Manipulation of P2X Receptor Activities by Light Stimulation

P2X receptors are involved in amplification of inflammatory responses in peripheral nociceptive fibers and in mediating pain-related signals to the CNS. Control of P2X activation has significant importance in managing unwanted hypersensitive neuron responses. To overcome the limitations of chemical...

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Main Author: Sang Seong Kim
Format: Article
Language:English
Published: Wiley 2016-01-01
Series:Mediators of Inflammation
Online Access:http://dx.doi.org/10.1155/2016/7852168
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author Sang Seong Kim
author_facet Sang Seong Kim
author_sort Sang Seong Kim
collection DOAJ
description P2X receptors are involved in amplification of inflammatory responses in peripheral nociceptive fibers and in mediating pain-related signals to the CNS. Control of P2X activation has significant importance in managing unwanted hypersensitive neuron responses. To overcome the limitations of chemical ligand treatment, optical stimulation methods of optogenetics and photoswitching achieve efficient control of P2X activation while allowing specificity at the target site and convenient stimulation by light illumination. There are many potential applications for photosensitive elements, such as improved uncaging methods, photoisomerizable ligands, photoswitches, and gold nanoparticles. Each technique has both advantages and downsides, and techniques are selected according to the purpose of the application. Technical advances not only provide novel approaches to manage inflammation or pain mediated by P2X receptors but also suggest a similar approach for controlling other ion channels.
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series Mediators of Inflammation
spelling doaj-art-64bc134f2b9e493c95644d6ef7e9281c2025-08-20T03:34:25ZengWileyMediators of Inflammation0962-93511466-18612016-01-01201610.1155/2016/78521687852168Manipulation of P2X Receptor Activities by Light StimulationSang Seong Kim0Department of Pharmacy, Hanyang University, ERICA Campus, 55 Hanyangdaehak-ro, Sangnok-gu, Ansan, Gyeonggi-do 426-791, Republic of KoreaP2X receptors are involved in amplification of inflammatory responses in peripheral nociceptive fibers and in mediating pain-related signals to the CNS. Control of P2X activation has significant importance in managing unwanted hypersensitive neuron responses. To overcome the limitations of chemical ligand treatment, optical stimulation methods of optogenetics and photoswitching achieve efficient control of P2X activation while allowing specificity at the target site and convenient stimulation by light illumination. There are many potential applications for photosensitive elements, such as improved uncaging methods, photoisomerizable ligands, photoswitches, and gold nanoparticles. Each technique has both advantages and downsides, and techniques are selected according to the purpose of the application. Technical advances not only provide novel approaches to manage inflammation or pain mediated by P2X receptors but also suggest a similar approach for controlling other ion channels.http://dx.doi.org/10.1155/2016/7852168
spellingShingle Sang Seong Kim
Manipulation of P2X Receptor Activities by Light Stimulation
Mediators of Inflammation
title Manipulation of P2X Receptor Activities by Light Stimulation
title_full Manipulation of P2X Receptor Activities by Light Stimulation
title_fullStr Manipulation of P2X Receptor Activities by Light Stimulation
title_full_unstemmed Manipulation of P2X Receptor Activities by Light Stimulation
title_short Manipulation of P2X Receptor Activities by Light Stimulation
title_sort manipulation of p2x receptor activities by light stimulation
url http://dx.doi.org/10.1155/2016/7852168
work_keys_str_mv AT sangseongkim manipulationofp2xreceptoractivitiesbylightstimulation