Functional genomic profiling of O-GlcNAc reveals its context-specific interplay with RNA polymerase II

Abstract Background How reversible glycosylation of DNA-bound proteins acts on transcription remains scarcely understood. O-linked β-N-acetylglucosamine (O-GlcNAc) is the only known form of glycosylation modifying nuclear proteins, including RNA polymerase II (RNA Pol II) and many transcription fact...

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Main Authors: Sofia Rucli, Nicolas Descostes, Yulia Ermakova, Urvashi Chitnavis, Jeanne Couturier, Ana Boskovic, Matthieu Boulard
Format: Article
Language:English
Published: BMC 2025-03-01
Series:Genome Biology
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Online Access:https://doi.org/10.1186/s13059-025-03537-2
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author Sofia Rucli
Nicolas Descostes
Yulia Ermakova
Urvashi Chitnavis
Jeanne Couturier
Ana Boskovic
Matthieu Boulard
author_facet Sofia Rucli
Nicolas Descostes
Yulia Ermakova
Urvashi Chitnavis
Jeanne Couturier
Ana Boskovic
Matthieu Boulard
author_sort Sofia Rucli
collection DOAJ
description Abstract Background How reversible glycosylation of DNA-bound proteins acts on transcription remains scarcely understood. O-linked β-N-acetylglucosamine (O-GlcNAc) is the only known form of glycosylation modifying nuclear proteins, including RNA polymerase II (RNA Pol II) and many transcription factors. Yet, the regulatory function of the O-GlcNAc modification in mammalian chromatin remains unclear. Results Here, we combine genome-wide profiling of O-GlcNAc-modified proteins with perturbations of intracellular glycosylation, RNA Pol II-degron, and super-resolution microscopy. Genomic profiling of O-GlcNAc-modified proteins shows a non-random distribution across the genome, with high densities in heterochromatin regions as well as on actively transcribed gene promoters. Large-scale intersection of the O-GlcNAc signal at promoters with public ChIP-seq datasets identifies a high overlap with RNA Pol II and specific cofactors. Knockdown of O-GlcNAc Transferase (Ogt) shows that most direct target genes are downregulated, supporting a global positive role of O-GlcNAc on the transcription of cellular genes. Rapid degradation of RNA Pol II results in the decrease of the O-GlcNAc levels at promoters encoding transcription factors and DNA modifying enzymes. RNA Pol II depletion also unexpectedly causes an increase of O-GlcNAc levels at a set of promoters encoding for the transcription machinery. Conclusions This study provides a deconvoluted genomic profiling of O-GlcNAc-modified proteins in murine and human cells. Perturbations of O-GlcNAc or RNA Pol II uncover a context-specific reciprocal functional interplay between the transcription machinery and the O-GlcNAc modification.
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spelling doaj-art-5e08b7d90dfc453a9ea0692cdf37396a2025-08-20T02:49:30ZengBMCGenome Biology1474-760X2025-03-0126112510.1186/s13059-025-03537-2Functional genomic profiling of O-GlcNAc reveals its context-specific interplay with RNA polymerase IISofia Rucli0Nicolas Descostes1Yulia Ermakova2Urvashi Chitnavis3Jeanne Couturier4Ana Boskovic5Matthieu Boulard6Epigenetics & Neurobiology Unit, European Molecular Biology Laboratory, EMBL RomeEpigenetics & Neurobiology Unit, European Molecular Biology Laboratory, EMBL RomeEpigenetics & Neurobiology Unit, European Molecular Biology Laboratory, EMBL RomeEpigenetics & Neurobiology Unit, European Molecular Biology Laboratory, EMBL RomeEpigenetics & Neurobiology Unit, European Molecular Biology Laboratory, EMBL RomeEpigenetics & Neurobiology Unit, European Molecular Biology Laboratory, EMBL RomeEpigenetics & Neurobiology Unit, European Molecular Biology Laboratory, EMBL RomeAbstract Background How reversible glycosylation of DNA-bound proteins acts on transcription remains scarcely understood. O-linked β-N-acetylglucosamine (O-GlcNAc) is the only known form of glycosylation modifying nuclear proteins, including RNA polymerase II (RNA Pol II) and many transcription factors. Yet, the regulatory function of the O-GlcNAc modification in mammalian chromatin remains unclear. Results Here, we combine genome-wide profiling of O-GlcNAc-modified proteins with perturbations of intracellular glycosylation, RNA Pol II-degron, and super-resolution microscopy. Genomic profiling of O-GlcNAc-modified proteins shows a non-random distribution across the genome, with high densities in heterochromatin regions as well as on actively transcribed gene promoters. Large-scale intersection of the O-GlcNAc signal at promoters with public ChIP-seq datasets identifies a high overlap with RNA Pol II and specific cofactors. Knockdown of O-GlcNAc Transferase (Ogt) shows that most direct target genes are downregulated, supporting a global positive role of O-GlcNAc on the transcription of cellular genes. Rapid degradation of RNA Pol II results in the decrease of the O-GlcNAc levels at promoters encoding transcription factors and DNA modifying enzymes. RNA Pol II depletion also unexpectedly causes an increase of O-GlcNAc levels at a set of promoters encoding for the transcription machinery. Conclusions This study provides a deconvoluted genomic profiling of O-GlcNAc-modified proteins in murine and human cells. Perturbations of O-GlcNAc or RNA Pol II uncover a context-specific reciprocal functional interplay between the transcription machinery and the O-GlcNAc modification.https://doi.org/10.1186/s13059-025-03537-2O-linked β-N-acetylglucosamineO-GlcNAcOGTGlycosylationTranscriptionPromoter
spellingShingle Sofia Rucli
Nicolas Descostes
Yulia Ermakova
Urvashi Chitnavis
Jeanne Couturier
Ana Boskovic
Matthieu Boulard
Functional genomic profiling of O-GlcNAc reveals its context-specific interplay with RNA polymerase II
Genome Biology
O-linked β-N-acetylglucosamine
O-GlcNAc
OGT
Glycosylation
Transcription
Promoter
title Functional genomic profiling of O-GlcNAc reveals its context-specific interplay with RNA polymerase II
title_full Functional genomic profiling of O-GlcNAc reveals its context-specific interplay with RNA polymerase II
title_fullStr Functional genomic profiling of O-GlcNAc reveals its context-specific interplay with RNA polymerase II
title_full_unstemmed Functional genomic profiling of O-GlcNAc reveals its context-specific interplay with RNA polymerase II
title_short Functional genomic profiling of O-GlcNAc reveals its context-specific interplay with RNA polymerase II
title_sort functional genomic profiling of o glcnac reveals its context specific interplay with rna polymerase ii
topic O-linked β-N-acetylglucosamine
O-GlcNAc
OGT
Glycosylation
Transcription
Promoter
url https://doi.org/10.1186/s13059-025-03537-2
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