The carRS-ompV-virK operon of Vibrio cholerae senses antimicrobial peptides and activates the expression of multiple resistance systems

Abstract Antimicrobial peptides are small cationic molecules produced by eukaryotic cells to combat infection, as well as by bacteria for niche competition. Polymyxin B (PmB), a cyclic antimicrobial peptide, is used prophylactically in livestock and as a last-resort treatment for multidrug-resistant...

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Main Authors: Annabelle Mathieu-Denoncourt, Gregory B Whitfield, Antony T Vincent, Cécile Berne, Julien Pauzé-Foixet, Feriel C Mahieddine, Yves V Brun, Marylise Duperthuy
Format: Article
Language:English
Published: Nature Portfolio 2025-04-01
Series:Scientific Reports
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Online Access:https://doi.org/10.1038/s41598-025-98217-3
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author Annabelle Mathieu-Denoncourt
Gregory B Whitfield
Antony T Vincent
Cécile Berne
Julien Pauzé-Foixet
Feriel C Mahieddine
Yves V Brun
Marylise Duperthuy
author_facet Annabelle Mathieu-Denoncourt
Gregory B Whitfield
Antony T Vincent
Cécile Berne
Julien Pauzé-Foixet
Feriel C Mahieddine
Yves V Brun
Marylise Duperthuy
author_sort Annabelle Mathieu-Denoncourt
collection DOAJ
description Abstract Antimicrobial peptides are small cationic molecules produced by eukaryotic cells to combat infection, as well as by bacteria for niche competition. Polymyxin B (PmB), a cyclic antimicrobial peptide, is used prophylactically in livestock and as a last-resort treatment for multidrug-resistant bacterial infections in humans. In this study, a transcriptomic analysis in Vibrio cholerae showed that expression of the uncharacterized gene ompV is stimulated in response to PmB. We found that ompV is organized in a conserved four-gene operon with the two-component system carRS and virK in V. cholerae. A virK deletion mutant and an ompV deletion mutant were more sensitive to antimicrobials, suggesting that both OmpV and VirK contribute to antimicrobial resistance. Our transcriptomic analysis showed that the efflux pump vexAB, a known effector of PmB resistance, was upregulated in an ompV-dependent manner in the presence of PmB. The predicted structure of OmpV revealed a lateral opening in the β-barrel wall with access to an electronegative pocket in the barrel lumen that can accommodate PmB. Such an interaction could facilitate intracellular signaling through a conformational change in OmpV. This provides the first evidence of a specialized operon governing multiple systems for antimicrobial resistance in V. cholerae.
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spelling doaj-art-5d4c28c2cd4b4ef59eeb25c7b613cd112025-08-20T02:20:06ZengNature PortfolioScientific Reports2045-23222025-04-0115112010.1038/s41598-025-98217-3The carRS-ompV-virK operon of Vibrio cholerae senses antimicrobial peptides and activates the expression of multiple resistance systemsAnnabelle Mathieu-Denoncourt0Gregory B Whitfield1Antony T Vincent2Cécile Berne3Julien Pauzé-Foixet4Feriel C Mahieddine5Yves V Brun6Marylise Duperthuy7Département de Microbiologie, Infectiologie et Immunologie, Faculté de médecine, Université de MontréalDépartement de Microbiologie, Infectiologie et Immunologie, Faculté de médecine, Université de MontréalDépartement des sciences animales, Faculté des sciences de l’agriculture et de l’alimentation, Université LavalDépartement de Microbiologie, Infectiologie et Immunologie, Faculté de médecine, Université de MontréalDépartement de Microbiologie, Infectiologie et Immunologie, Faculté de médecine, Université de MontréalDépartement de Microbiologie, Infectiologie et Immunologie, Faculté de médecine, Université de MontréalDépartement de Microbiologie, Infectiologie et Immunologie, Faculté de médecine, Université de MontréalDépartement de Microbiologie, Infectiologie et Immunologie, Faculté de médecine, Université de MontréalAbstract Antimicrobial peptides are small cationic molecules produced by eukaryotic cells to combat infection, as well as by bacteria for niche competition. Polymyxin B (PmB), a cyclic antimicrobial peptide, is used prophylactically in livestock and as a last-resort treatment for multidrug-resistant bacterial infections in humans. In this study, a transcriptomic analysis in Vibrio cholerae showed that expression of the uncharacterized gene ompV is stimulated in response to PmB. We found that ompV is organized in a conserved four-gene operon with the two-component system carRS and virK in V. cholerae. A virK deletion mutant and an ompV deletion mutant were more sensitive to antimicrobials, suggesting that both OmpV and VirK contribute to antimicrobial resistance. Our transcriptomic analysis showed that the efflux pump vexAB, a known effector of PmB resistance, was upregulated in an ompV-dependent manner in the presence of PmB. The predicted structure of OmpV revealed a lateral opening in the β-barrel wall with access to an electronegative pocket in the barrel lumen that can accommodate PmB. Such an interaction could facilitate intracellular signaling through a conformational change in OmpV. This provides the first evidence of a specialized operon governing multiple systems for antimicrobial resistance in V. cholerae.https://doi.org/10.1038/s41598-025-98217-3Vibrio choleraeOmpVPolymyxin BAntimicrobial peptidesAntimicrobial resistanceResistance Operon
spellingShingle Annabelle Mathieu-Denoncourt
Gregory B Whitfield
Antony T Vincent
Cécile Berne
Julien Pauzé-Foixet
Feriel C Mahieddine
Yves V Brun
Marylise Duperthuy
The carRS-ompV-virK operon of Vibrio cholerae senses antimicrobial peptides and activates the expression of multiple resistance systems
Scientific Reports
Vibrio cholerae
OmpV
Polymyxin B
Antimicrobial peptides
Antimicrobial resistance
Resistance Operon
title The carRS-ompV-virK operon of Vibrio cholerae senses antimicrobial peptides and activates the expression of multiple resistance systems
title_full The carRS-ompV-virK operon of Vibrio cholerae senses antimicrobial peptides and activates the expression of multiple resistance systems
title_fullStr The carRS-ompV-virK operon of Vibrio cholerae senses antimicrobial peptides and activates the expression of multiple resistance systems
title_full_unstemmed The carRS-ompV-virK operon of Vibrio cholerae senses antimicrobial peptides and activates the expression of multiple resistance systems
title_short The carRS-ompV-virK operon of Vibrio cholerae senses antimicrobial peptides and activates the expression of multiple resistance systems
title_sort carrs ompv virk operon of vibrio cholerae senses antimicrobial peptides and activates the expression of multiple resistance systems
topic Vibrio cholerae
OmpV
Polymyxin B
Antimicrobial peptides
Antimicrobial resistance
Resistance Operon
url https://doi.org/10.1038/s41598-025-98217-3
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