<i>Marantodes pumilum</i> var. <i>alata</i> Enhances Fracture Healing Through Gene Regulation in a Postmenopausal Rat Model

<b>Background:</b> <i>Marantodes pumilum</i> var. <i>alata</i> (<i>MPva</i>) has been reported to promote fracture repair. This study investigates the role of <i>MPva</i> leaf extract on biochemical markers and bone-repair genes in a postme...

Full description

Saved in:
Bibliographic Details
Main Authors: Tijjani Rabiu Giaze, Norazlina Mohamed, Syed Alhafiz Syed Hashim, Ahmad Nazrun Shuid, Ima Nirwana Soelaiman, Norliza Muhammad, Fadhlullah Zuhair Jafar Sidik, Jamia Azdina Jamal
Format: Article
Language:English
Published: MDPI AG 2025-05-01
Series:Pharmaceuticals
Subjects:
Online Access:https://www.mdpi.com/1424-8247/18/5/736
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850126912510230528
author Tijjani Rabiu Giaze
Norazlina Mohamed
Syed Alhafiz Syed Hashim
Ahmad Nazrun Shuid
Ima Nirwana Soelaiman
Norliza Muhammad
Fadhlullah Zuhair Jafar Sidik
Jamia Azdina Jamal
author_facet Tijjani Rabiu Giaze
Norazlina Mohamed
Syed Alhafiz Syed Hashim
Ahmad Nazrun Shuid
Ima Nirwana Soelaiman
Norliza Muhammad
Fadhlullah Zuhair Jafar Sidik
Jamia Azdina Jamal
author_sort Tijjani Rabiu Giaze
collection DOAJ
description <b>Background:</b> <i>Marantodes pumilum</i> var. <i>alata</i> (<i>MPva</i>) has been reported to promote fracture repair. This study investigates the role of <i>MPva</i> leaf extract on biochemical markers and bone-repair genes in a postmenopausal rat model to understand its fracture-healing properties. <b>Methods</b>: Thirty female Sprague Dawley rats were grouped into sham-operated (Sham), ovariectomized control (OVXC), estrogen treatment (ERT), and plant treatment (MPv20 and MPv100) groups. After ovariectomy, the right tibiae of rats were fractured. The ERT group was treated with 64.5 μg/kg/day of estrogen, while the MPv20 and MPv100 groups received 20 and 100 mg/kg/day doses of <i>MPva</i> leaf extract, respectively, for 8 weeks. Sham and OVXC acted as untreated controls. Blood samples collected before and after treatment were assayed for pro-inflammatory cytokines (IL-6 and TNF-α), while bone samples were assayed for bone-turnover markers: osteocalcin and pyridinoline, oxidative-status markers (GPx, SOD, and MDA), and bone-repair genes (<i>Bglap</i>, <i>Spp1</i>, <i>Dkk1</i>, <i>Igf1</i>, <i>Tnfsf11</i>, and <i>Fgf23</i>). <b>Results</b>: IL-6, GPx, and SOD levels were significantly increased in both MPv groups (<i>p</i> < 0.05). <i>IGF1</i> was significantly upregulated in both MPv groups, while <i>Tnfsf11</i> was downregulated in the MPv20 group (<i>p</i> < 0.05). <b>Conclusions</b>: <i>MPva</i> leaf extract may promote bone repair by stimulating pro-inflammatory and antioxidant responses, which are associated with its regulation of <i>Igf1</i> and <i>Tnfsf11 genes</i>.
format Article
id doaj-art-7d41a912807d4e02840b870aced0c2ad
institution OA Journals
issn 1424-8247
language English
publishDate 2025-05-01
publisher MDPI AG
record_format Article
series Pharmaceuticals
spelling doaj-art-7d41a912807d4e02840b870aced0c2ad2025-08-20T02:33:48ZengMDPI AGPharmaceuticals1424-82472025-05-0118573610.3390/ph18050736<i>Marantodes pumilum</i> var. <i>alata</i> Enhances Fracture Healing Through Gene Regulation in a Postmenopausal Rat ModelTijjani Rabiu Giaze0Norazlina Mohamed1Syed Alhafiz Syed Hashim2Ahmad Nazrun Shuid3Ima Nirwana Soelaiman4Norliza Muhammad5Fadhlullah Zuhair Jafar Sidik6Jamia Azdina Jamal7Department of Pharmacology, Faculty of Medicine, Universiti Kebangsaan Malaysia, Cheras, Kuala Lumpur 56000, Selangor, MalaysiaDepartment of Pharmacology, Faculty of Medicine, Universiti Kebangsaan Malaysia, Cheras, Kuala Lumpur 56000, Selangor, MalaysiaDepartment of Pharmacology, Faculty of Medicine, Universiti Kebangsaan Malaysia, Cheras, Kuala Lumpur 56000, Selangor, MalaysiaDepartment of Pharmacology, Faculty of Medicine, Universiti Teknologi Mara, Sungai Buloh 47000, Selangor, MalaysiaDepartment of Pharmacology, Faculty of Medicine, Universiti Kebangsaan Malaysia, Cheras, Kuala Lumpur 56000, Selangor, MalaysiaDepartment of Pharmacology, Faculty of Medicine, Universiti Kebangsaan Malaysia, Cheras, Kuala Lumpur 56000, Selangor, MalaysiaFaculty of Pharmacy, Universiti Kebangsaan Malaysia, Cheras, Kuala Lumpur 56000, Selangor, MalaysiaFaculty of Pharmacy, Universiti Kebangsaan Malaysia, Cheras, Kuala Lumpur 56000, Selangor, Malaysia<b>Background:</b> <i>Marantodes pumilum</i> var. <i>alata</i> (<i>MPva</i>) has been reported to promote fracture repair. This study investigates the role of <i>MPva</i> leaf extract on biochemical markers and bone-repair genes in a postmenopausal rat model to understand its fracture-healing properties. <b>Methods</b>: Thirty female Sprague Dawley rats were grouped into sham-operated (Sham), ovariectomized control (OVXC), estrogen treatment (ERT), and plant treatment (MPv20 and MPv100) groups. After ovariectomy, the right tibiae of rats were fractured. The ERT group was treated with 64.5 μg/kg/day of estrogen, while the MPv20 and MPv100 groups received 20 and 100 mg/kg/day doses of <i>MPva</i> leaf extract, respectively, for 8 weeks. Sham and OVXC acted as untreated controls. Blood samples collected before and after treatment were assayed for pro-inflammatory cytokines (IL-6 and TNF-α), while bone samples were assayed for bone-turnover markers: osteocalcin and pyridinoline, oxidative-status markers (GPx, SOD, and MDA), and bone-repair genes (<i>Bglap</i>, <i>Spp1</i>, <i>Dkk1</i>, <i>Igf1</i>, <i>Tnfsf11</i>, and <i>Fgf23</i>). <b>Results</b>: IL-6, GPx, and SOD levels were significantly increased in both MPv groups (<i>p</i> < 0.05). <i>IGF1</i> was significantly upregulated in both MPv groups, while <i>Tnfsf11</i> was downregulated in the MPv20 group (<i>p</i> < 0.05). <b>Conclusions</b>: <i>MPva</i> leaf extract may promote bone repair by stimulating pro-inflammatory and antioxidant responses, which are associated with its regulation of <i>Igf1</i> and <i>Tnfsf11 genes</i>.https://www.mdpi.com/1424-8247/18/5/736fracturegene expression<i>Marantodes pumilum</i>osteoporosisovariectomized rats
spellingShingle Tijjani Rabiu Giaze
Norazlina Mohamed
Syed Alhafiz Syed Hashim
Ahmad Nazrun Shuid
Ima Nirwana Soelaiman
Norliza Muhammad
Fadhlullah Zuhair Jafar Sidik
Jamia Azdina Jamal
<i>Marantodes pumilum</i> var. <i>alata</i> Enhances Fracture Healing Through Gene Regulation in a Postmenopausal Rat Model
Pharmaceuticals
fracture
gene expression
<i>Marantodes pumilum</i>
osteoporosis
ovariectomized rats
title <i>Marantodes pumilum</i> var. <i>alata</i> Enhances Fracture Healing Through Gene Regulation in a Postmenopausal Rat Model
title_full <i>Marantodes pumilum</i> var. <i>alata</i> Enhances Fracture Healing Through Gene Regulation in a Postmenopausal Rat Model
title_fullStr <i>Marantodes pumilum</i> var. <i>alata</i> Enhances Fracture Healing Through Gene Regulation in a Postmenopausal Rat Model
title_full_unstemmed <i>Marantodes pumilum</i> var. <i>alata</i> Enhances Fracture Healing Through Gene Regulation in a Postmenopausal Rat Model
title_short <i>Marantodes pumilum</i> var. <i>alata</i> Enhances Fracture Healing Through Gene Regulation in a Postmenopausal Rat Model
title_sort i marantodes pumilum i var i alata i enhances fracture healing through gene regulation in a postmenopausal rat model
topic fracture
gene expression
<i>Marantodes pumilum</i>
osteoporosis
ovariectomized rats
url https://www.mdpi.com/1424-8247/18/5/736
work_keys_str_mv AT tijjanirabiugiaze imarantodespumilumivarialataienhancesfracturehealingthroughgeneregulationinapostmenopausalratmodel
AT norazlinamohamed imarantodespumilumivarialataienhancesfracturehealingthroughgeneregulationinapostmenopausalratmodel
AT syedalhafizsyedhashim imarantodespumilumivarialataienhancesfracturehealingthroughgeneregulationinapostmenopausalratmodel
AT ahmadnazrunshuid imarantodespumilumivarialataienhancesfracturehealingthroughgeneregulationinapostmenopausalratmodel
AT imanirwanasoelaiman imarantodespumilumivarialataienhancesfracturehealingthroughgeneregulationinapostmenopausalratmodel
AT norlizamuhammad imarantodespumilumivarialataienhancesfracturehealingthroughgeneregulationinapostmenopausalratmodel
AT fadhlullahzuhairjafarsidik imarantodespumilumivarialataienhancesfracturehealingthroughgeneregulationinapostmenopausalratmodel
AT jamiaazdinajamal imarantodespumilumivarialataienhancesfracturehealingthroughgeneregulationinapostmenopausalratmodel