Quercetin: A Natural Ally in Combating Breast Cancer

Zi-Yun Wu, Kang-Yu Qiu, Yan-Jun Gai, Jia-Hui Wu, Bo-Xuan Zhou, Qing-Feng Shi Department of Breast Disease Center, The First Affiliated Hospital of Nanchang University, The First Clinical Medical College of Nanchang University, Jiangxi Medical College, Nanchang, 330006, People’s Republic of ChinaCorr...

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Main Authors: Wu ZY, Qiu KY, Gai YJ, Wu JH, Zhou BX, Shi QF
Format: Article
Language:English
Published: Dove Medical Press 2025-07-01
Series:International Journal of Nanomedicine
Subjects:
Online Access:https://www.dovepress.com/quercetin-a-natural-ally-in-combating-breast-cancer-peer-reviewed-fulltext-article-IJN
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author Wu ZY
Qiu KY
Gai YJ
Wu JH
Zhou BX
Shi QF
author_facet Wu ZY
Qiu KY
Gai YJ
Wu JH
Zhou BX
Shi QF
author_sort Wu ZY
collection DOAJ
description Zi-Yun Wu, Kang-Yu Qiu, Yan-Jun Gai, Jia-Hui Wu, Bo-Xuan Zhou, Qing-Feng Shi Department of Breast Disease Center, The First Affiliated Hospital of Nanchang University, The First Clinical Medical College of Nanchang University, Jiangxi Medical College, Nanchang, 330006, People’s Republic of ChinaCorrespondence: Bo-Xuan Zhou, Email zhoubx@ncu.edu.cn Qing-Feng Shi, Email A1169627331@163.comAbstract: Breast cancer is one of the most common cancers among women worldwide, exhibiting notably high incidence and mortality rates. Despite its high fatality, a comprehensive study that mechanism and treatment of herbal medicines has not yet been conducted. Quercetin, a natural flavonoid, exhibits multi-targeted therapeutic potential against breast cancer. The aim of this study is to investigate and assess the mechanism and treatment of quercetin in breast cancer. We collected articles published within five years using PubMed, Google Scholar, and Web of Science with “breast cancer” and “quercetin” as keywords. Correspondingly, a total of 272 relevant articles were retrieved. Quercetin exhibits multi-modal therapeutic potential in breast cancer through its ability to orchestrate diverse molecular mechanisms, particularly in TNBC, such as targeting IGF1/IGF1R pathway, PI3K/Akt/mTOR, Wnt/β-catenin, MAPK/ERK cascades, and PTEN promoter demethylation. Critically, quercetin demonstrates synergistic activity with chemotherapy by overcoming drug resistance and reducing toxicity. Its therapeutic efficacy arises from concurrently inducing apoptosis and inhibiting proliferation, migration, invasion and metastasis. This profile positions quercetin as a strategic agent against breast cancer’s complex pathophysiology, effectively disrupting breast cancer malignant progression.Keywords: quercetin, breast cancer, apoptosis, drug carrier, combination therapy
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publisher Dove Medical Press
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series International Journal of Nanomedicine
spelling doaj-art-6c569c7a8fa744a7a196b4c460b412dc2025-08-20T02:39:38ZengDove Medical PressInternational Journal of Nanomedicine1178-20132025-07-01Volume 20Issue 191559177104961Quercetin: A Natural Ally in Combating Breast CancerWu ZY0Qiu KYGai YJWu JHZhou BX1Shi QF2the First Clinical Medical Collegebreast cancer centerThe First Affiliated Hospital of Nanchang UniversityZi-Yun Wu, Kang-Yu Qiu, Yan-Jun Gai, Jia-Hui Wu, Bo-Xuan Zhou, Qing-Feng Shi Department of Breast Disease Center, The First Affiliated Hospital of Nanchang University, The First Clinical Medical College of Nanchang University, Jiangxi Medical College, Nanchang, 330006, People’s Republic of ChinaCorrespondence: Bo-Xuan Zhou, Email zhoubx@ncu.edu.cn Qing-Feng Shi, Email A1169627331@163.comAbstract: Breast cancer is one of the most common cancers among women worldwide, exhibiting notably high incidence and mortality rates. Despite its high fatality, a comprehensive study that mechanism and treatment of herbal medicines has not yet been conducted. Quercetin, a natural flavonoid, exhibits multi-targeted therapeutic potential against breast cancer. The aim of this study is to investigate and assess the mechanism and treatment of quercetin in breast cancer. We collected articles published within five years using PubMed, Google Scholar, and Web of Science with “breast cancer” and “quercetin” as keywords. Correspondingly, a total of 272 relevant articles were retrieved. Quercetin exhibits multi-modal therapeutic potential in breast cancer through its ability to orchestrate diverse molecular mechanisms, particularly in TNBC, such as targeting IGF1/IGF1R pathway, PI3K/Akt/mTOR, Wnt/β-catenin, MAPK/ERK cascades, and PTEN promoter demethylation. Critically, quercetin demonstrates synergistic activity with chemotherapy by overcoming drug resistance and reducing toxicity. Its therapeutic efficacy arises from concurrently inducing apoptosis and inhibiting proliferation, migration, invasion and metastasis. This profile positions quercetin as a strategic agent against breast cancer’s complex pathophysiology, effectively disrupting breast cancer malignant progression.Keywords: quercetin, breast cancer, apoptosis, drug carrier, combination therapyhttps://www.dovepress.com/quercetin-a-natural-ally-in-combating-breast-cancer-peer-reviewed-fulltext-article-IJNQuercetinBreast cancerApoptosisDrug carrierCombination therapy
spellingShingle Wu ZY
Qiu KY
Gai YJ
Wu JH
Zhou BX
Shi QF
Quercetin: A Natural Ally in Combating Breast Cancer
International Journal of Nanomedicine
Quercetin
Breast cancer
Apoptosis
Drug carrier
Combination therapy
title Quercetin: A Natural Ally in Combating Breast Cancer
title_full Quercetin: A Natural Ally in Combating Breast Cancer
title_fullStr Quercetin: A Natural Ally in Combating Breast Cancer
title_full_unstemmed Quercetin: A Natural Ally in Combating Breast Cancer
title_short Quercetin: A Natural Ally in Combating Breast Cancer
title_sort quercetin a natural ally in combating breast cancer
topic Quercetin
Breast cancer
Apoptosis
Drug carrier
Combination therapy
url https://www.dovepress.com/quercetin-a-natural-ally-in-combating-breast-cancer-peer-reviewed-fulltext-article-IJN
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AT gaiyj quercetinanaturalallyincombatingbreastcancer
AT wujh quercetinanaturalallyincombatingbreastcancer
AT zhoubx quercetinanaturalallyincombatingbreastcancer
AT shiqf quercetinanaturalallyincombatingbreastcancer