Testosterone and 5 Alpha Reductase Inhibitor (5ARI) in Benign Prostatic Hyperplasia (BPH): A historical perspective

This paper provides a review of the historical and scientific evolution of testosterone and 5ARI research. It chronicles the evolution from early empirical practices like castration, through the formal discovery of testosterone in the 20th century, to the eventual synthesis of testosterone and ident...

Full description

Saved in:
Bibliographic Details
Main Authors: Ananias C. Diokno, Avaneesh Kunta, Ryan Bowen
Format: Article
Language:English
Published: Elsevier 2024-12-01
Series:Continence
Subjects:
Online Access:http://www.sciencedirect.com/science/article/pii/S2772973724006441
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850124423684685824
author Ananias C. Diokno
Avaneesh Kunta
Ryan Bowen
author_facet Ananias C. Diokno
Avaneesh Kunta
Ryan Bowen
author_sort Ananias C. Diokno
collection DOAJ
description This paper provides a review of the historical and scientific evolution of testosterone and 5ARI research. It chronicles the evolution from early empirical practices like castration, through the formal discovery of testosterone in the 20th century, to the eventual synthesis of testosterone and identification of Leydig cells. Testosterone’s crucial role in male development and its influence on the development and maturation process of the prostate gland are also presented. The introduction of 5ARIs in the 1990s, such as finasteride, marked a significant advancement in managing BPH by reducing dihydrotestosterone (DHT) levels. The controversy regarding the therapeutic use of 5ARIs is discussed, given concerns about their association with high-grade prostate cancer and other systemic risks. Likewise, emerging evidence challenges the traditional view that testosterone exacerbates prostate conditions, suggesting that testosterone replacement therapy (TRT) may improve symptoms of low testosterone without increasing BPH symptoms, prostate cancer (PCa), or cardiovascular risk. Several new studies are discussed suggesting that low or declining testosterone level could be a risk factor for prostate tumorigenesis. This review emphasizes the need for continued research on Testosterone and 5ARI to further define their role in men’s health.
format Article
id doaj-art-66bdfbd797224a53854bc54f00e28e73
institution OA Journals
issn 2772-9737
language English
publishDate 2024-12-01
publisher Elsevier
record_format Article
series Continence
spelling doaj-art-66bdfbd797224a53854bc54f00e28e732025-08-20T02:34:19ZengElsevierContinence2772-97372024-12-011210171110.1016/j.cont.2024.101711Testosterone and 5 Alpha Reductase Inhibitor (5ARI) in Benign Prostatic Hyperplasia (BPH): A historical perspectiveAnanias C. Diokno0Avaneesh Kunta1Ryan Bowen2Oakland University William Beaumont School of Medicine, Rochester, MI, United States of America; University of Central Florida College of Medicine (UCF COM), Orlando, FL, United States of America; Corresponding author at: University of Central Florida College of Medicine (UCF COM), Orlando, FL, United States of America.University of Central Florida College of Medicine (UCF COM), Orlando, FL, United States of AmericaUniversity of Central Florida College of Medicine (UCF COM), Orlando, FL, United States of AmericaThis paper provides a review of the historical and scientific evolution of testosterone and 5ARI research. It chronicles the evolution from early empirical practices like castration, through the formal discovery of testosterone in the 20th century, to the eventual synthesis of testosterone and identification of Leydig cells. Testosterone’s crucial role in male development and its influence on the development and maturation process of the prostate gland are also presented. The introduction of 5ARIs in the 1990s, such as finasteride, marked a significant advancement in managing BPH by reducing dihydrotestosterone (DHT) levels. The controversy regarding the therapeutic use of 5ARIs is discussed, given concerns about their association with high-grade prostate cancer and other systemic risks. Likewise, emerging evidence challenges the traditional view that testosterone exacerbates prostate conditions, suggesting that testosterone replacement therapy (TRT) may improve symptoms of low testosterone without increasing BPH symptoms, prostate cancer (PCa), or cardiovascular risk. Several new studies are discussed suggesting that low or declining testosterone level could be a risk factor for prostate tumorigenesis. This review emphasizes the need for continued research on Testosterone and 5ARI to further define their role in men’s health.http://www.sciencedirect.com/science/article/pii/S2772973724006441Testosterone5 alpha reductase inhibitorsBenign Prostatic HyperplasiaProstate CancerHypogonadismTestosterone Replacement Therapy
spellingShingle Ananias C. Diokno
Avaneesh Kunta
Ryan Bowen
Testosterone and 5 Alpha Reductase Inhibitor (5ARI) in Benign Prostatic Hyperplasia (BPH): A historical perspective
Continence
Testosterone
5 alpha reductase inhibitors
Benign Prostatic Hyperplasia
Prostate Cancer
Hypogonadism
Testosterone Replacement Therapy
title Testosterone and 5 Alpha Reductase Inhibitor (5ARI) in Benign Prostatic Hyperplasia (BPH): A historical perspective
title_full Testosterone and 5 Alpha Reductase Inhibitor (5ARI) in Benign Prostatic Hyperplasia (BPH): A historical perspective
title_fullStr Testosterone and 5 Alpha Reductase Inhibitor (5ARI) in Benign Prostatic Hyperplasia (BPH): A historical perspective
title_full_unstemmed Testosterone and 5 Alpha Reductase Inhibitor (5ARI) in Benign Prostatic Hyperplasia (BPH): A historical perspective
title_short Testosterone and 5 Alpha Reductase Inhibitor (5ARI) in Benign Prostatic Hyperplasia (BPH): A historical perspective
title_sort testosterone and 5 alpha reductase inhibitor 5ari in benign prostatic hyperplasia bph a historical perspective
topic Testosterone
5 alpha reductase inhibitors
Benign Prostatic Hyperplasia
Prostate Cancer
Hypogonadism
Testosterone Replacement Therapy
url http://www.sciencedirect.com/science/article/pii/S2772973724006441
work_keys_str_mv AT ananiascdiokno testosteroneand5alphareductaseinhibitor5ariinbenignprostatichyperplasiabphahistoricalperspective
AT avaneeshkunta testosteroneand5alphareductaseinhibitor5ariinbenignprostatichyperplasiabphahistoricalperspective
AT ryanbowen testosteroneand5alphareductaseinhibitor5ariinbenignprostatichyperplasiabphahistoricalperspective