Rutin Protects Pancreatic Islets Against Methylglyoxal-Induced Oxidative Stress and Elevates Insulin Secretion

Objective: Hyperglycemia is the main characteristic of diabetes, which leads to complications, including oxidative stress (OS). Pancreatic β-cells are susceptible to damage against OS, which results in a disruption in insulin secretion. The current study focused on the antioxidant features of rutin...

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Main Authors: Elnaz Harooni, Vahid Radmehr, Reza Noei Razliqi, Akram Ahangarpour, Hadi Bazyar
Format: Article
Language:English
Published: Galenos Publishing House 2025-04-01
Series:Gazi Medical Journal
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Online Access:https://gazimedj.com/articles/rutin-protects-pancreatic-islets-against-methylglyoxal-induced-oxidative-stress-and-elevates-insulin-secretion/doi/gmj.2024.4236
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author Elnaz Harooni
Vahid Radmehr
Reza Noei Razliqi
Akram Ahangarpour
Hadi Bazyar
author_facet Elnaz Harooni
Vahid Radmehr
Reza Noei Razliqi
Akram Ahangarpour
Hadi Bazyar
author_sort Elnaz Harooni
collection DOAJ
description Objective: Hyperglycemia is the main characteristic of diabetes, which leads to complications, including oxidative stress (OS). Pancreatic β-cells are susceptible to damage against OS, which results in a disruption in insulin secretion. The current study focused on the antioxidant features of rutin (Rtn) flavonoid to prevent methylglyoxal (MG-)induced oxidative damage in pancreatic islets isolated from mice. Methods: After isolating islets from twenty-four male mice, we conducted two experimental parts, (1) with exposure to MG- and (2) without exposure to MG. Experiments were carried out in both culture media with 5.6- and 16.7-mM glucose concentrations. Islets were transferred to the culture medium and exposed to different substances. In the end, insulin secretion, antioxidant enzyme activities, and malondialdehyde (MDA) concentration were investigated by ELISA. Results: The reduced levels of insulin in MG-exposed islets (p=0.01, p<0.001 in 5.6- and 16.7-mM glucose concentration, respectively) were reversed by Rtn treatment. MG- increased MDA levels in 5.6- and 16.7-mM glucose concentrations (p<0.001 for 5.6 mM and p=0.005 for 16.7 mM. Also, we observed a remarkable decrease in the activities of catalase, superoxide dismutase, and glutathione peroxidase due to 300 μM MG- exposure in islets, in 5.6- and 16.7-mM glucose concentrations. Rtn at doses of 1 and 2 µM significantly reduced MDA levels. Moreover, Rtn had beneficial effects on antioxidant activities. Conclusion: Rtn significantly protected pancreatic islets by reducing lipid peroxidation and enhancing antioxidant activity. The decreased insulin levels in MG-exposed islets were effectively restored in the Rtn-treated groups.
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issn 2147-2092
language English
publishDate 2025-04-01
publisher Galenos Publishing House
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series Gazi Medical Journal
spelling doaj-art-5c151515b2214402bd01ac3dacd68f492025-08-20T03:10:22ZengGalenos Publishing HouseGazi Medical Journal2147-20922025-04-0136217718310.12996/gmj.2024.4236Rutin Protects Pancreatic Islets Against Methylglyoxal-Induced Oxidative Stress and Elevates Insulin SecretionElnaz Harooni0https://orcid.org/0000-0002-0775-7933Vahid Radmehr1https://orcid.org/0000-0002-1889-2233Reza Noei Razliqi2https://orcid.org/0000-0002-4249-0322Akram Ahangarpour3https://orcid.org/0000-0002-9534-9699Hadi Bazyar4https://orcid.org/0000-0002-1627-7122Student Research Committee, Ahvaz Jundishapur University of Medical Sciences, Ahvaz, IranDiabetes Research Center, Health Research Institute, Ahvaz Jundishapur University of Medical Sciences, Ahvaz, IranDepartment of Physiology, Faculty of Medicine, Islamic Azad University Tehran Medical Sciences, Tehran, IranPersian Gulf Physiology Research Center, Medical Basic Sciences Research Institute, Ahvaz Jundishapur University of Medical Sciences, Ahvaz, IranDepartment of Public Health, Sirjan School of Medical Sciences, Sirjan, IranObjective: Hyperglycemia is the main characteristic of diabetes, which leads to complications, including oxidative stress (OS). Pancreatic β-cells are susceptible to damage against OS, which results in a disruption in insulin secretion. The current study focused on the antioxidant features of rutin (Rtn) flavonoid to prevent methylglyoxal (MG-)induced oxidative damage in pancreatic islets isolated from mice. Methods: After isolating islets from twenty-four male mice, we conducted two experimental parts, (1) with exposure to MG- and (2) without exposure to MG. Experiments were carried out in both culture media with 5.6- and 16.7-mM glucose concentrations. Islets were transferred to the culture medium and exposed to different substances. In the end, insulin secretion, antioxidant enzyme activities, and malondialdehyde (MDA) concentration were investigated by ELISA. Results: The reduced levels of insulin in MG-exposed islets (p=0.01, p<0.001 in 5.6- and 16.7-mM glucose concentration, respectively) were reversed by Rtn treatment. MG- increased MDA levels in 5.6- and 16.7-mM glucose concentrations (p<0.001 for 5.6 mM and p=0.005 for 16.7 mM. Also, we observed a remarkable decrease in the activities of catalase, superoxide dismutase, and glutathione peroxidase due to 300 μM MG- exposure in islets, in 5.6- and 16.7-mM glucose concentrations. Rtn at doses of 1 and 2 µM significantly reduced MDA levels. Moreover, Rtn had beneficial effects on antioxidant activities. Conclusion: Rtn significantly protected pancreatic islets by reducing lipid peroxidation and enhancing antioxidant activity. The decreased insulin levels in MG-exposed islets were effectively restored in the Rtn-treated groups.https://gazimedj.com/articles/rutin-protects-pancreatic-islets-against-methylglyoxal-induced-oxidative-stress-and-elevates-insulin-secretion/doi/gmj.2024.4236flavonoidshyperglycemiainsulinmethylglyoxaloxidative stressrutin
spellingShingle Elnaz Harooni
Vahid Radmehr
Reza Noei Razliqi
Akram Ahangarpour
Hadi Bazyar
Rutin Protects Pancreatic Islets Against Methylglyoxal-Induced Oxidative Stress and Elevates Insulin Secretion
Gazi Medical Journal
flavonoids
hyperglycemia
insulin
methylglyoxal
oxidative stress
rutin
title Rutin Protects Pancreatic Islets Against Methylglyoxal-Induced Oxidative Stress and Elevates Insulin Secretion
title_full Rutin Protects Pancreatic Islets Against Methylglyoxal-Induced Oxidative Stress and Elevates Insulin Secretion
title_fullStr Rutin Protects Pancreatic Islets Against Methylglyoxal-Induced Oxidative Stress and Elevates Insulin Secretion
title_full_unstemmed Rutin Protects Pancreatic Islets Against Methylglyoxal-Induced Oxidative Stress and Elevates Insulin Secretion
title_short Rutin Protects Pancreatic Islets Against Methylglyoxal-Induced Oxidative Stress and Elevates Insulin Secretion
title_sort rutin protects pancreatic islets against methylglyoxal induced oxidative stress and elevates insulin secretion
topic flavonoids
hyperglycemia
insulin
methylglyoxal
oxidative stress
rutin
url https://gazimedj.com/articles/rutin-protects-pancreatic-islets-against-methylglyoxal-induced-oxidative-stress-and-elevates-insulin-secretion/doi/gmj.2024.4236
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AT rezanoeirazliqi rutinprotectspancreaticisletsagainstmethylglyoxalinducedoxidativestressandelevatesinsulinsecretion
AT akramahangarpour rutinprotectspancreaticisletsagainstmethylglyoxalinducedoxidativestressandelevatesinsulinsecretion
AT hadibazyar rutinprotectspancreaticisletsagainstmethylglyoxalinducedoxidativestressandelevatesinsulinsecretion