Synthesis of Novel Schiff Base and Azetidinone Derivatives and their Antibacterial Activity

A series of Compound 4-(2᾽-hydroxy-3᾽-chloro-5᾽-ethyl phen-1᾽-yl)-1-(4᾽-tolyl)-3-chloro-2-azetidinone 4a-j have been prepared by the reaction of 2 -hydroxy-3 -chloro-5 -ethyl-N-(p-tolyl)-chalconimines 3a-j with chloroacetyl chloride in the presence of triethylamine. The Schiff base derivatives 3a-j...

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Main Authors: Kamal Vashi, H. B. Naik
Format: Article
Language:English
Published: Wiley 2004-01-01
Series:E-Journal of Chemistry
Online Access:http://dx.doi.org/10.1155/2004/158924
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author Kamal Vashi
H. B. Naik
author_facet Kamal Vashi
H. B. Naik
author_sort Kamal Vashi
collection DOAJ
description A series of Compound 4-(2᾽-hydroxy-3᾽-chloro-5᾽-ethyl phen-1᾽-yl)-1-(4᾽-tolyl)-3-chloro-2-azetidinone 4a-j have been prepared by the reaction of 2 -hydroxy-3 -chloro-5 -ethyl-N-(p-tolyl)-chalconimines 3a-j with chloroacetyl chloride in the presence of triethylamine. The Schiff base derivatives 3a-j has been prepared by the condensation of different substituted chalone derivatives 1 with p-toluidine 2. The synthesized compounds were screened for their antibacterial activity against Staphylococcus aureus and Escherichia coli.
format Article
id doaj-art-77f37d2e6add484a9b28f7ea890d477f
institution Kabale University
issn 0973-4945
2090-9810
language English
publishDate 2004-01-01
publisher Wiley
record_format Article
series E-Journal of Chemistry
spelling doaj-art-77f37d2e6add484a9b28f7ea890d477f2025-08-20T03:35:36ZengWileyE-Journal of Chemistry0973-49452090-98102004-01-011527227510.1155/2004/158924Synthesis of Novel Schiff Base and Azetidinone Derivatives and their Antibacterial ActivityKamal Vashi0H. B. Naik1Department of Chemistry, Veer Narmad South Gujarat University, Surat 395007, IndiaDepartment of Chemistry, Veer Narmad South Gujarat University, Surat 395007, IndiaA series of Compound 4-(2᾽-hydroxy-3᾽-chloro-5᾽-ethyl phen-1᾽-yl)-1-(4᾽-tolyl)-3-chloro-2-azetidinone 4a-j have been prepared by the reaction of 2 -hydroxy-3 -chloro-5 -ethyl-N-(p-tolyl)-chalconimines 3a-j with chloroacetyl chloride in the presence of triethylamine. The Schiff base derivatives 3a-j has been prepared by the condensation of different substituted chalone derivatives 1 with p-toluidine 2. The synthesized compounds were screened for their antibacterial activity against Staphylococcus aureus and Escherichia coli.http://dx.doi.org/10.1155/2004/158924
spellingShingle Kamal Vashi
H. B. Naik
Synthesis of Novel Schiff Base and Azetidinone Derivatives and their Antibacterial Activity
E-Journal of Chemistry
title Synthesis of Novel Schiff Base and Azetidinone Derivatives and their Antibacterial Activity
title_full Synthesis of Novel Schiff Base and Azetidinone Derivatives and their Antibacterial Activity
title_fullStr Synthesis of Novel Schiff Base and Azetidinone Derivatives and their Antibacterial Activity
title_full_unstemmed Synthesis of Novel Schiff Base and Azetidinone Derivatives and their Antibacterial Activity
title_short Synthesis of Novel Schiff Base and Azetidinone Derivatives and their Antibacterial Activity
title_sort synthesis of novel schiff base and azetidinone derivatives and their antibacterial activity
url http://dx.doi.org/10.1155/2004/158924
work_keys_str_mv AT kamalvashi synthesisofnovelschiffbaseandazetidinonederivativesandtheirantibacterialactivity
AT hbnaik synthesisofnovelschiffbaseandazetidinonederivativesandtheirantibacterialactivity