Prodrug Strategy for PROTACs: High Efficiency and Low Toxicity

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Main Authors: Yuqing Li, Yongcheng Guo, Simin Ma, Baobang Long, Rui Kong, Xin Huang, Kun Zhao, Ying Zhi
Format: Article
Language:English
Published: American Chemical Society 2025-06-01
Series:ACS Omega
Online Access:https://doi.org/10.1021/acsomega.5c01241
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author Yuqing Li
Yongcheng Guo
Simin Ma
Baobang Long
Rui Kong
Xin Huang
Kun Zhao
Ying Zhi
author_facet Yuqing Li
Yongcheng Guo
Simin Ma
Baobang Long
Rui Kong
Xin Huang
Kun Zhao
Ying Zhi
author_sort Yuqing Li
collection DOAJ
format Article
id doaj-art-5cc956a0810845c9b41e0dbfca15a4f1
institution Kabale University
issn 2470-1343
language English
publishDate 2025-06-01
publisher American Chemical Society
record_format Article
series ACS Omega
spelling doaj-art-5cc956a0810845c9b41e0dbfca15a4f12025-08-20T03:45:40ZengAmerican Chemical SocietyACS Omega2470-13432025-06-011023239262394210.1021/acsomega.5c01241Prodrug Strategy for PROTACs: High Efficiency and Low ToxicityYuqing Li0Yongcheng Guo1Simin Ma2Baobang Long3Rui Kong4Xin Huang5Kun Zhao6Ying Zhi7School of Pharmaceutical Sciences & Institute of Materia Medica, Shandong First Medical University & Shandong Academy of Medical Sciences, Jinan, Shandong, ChinaSchool of Pharmaceutical Sciences & Institute of Materia Medica, Shandong First Medical University & Shandong Academy of Medical Sciences, Jinan, Shandong, ChinaSchool of Pharmaceutical Sciences & Institute of Materia Medica, Shandong First Medical University & Shandong Academy of Medical Sciences, Jinan, Shandong, ChinaSchool of Clinical and Basic Medical Sciences, Shandong First Medical University & Shandong Academy of Medical Sciences, Jinan, Shandong, ChinaSchool of Pharmaceutical Sciences & Institute of Materia Medica, Shandong First Medical University & Shandong Academy of Medical Sciences, Jinan, Shandong, ChinaSchool of Pharmaceutical Sciences & Institute of Materia Medica, Shandong First Medical University & Shandong Academy of Medical Sciences, Jinan, Shandong, ChinaSchool of Pharmaceutical Sciences, Shandong University, Jinan, ChinaSchool of Pharmaceutical Sciences & Institute of Materia Medica, Shandong First Medical University & Shandong Academy of Medical Sciences, Jinan, Shandong, Chinahttps://doi.org/10.1021/acsomega.5c01241
spellingShingle Yuqing Li
Yongcheng Guo
Simin Ma
Baobang Long
Rui Kong
Xin Huang
Kun Zhao
Ying Zhi
Prodrug Strategy for PROTACs: High Efficiency and Low Toxicity
ACS Omega
title Prodrug Strategy for PROTACs: High Efficiency and Low Toxicity
title_full Prodrug Strategy for PROTACs: High Efficiency and Low Toxicity
title_fullStr Prodrug Strategy for PROTACs: High Efficiency and Low Toxicity
title_full_unstemmed Prodrug Strategy for PROTACs: High Efficiency and Low Toxicity
title_short Prodrug Strategy for PROTACs: High Efficiency and Low Toxicity
title_sort prodrug strategy for protacs high efficiency and low toxicity
url https://doi.org/10.1021/acsomega.5c01241
work_keys_str_mv AT yuqingli prodrugstrategyforprotacshighefficiencyandlowtoxicity
AT yongchengguo prodrugstrategyforprotacshighefficiencyandlowtoxicity
AT siminma prodrugstrategyforprotacshighefficiencyandlowtoxicity
AT baobanglong prodrugstrategyforprotacshighefficiencyandlowtoxicity
AT ruikong prodrugstrategyforprotacshighefficiencyandlowtoxicity
AT xinhuang prodrugstrategyforprotacshighefficiencyandlowtoxicity
AT kunzhao prodrugstrategyforprotacshighefficiencyandlowtoxicity
AT yingzhi prodrugstrategyforprotacshighefficiencyandlowtoxicity