Methadone and Buprenorphine as Medication for Addiction Treatment Diversely Affect Inflammation and Craving Depending on Their Doses

Buprenorphine and methadone are widely used as medication for addiction treatment (MAT) in patients with opioid use disorders. However, there is no compelling evidence of their impact on the immune–endocrine response. Therefore, the aim of this study was to examine the effects of the aforementioned...

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Main Authors: Christonikos Leventelis, Aristidis S. Veskoukis, Andrea Paola Rojas Gil, Panagiotis Papadopoulos, Maria Garderi, Asimina Angeli, Antzouletta Kampitsi, Maria Tsironi
Format: Article
Language:English
Published: MDPI AG 2025-03-01
Series:Pharmacy
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Online Access:https://www.mdpi.com/2226-4787/13/2/40
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author Christonikos Leventelis
Aristidis S. Veskoukis
Andrea Paola Rojas Gil
Panagiotis Papadopoulos
Maria Garderi
Asimina Angeli
Antzouletta Kampitsi
Maria Tsironi
author_facet Christonikos Leventelis
Aristidis S. Veskoukis
Andrea Paola Rojas Gil
Panagiotis Papadopoulos
Maria Garderi
Asimina Angeli
Antzouletta Kampitsi
Maria Tsironi
author_sort Christonikos Leventelis
collection DOAJ
description Buprenorphine and methadone are widely used as medication for addiction treatment (MAT) in patients with opioid use disorders. However, there is no compelling evidence of their impact on the immune–endocrine response. Therefore, the aim of this study was to examine the effects of the aforementioned medications on craving and on biomarkers of inflammation and cortisol, approaching the dose issue concurrently. Sixty-six patients (thirty-four under methadone and thirty-two under buprenorphine) who had just entered a MAT program and were stabilized with the suitable administered doses after a two-week process were divided into four groups based on medication dose (i.e., methadone high dose, buprenorphine high dose, methadone medium dose, and buprenorphine medium dose). The heroin craving questionnaire for craving assessment was completed, and the blood biomarkers were measured on Days 1 and 180. According to the results, high doses of both medications were accompanied by low levels of craving, cortisol, and inflammation on Day 1, and no alterations were observed on Day 180. On the contrary, medium doses reduced the tested psychosocial and biochemical parameters in terms of time, indicating a positive action for the patients. Concludingly, modifications in MAT doses are needed soon after the stabilization process to prevent inflammation and avoid relapse, thus helping opioid-addicted patients toward rehabilitation.
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spelling doaj-art-73e0555d19a2465a8ad5258bc93bd41e2025-08-20T02:18:20ZengMDPI AGPharmacy2226-47872025-03-011324010.3390/pharmacy13020040Methadone and Buprenorphine as Medication for Addiction Treatment Diversely Affect Inflammation and Craving Depending on Their DosesChristonikos Leventelis0Aristidis S. Veskoukis1Andrea Paola Rojas Gil2Panagiotis Papadopoulos3Maria Garderi4Asimina Angeli5Antzouletta Kampitsi6Maria Tsironi7Department of Nursing, University of Peloponnese, 22100 Tripoli, GreeceDepartment of Nutrition and Dietetics, University of Thessaly, Argonafton 1, 42132 Trikala, GreeceDepartment of Nursing, University of Peloponnese, 22100 Tripoli, GreeceOrganization Against Drugs, 10433 Athens, GreeceOrganization Against Drugs, 10433 Athens, GreeceOrganization Against Drugs, 10433 Athens, GreeceGeneral Anticancer Hospital “Agios Savvas”, 11522 Athens, GreeceDepartment of Nursing, University of Peloponnese, 22100 Tripoli, GreeceBuprenorphine and methadone are widely used as medication for addiction treatment (MAT) in patients with opioid use disorders. However, there is no compelling evidence of their impact on the immune–endocrine response. Therefore, the aim of this study was to examine the effects of the aforementioned medications on craving and on biomarkers of inflammation and cortisol, approaching the dose issue concurrently. Sixty-six patients (thirty-four under methadone and thirty-two under buprenorphine) who had just entered a MAT program and were stabilized with the suitable administered doses after a two-week process were divided into four groups based on medication dose (i.e., methadone high dose, buprenorphine high dose, methadone medium dose, and buprenorphine medium dose). The heroin craving questionnaire for craving assessment was completed, and the blood biomarkers were measured on Days 1 and 180. According to the results, high doses of both medications were accompanied by low levels of craving, cortisol, and inflammation on Day 1, and no alterations were observed on Day 180. On the contrary, medium doses reduced the tested psychosocial and biochemical parameters in terms of time, indicating a positive action for the patients. Concludingly, modifications in MAT doses are needed soon after the stabilization process to prevent inflammation and avoid relapse, thus helping opioid-addicted patients toward rehabilitation.https://www.mdpi.com/2226-4787/13/2/40methadonebuprenorphineopioid maintenance treatmentinflammationgrowth factorscytokines
spellingShingle Christonikos Leventelis
Aristidis S. Veskoukis
Andrea Paola Rojas Gil
Panagiotis Papadopoulos
Maria Garderi
Asimina Angeli
Antzouletta Kampitsi
Maria Tsironi
Methadone and Buprenorphine as Medication for Addiction Treatment Diversely Affect Inflammation and Craving Depending on Their Doses
Pharmacy
methadone
buprenorphine
opioid maintenance treatment
inflammation
growth factors
cytokines
title Methadone and Buprenorphine as Medication for Addiction Treatment Diversely Affect Inflammation and Craving Depending on Their Doses
title_full Methadone and Buprenorphine as Medication for Addiction Treatment Diversely Affect Inflammation and Craving Depending on Their Doses
title_fullStr Methadone and Buprenorphine as Medication for Addiction Treatment Diversely Affect Inflammation and Craving Depending on Their Doses
title_full_unstemmed Methadone and Buprenorphine as Medication for Addiction Treatment Diversely Affect Inflammation and Craving Depending on Their Doses
title_short Methadone and Buprenorphine as Medication for Addiction Treatment Diversely Affect Inflammation and Craving Depending on Their Doses
title_sort methadone and buprenorphine as medication for addiction treatment diversely affect inflammation and craving depending on their doses
topic methadone
buprenorphine
opioid maintenance treatment
inflammation
growth factors
cytokines
url https://www.mdpi.com/2226-4787/13/2/40
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