Effect of Chronic Administration of <i>Justicia secunda</i> Vahl in Mice Diabetized with Streptozotocin

Certain pharmacological properties of the methanolic extract of <i>Justicia secunda</i> Vahl leaves (<i>Acanthaceae</i>) were evaluated in Streptozotocin (STZ)-treated albino mice to confirm whether it could be considered an alternative candidate for the treatment of diabetes...

Full description

Saved in:
Bibliographic Details
Main Authors: Tomás Fregoso-Aguilar, Perla Xóchitl Escamilla-Ramírez, Dulce E. Nicolás-Álvarez, Jorge Alberto Mendoza-Pérez, Eduardo Osiris Madrigal-Santillán, Judith Margarita Tirado-Lule, Elda Victoria Rodríguez-Negrete, Eduardo Madrigal-Bujaidar, Isela Álvarez-González, Gabriela Ibáñez-Cervantes, Ángel Morales-González, José A. Morales-Gonzalez
Format: Article
Language:English
Published: MDPI AG 2025-06-01
Series:Diabetology
Subjects:
Online Access:https://www.mdpi.com/2673-4540/6/6/56
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849431973066440704
author Tomás Fregoso-Aguilar
Perla Xóchitl Escamilla-Ramírez
Dulce E. Nicolás-Álvarez
Jorge Alberto Mendoza-Pérez
Eduardo Osiris Madrigal-Santillán
Judith Margarita Tirado-Lule
Elda Victoria Rodríguez-Negrete
Eduardo Madrigal-Bujaidar
Isela Álvarez-González
Gabriela Ibáñez-Cervantes
Ángel Morales-González
José A. Morales-Gonzalez
author_facet Tomás Fregoso-Aguilar
Perla Xóchitl Escamilla-Ramírez
Dulce E. Nicolás-Álvarez
Jorge Alberto Mendoza-Pérez
Eduardo Osiris Madrigal-Santillán
Judith Margarita Tirado-Lule
Elda Victoria Rodríguez-Negrete
Eduardo Madrigal-Bujaidar
Isela Álvarez-González
Gabriela Ibáñez-Cervantes
Ángel Morales-González
José A. Morales-Gonzalez
author_sort Tomás Fregoso-Aguilar
collection DOAJ
description Certain pharmacological properties of the methanolic extract of <i>Justicia secunda</i> Vahl leaves (<i>Acanthaceae</i>) were evaluated in Streptozotocin (STZ)-treated albino mice to confirm whether it could be considered an alternative candidate for the treatment of diabetes. Using qualitative phytochemistry, alkaloids, flavonoids, and tannins were detected. In an in vitro DPPH antioxidant activity test, high extract concentrations inhibited the radical by 90% during the first minutes of the reaction. The extract presented a slight genoprotective effect on mouse peripheral blood during the last days of the micronucleus test. Oral administration of the extract at a high dose every two days for 6 weeks caused a hypoglycemic effect in STZ-treated mice, protection against weight loss, and decreased blood triglyceride levels from week 3 of treatment. These effects could be mediated by the antioxidant activity of the detected metabolites and, perhaps, by an inhibitory effect on intestinal α-glucosidase. This renders <i>J. secunda</i> a good candidate for the long-term alternative treatment of diabetes without abandoning allopathic therapy.
format Article
id doaj-art-76941518cc0b4108bfdcaf39e989cd0f
institution Kabale University
issn 2673-4540
language English
publishDate 2025-06-01
publisher MDPI AG
record_format Article
series Diabetology
spelling doaj-art-76941518cc0b4108bfdcaf39e989cd0f2025-08-20T03:27:28ZengMDPI AGDiabetology2673-45402025-06-01665610.3390/diabetology6060056Effect of Chronic Administration of <i>Justicia secunda</i> Vahl in Mice Diabetized with StreptozotocinTomás Fregoso-Aguilar0Perla Xóchitl Escamilla-Ramírez1Dulce E. Nicolás-Álvarez2Jorge Alberto Mendoza-Pérez3Eduardo Osiris Madrigal-Santillán4Judith Margarita Tirado-Lule5Elda Victoria Rodríguez-Negrete6Eduardo Madrigal-Bujaidar7Isela Álvarez-González8Gabriela Ibáñez-Cervantes9Ángel Morales-González10José A. Morales-Gonzalez11Escuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional, Departamento de Fisiología, Av. Wilfrido Massieu s/n, Col. Nueva Industrial Vallejo, Alcaldía Gustavo A. Madero, Ciudad de México C.P. 07700, MexicoEscuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional, Departamento de Fisiología, Av. Wilfrido Massieu s/n, Col. Nueva Industrial Vallejo, Alcaldía Gustavo A. Madero, Ciudad de México C.P. 07700, MexicoEscuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional, Departamento de Fisiología, Av. Wilfrido Massieu s/n, Col. Nueva Industrial Vallejo, Alcaldía Gustavo A. Madero, Ciudad de México C.P. 07700, MexicoEscuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional, Departamento de Ingeniería en Sistemas Ambientales, Av. Wilfrido Massieu s/n, Col. Nueva Industrial Vallejo, Alcaldía Gustavo A. Madero, Ciudad de México C.P. 07700, MexicoLaboratorio de Medicina de Conservación, Escuela Superior de Medicina, Instituto Politécnico Nacional, Plan de San Luis y Díaz Mirón, Col. Casco de Santo Tomás, Alcaldía Miguel Hidalgo, Ciudad de México C.P. 11340, MexicoEscuela Superior de Cómputo, Instituto Politécnico Nacional, Unidad Profesional “A. López Mateos”, Ciudad de México C.P. 07738, MexicoLaboratorio de Medicina de Conservación, Escuela Superior de Medicina, Instituto Politécnico Nacional, Plan de San Luis y Díaz Mirón, Col. Casco de Santo Tomás, Alcaldía Miguel Hidalgo, Ciudad de México C.P. 11340, MexicoLaboratorio de Genética, Escuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional, Av. Wilfrido Massieu s/n, Zacatenco, Gustavo A. Madero, Mexico City C.P. 07738, MexicoLaboratorio de Genética, Escuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional, Av. Wilfrido Massieu s/n, Zacatenco, Gustavo A. Madero, Mexico City C.P. 07738, MexicoSección de Estudios de Posgrado e Investigación, Escuela Superior de Medicina, Instituto Politécnico Nacional, Plan de San Luis y Díaz Mirón, Col. Casco de Santo Tomás, Alcaldía Miguel Hidalgo, Ciudad de México, C.P. 11340, MexicoEscuela Superior de Cómputo, Instituto Politécnico Nacional, Unidad Profesional “A. López Mateos”, Ciudad de México C.P. 07738, MexicoLaboratorio de Medicina de Conservación, Escuela Superior de Medicina, Instituto Politécnico Nacional, Plan de San Luis y Díaz Mirón, Col. Casco de Santo Tomás, Alcaldía Miguel Hidalgo, Ciudad de México C.P. 11340, MexicoCertain pharmacological properties of the methanolic extract of <i>Justicia secunda</i> Vahl leaves (<i>Acanthaceae</i>) were evaluated in Streptozotocin (STZ)-treated albino mice to confirm whether it could be considered an alternative candidate for the treatment of diabetes. Using qualitative phytochemistry, alkaloids, flavonoids, and tannins were detected. In an in vitro DPPH antioxidant activity test, high extract concentrations inhibited the radical by 90% during the first minutes of the reaction. The extract presented a slight genoprotective effect on mouse peripheral blood during the last days of the micronucleus test. Oral administration of the extract at a high dose every two days for 6 weeks caused a hypoglycemic effect in STZ-treated mice, protection against weight loss, and decreased blood triglyceride levels from week 3 of treatment. These effects could be mediated by the antioxidant activity of the detected metabolites and, perhaps, by an inhibitory effect on intestinal α-glucosidase. This renders <i>J. secunda</i> a good candidate for the long-term alternative treatment of diabetes without abandoning allopathic therapy.https://www.mdpi.com/2673-4540/6/6/56diabetesmice<i>Justicia secunda</i>antioxidanthypoglycemicgenoprotective effect
spellingShingle Tomás Fregoso-Aguilar
Perla Xóchitl Escamilla-Ramírez
Dulce E. Nicolás-Álvarez
Jorge Alberto Mendoza-Pérez
Eduardo Osiris Madrigal-Santillán
Judith Margarita Tirado-Lule
Elda Victoria Rodríguez-Negrete
Eduardo Madrigal-Bujaidar
Isela Álvarez-González
Gabriela Ibáñez-Cervantes
Ángel Morales-González
José A. Morales-Gonzalez
Effect of Chronic Administration of <i>Justicia secunda</i> Vahl in Mice Diabetized with Streptozotocin
Diabetology
diabetes
mice
<i>Justicia secunda</i>
antioxidant
hypoglycemic
genoprotective effect
title Effect of Chronic Administration of <i>Justicia secunda</i> Vahl in Mice Diabetized with Streptozotocin
title_full Effect of Chronic Administration of <i>Justicia secunda</i> Vahl in Mice Diabetized with Streptozotocin
title_fullStr Effect of Chronic Administration of <i>Justicia secunda</i> Vahl in Mice Diabetized with Streptozotocin
title_full_unstemmed Effect of Chronic Administration of <i>Justicia secunda</i> Vahl in Mice Diabetized with Streptozotocin
title_short Effect of Chronic Administration of <i>Justicia secunda</i> Vahl in Mice Diabetized with Streptozotocin
title_sort effect of chronic administration of i justicia secunda i vahl in mice diabetized with streptozotocin
topic diabetes
mice
<i>Justicia secunda</i>
antioxidant
hypoglycemic
genoprotective effect
url https://www.mdpi.com/2673-4540/6/6/56
work_keys_str_mv AT tomasfregosoaguilar effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin
AT perlaxochitlescamillaramirez effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin
AT dulceenicolasalvarez effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin
AT jorgealbertomendozaperez effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin
AT eduardoosirismadrigalsantillan effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin
AT judithmargaritatiradolule effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin
AT eldavictoriarodrigueznegrete effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin
AT eduardomadrigalbujaidar effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin
AT iselaalvarezgonzalez effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin
AT gabrielaibanezcervantes effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin
AT angelmoralesgonzalez effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin
AT joseamoralesgonzalez effectofchronicadministrationofijusticiasecundaivahlinmicediabetizedwithstreptozotocin