morphogenesis, development and determination of fungal-specific molecular features. Fungal walls are characterized by a network of interconnected glycoproteins and polysacchar...

Full description

Saved in:
Bibliographic Details
Main Authors: Gea Guerriero, Lucia Silvestrini, Michael Obersriebnig, Marco Salerno, Dietmar Pum, Joseph Strauss
Format: Article
Language:English
Published: Public Library of Science (PLoS) 2013-01-01
Series:PLoS ONE
Online Access:https://journals.plos.org/plosone/article/file?id=10.1371/journal.pone.0080038&type=printable
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850125112808833024
author Gea Guerriero
Lucia Silvestrini
Michael Obersriebnig
Marco Salerno
Dietmar Pum
Joseph Strauss
author_facet Gea Guerriero
Lucia Silvestrini
Michael Obersriebnig
Marco Salerno
Dietmar Pum
Joseph Strauss
author_sort Gea Guerriero
collection DOAJ
description The fungal cell wall constitutes an important target for the development of antifungal drugs, because of its central role in morphogenesis, development and determination of fungal-specific molecular features. Fungal walls are characterized by a network of interconnected glycoproteins and polysaccharides, namely α-, β-glucans and chitin. Cell walls promptly and dynamically respond to environmental stimuli by a signaling mechanism, which triggers, among other responses, modulations in wall biosynthetic genes' expression. Despite the absence of cellulose in the wall of the model filamentous fungus Aspergillus nidulans, we found in this study that fungal growth, spore germination and morphology are affected by the addition of the cellulose synthase inhibitor dichlobenil. Expression analysis of selected genes putatively involved in cell wall biosynthesis, carried out at different time points of drug exposure (i.e. 0, 1, 3, 6 and 24 h), revealed increased expression for the putative mixed linkage β-1,3;1,4 glucan synthase celA together with the β-1,3-glucan synthase fksA and the Rho-related GTPase rhoA. We also compared these data with the response to Congo Red, a known plant/fungal drug affecting both chitin and cellulose biosynthesis. The two drugs exerted different effects at the cell wall level, as shown by gene expression analysis and the ultrastructural features observed through atomic force microscopy and scanning electron microscopy. Although the concentration of dichlobenil required to affect growth of A. nidulans is approximately 10-fold higher than that required to inhibit plant cellulose biosynthesis, our work for the first time demonstrates that a cellulose biosynthesis inhibitor affects fungal growth, changes fungal morphology and expression of genes connected to fungal cell wall biosynthesis.
format Article
id doaj-art-8316d2de2d664485baefa3f088b96d6e
institution OA Journals
issn 1932-6203
language English
publishDate 2013-01-01
publisher Public Library of Science (PLoS)
record_format Article
series PLoS ONE
spelling doaj-art-8316d2de2d664485baefa3f088b96d6e2025-08-20T02:34:10ZengPublic Library of Science (PLoS)PLoS ONE1932-62032013-01-01811e8003810.1371/journal.pone.0080038Sensitivity of Aspergillus nidulans to the cellulose synthase inhibitor dichlobenil: insights from wall-related genes' expression and ultrastructural hyphal morphologies.Gea GuerrieroLucia SilvestriniMichael ObersriebnigMarco SalernoDietmar PumJoseph StraussThe fungal cell wall constitutes an important target for the development of antifungal drugs, because of its central role in morphogenesis, development and determination of fungal-specific molecular features. Fungal walls are characterized by a network of interconnected glycoproteins and polysaccharides, namely α-, β-glucans and chitin. Cell walls promptly and dynamically respond to environmental stimuli by a signaling mechanism, which triggers, among other responses, modulations in wall biosynthetic genes' expression. Despite the absence of cellulose in the wall of the model filamentous fungus Aspergillus nidulans, we found in this study that fungal growth, spore germination and morphology are affected by the addition of the cellulose synthase inhibitor dichlobenil. Expression analysis of selected genes putatively involved in cell wall biosynthesis, carried out at different time points of drug exposure (i.e. 0, 1, 3, 6 and 24 h), revealed increased expression for the putative mixed linkage β-1,3;1,4 glucan synthase celA together with the β-1,3-glucan synthase fksA and the Rho-related GTPase rhoA. We also compared these data with the response to Congo Red, a known plant/fungal drug affecting both chitin and cellulose biosynthesis. The two drugs exerted different effects at the cell wall level, as shown by gene expression analysis and the ultrastructural features observed through atomic force microscopy and scanning electron microscopy. Although the concentration of dichlobenil required to affect growth of A. nidulans is approximately 10-fold higher than that required to inhibit plant cellulose biosynthesis, our work for the first time demonstrates that a cellulose biosynthesis inhibitor affects fungal growth, changes fungal morphology and expression of genes connected to fungal cell wall biosynthesis.https://journals.plos.org/plosone/article/file?id=10.1371/journal.pone.0080038&type=printable
spellingShingle Gea Guerriero
Lucia Silvestrini
Michael Obersriebnig
Marco Salerno
Dietmar Pum
Joseph Strauss
Sensitivity of Aspergillus nidulans to the cellulose synthase inhibitor dichlobenil: insights from wall-related genes' expression and ultrastructural hyphal morphologies.
PLoS ONE
title Sensitivity of Aspergillus nidulans to the cellulose synthase inhibitor dichlobenil: insights from wall-related genes' expression and ultrastructural hyphal morphologies.
title_full Sensitivity of Aspergillus nidulans to the cellulose synthase inhibitor dichlobenil: insights from wall-related genes' expression and ultrastructural hyphal morphologies.
title_fullStr Sensitivity of Aspergillus nidulans to the cellulose synthase inhibitor dichlobenil: insights from wall-related genes' expression and ultrastructural hyphal morphologies.
title_full_unstemmed Sensitivity of Aspergillus nidulans to the cellulose synthase inhibitor dichlobenil: insights from wall-related genes' expression and ultrastructural hyphal morphologies.
title_short Sensitivity of Aspergillus nidulans to the cellulose synthase inhibitor dichlobenil: insights from wall-related genes' expression and ultrastructural hyphal morphologies.
title_sort sensitivity of aspergillus nidulans to the cellulose synthase inhibitor dichlobenil insights from wall related genes expression and ultrastructural hyphal morphologies
url https://journals.plos.org/plosone/article/file?id=10.1371/journal.pone.0080038&type=printable
work_keys_str_mv AT geaguerriero sensitivityofaspergillusnidulanstothecellulosesynthaseinhibitordichlobenilinsightsfromwallrelatedgenesexpressionandultrastructuralhyphalmorphologies
AT luciasilvestrini sensitivityofaspergillusnidulanstothecellulosesynthaseinhibitordichlobenilinsightsfromwallrelatedgenesexpressionandultrastructuralhyphalmorphologies
AT michaelobersriebnig sensitivityofaspergillusnidulanstothecellulosesynthaseinhibitordichlobenilinsightsfromwallrelatedgenesexpressionandultrastructuralhyphalmorphologies
AT marcosalerno sensitivityofaspergillusnidulanstothecellulosesynthaseinhibitordichlobenilinsightsfromwallrelatedgenesexpressionandultrastructuralhyphalmorphologies
AT dietmarpum sensitivityofaspergillusnidulanstothecellulosesynthaseinhibitordichlobenilinsightsfromwallrelatedgenesexpressionandultrastructuralhyphalmorphologies
AT josephstrauss sensitivityofaspergillusnidulanstothecellulosesynthaseinhibitordichlobenilinsightsfromwallrelatedgenesexpressionandultrastructuralhyphalmorphologies