A Physical-Chemical Study of the Interference of Ceftriaxone Antibiotic with Copper Chloride Salt

The nano-CuCl2.2H2O salt was prepared by the ball milling method. The association parameters for bulk and nano-CuCl2 salts in H2O are estimated at different temperatures using the conductivity method by applying the Fuoss–Shedlovsky equation and it was higher for nano-CuCl2 than bulk CuCl2 salt. The...

Full description

Saved in:
Bibliographic Details
Main Authors: Elsayed M. AbouElleef, Mowafak M. Mahrouka, Sherine E. Salem
Format: Article
Language:English
Published: Wiley 2021-01-01
Series:Bioinorganic Chemistry and Applications
Online Access:http://dx.doi.org/10.1155/2021/4018843
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850220232648425472
author Elsayed M. AbouElleef
Mowafak M. Mahrouka
Sherine E. Salem
author_facet Elsayed M. AbouElleef
Mowafak M. Mahrouka
Sherine E. Salem
author_sort Elsayed M. AbouElleef
collection DOAJ
description The nano-CuCl2.2H2O salt was prepared by the ball milling method. The association parameters for bulk and nano-CuCl2 salts in H2O are estimated at different temperatures using the conductivity method by applying the Fuoss–Shedlovsky equation and it was higher for nano-CuCl2 than bulk CuCl2 salt. The interaction between the cation (Cu2+) and ligand (ceftriaxone) in H2O was determined also by the conductometric method. Two stoichiometric complexes 1/2 and 1/1 (M/L) are estimated and follow the order Kf (1/1) > Kf (1 : 2) and ∆Gf (1/1) > ∆Gf (1/2) for (M : L) (in negative values) indicate the favorable of formation of (1/1) complex compared to the (1 : 2) complex. The Gibbs free energies change was increased in negative signs with increasing the temperature. The antimicrobial activities of CFT, bulk Cu-CFT complex, and nano-Cu-CFT complex were studied on LB agar by the disc diffusion technique against clinical isolates of gram-negative bacteria (Klebsiella pneumonia and Pseudomonas aeruginosa) and Fungi (Candida albicans). It was observed that (CFT) has a higher zone of inhibition and antibacterial activity than that of bulk and nano-Cu-CFT complexes in Klebsiella pneumonia and Pseudomonas aeruginosa (gram-negative bacteria). The nano-Cu-CFT complex showed a higher clear zone of inhibition and antifungal activity against candida than bulk Cu-CFT complex while the absence of the inhibition zone in CFT, so nano-Cu-CFT complex, can be used as an antifungal drug.
format Article
id doaj-art-7823219a787b451aa4012d3917a665be
institution OA Journals
issn 1565-3633
1687-479X
language English
publishDate 2021-01-01
publisher Wiley
record_format Article
series Bioinorganic Chemistry and Applications
spelling doaj-art-7823219a787b451aa4012d3917a665be2025-08-20T02:07:08ZengWileyBioinorganic Chemistry and Applications1565-36331687-479X2021-01-01202110.1155/2021/40188434018843A Physical-Chemical Study of the Interference of Ceftriaxone Antibiotic with Copper Chloride SaltElsayed M. AbouElleef0Mowafak M. Mahrouka1Sherine E. Salem2Chemistry Department, Faculty of Arts and Science, Rafha Northern Border University, 91911 Rafha, Saudi ArabiaChemistry Department, Faculty of Arts and Science, Rafha Northern Border University, 91911 Rafha, Saudi ArabiaChemistry Department, Faculty of Science, Mansoura University, 35516 Mansoura, EgyptThe nano-CuCl2.2H2O salt was prepared by the ball milling method. The association parameters for bulk and nano-CuCl2 salts in H2O are estimated at different temperatures using the conductivity method by applying the Fuoss–Shedlovsky equation and it was higher for nano-CuCl2 than bulk CuCl2 salt. The interaction between the cation (Cu2+) and ligand (ceftriaxone) in H2O was determined also by the conductometric method. Two stoichiometric complexes 1/2 and 1/1 (M/L) are estimated and follow the order Kf (1/1) > Kf (1 : 2) and ∆Gf (1/1) > ∆Gf (1/2) for (M : L) (in negative values) indicate the favorable of formation of (1/1) complex compared to the (1 : 2) complex. The Gibbs free energies change was increased in negative signs with increasing the temperature. The antimicrobial activities of CFT, bulk Cu-CFT complex, and nano-Cu-CFT complex were studied on LB agar by the disc diffusion technique against clinical isolates of gram-negative bacteria (Klebsiella pneumonia and Pseudomonas aeruginosa) and Fungi (Candida albicans). It was observed that (CFT) has a higher zone of inhibition and antibacterial activity than that of bulk and nano-Cu-CFT complexes in Klebsiella pneumonia and Pseudomonas aeruginosa (gram-negative bacteria). The nano-Cu-CFT complex showed a higher clear zone of inhibition and antifungal activity against candida than bulk Cu-CFT complex while the absence of the inhibition zone in CFT, so nano-Cu-CFT complex, can be used as an antifungal drug.http://dx.doi.org/10.1155/2021/4018843
spellingShingle Elsayed M. AbouElleef
Mowafak M. Mahrouka
Sherine E. Salem
A Physical-Chemical Study of the Interference of Ceftriaxone Antibiotic with Copper Chloride Salt
Bioinorganic Chemistry and Applications
title A Physical-Chemical Study of the Interference of Ceftriaxone Antibiotic with Copper Chloride Salt
title_full A Physical-Chemical Study of the Interference of Ceftriaxone Antibiotic with Copper Chloride Salt
title_fullStr A Physical-Chemical Study of the Interference of Ceftriaxone Antibiotic with Copper Chloride Salt
title_full_unstemmed A Physical-Chemical Study of the Interference of Ceftriaxone Antibiotic with Copper Chloride Salt
title_short A Physical-Chemical Study of the Interference of Ceftriaxone Antibiotic with Copper Chloride Salt
title_sort physical chemical study of the interference of ceftriaxone antibiotic with copper chloride salt
url http://dx.doi.org/10.1155/2021/4018843
work_keys_str_mv AT elsayedmabouelleef aphysicalchemicalstudyoftheinterferenceofceftriaxoneantibioticwithcopperchloridesalt
AT mowafakmmahrouka aphysicalchemicalstudyoftheinterferenceofceftriaxoneantibioticwithcopperchloridesalt
AT sherineesalem aphysicalchemicalstudyoftheinterferenceofceftriaxoneantibioticwithcopperchloridesalt
AT elsayedmabouelleef physicalchemicalstudyoftheinterferenceofceftriaxoneantibioticwithcopperchloridesalt
AT mowafakmmahrouka physicalchemicalstudyoftheinterferenceofceftriaxoneantibioticwithcopperchloridesalt
AT sherineesalem physicalchemicalstudyoftheinterferenceofceftriaxoneantibioticwithcopperchloridesalt