Synthesis and Characterization of Some New Morpholine Derivatives

In this paper a new series of morpholine derivatives was prepared by reacting the morpholine with ethyl chloro acetate in the presence triethylamine as a catalyst in benzene gave morpholin-N-ethyl acetate(1) which reacted with hydrazine hydrate in ethanol, and gave morpholin-N-ethyl acetohydrazid...

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Main Author: Baghdad Science Journal
Format: Article
Language:English
Published: University of Baghdad, College of Science for Women 2016-06-01
Series:مجلة بغداد للعلوم
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Online Access:http://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/2771
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author Baghdad Science Journal
author_facet Baghdad Science Journal
author_sort Baghdad Science Journal
collection DOAJ
description In this paper a new series of morpholine derivatives was prepared by reacting the morpholine with ethyl chloro acetate in the presence triethylamine as a catalyst in benzene gave morpholin-N-ethyl acetate(1) which reacted with hydrazine hydrate in ethanol, and gave morpholin-N-ethyl acetohydrazide (2) . Morpholin-N-aceto semithiocarbazide (3) were prepared by reacting compound(2) with ammonium thiocyanate , concentrated hydrochloric acid and ethanol as a solvent .Compound (3) reacted with sodium hydroxide and hydrochloric acid to give 5-(morpholin-N-methylene)-1H-1,2,4-triazole-3-thiol (4) .The new series of 1,2,4-triazol derivatives (5-8) was synthesized by reaction of compound(4) with formaldehyde , DMF as a solvent and different secondary amines. Preparation of new 1,2,4-triazoline derivatives (9) by reaction compound (4) with bromo acetic acid . Reaction of compound (9) with different aromatic aldehyde and dimethyl sulfoxide as a solvent obtained compounds (10-13).
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publisher University of Baghdad, College of Science for Women
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series مجلة بغداد للعلوم
spelling doaj-art-5b5fc83c36d248e5a2573b76948c585d2025-08-20T03:56:18ZengUniversity of Baghdad, College of Science for Womenمجلة بغداد للعلوم2078-86652411-79862016-06-0113210.21123/bsj.13.2.253-265Synthesis and Characterization of Some New Morpholine DerivativesBaghdad Science JournalIn this paper a new series of morpholine derivatives was prepared by reacting the morpholine with ethyl chloro acetate in the presence triethylamine as a catalyst in benzene gave morpholin-N-ethyl acetate(1) which reacted with hydrazine hydrate in ethanol, and gave morpholin-N-ethyl acetohydrazide (2) . Morpholin-N-aceto semithiocarbazide (3) were prepared by reacting compound(2) with ammonium thiocyanate , concentrated hydrochloric acid and ethanol as a solvent .Compound (3) reacted with sodium hydroxide and hydrochloric acid to give 5-(morpholin-N-methylene)-1H-1,2,4-triazole-3-thiol (4) .The new series of 1,2,4-triazol derivatives (5-8) was synthesized by reaction of compound(4) with formaldehyde , DMF as a solvent and different secondary amines. Preparation of new 1,2,4-triazoline derivatives (9) by reaction compound (4) with bromo acetic acid . Reaction of compound (9) with different aromatic aldehyde and dimethyl sulfoxide as a solvent obtained compounds (10-13).http://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/2771"Morpholine , 1,2,4-triazole and Mannich Reaction"
spellingShingle Baghdad Science Journal
Synthesis and Characterization of Some New Morpholine Derivatives
مجلة بغداد للعلوم
"Morpholine , 1,2,4-triazole and Mannich Reaction"
title Synthesis and Characterization of Some New Morpholine Derivatives
title_full Synthesis and Characterization of Some New Morpholine Derivatives
title_fullStr Synthesis and Characterization of Some New Morpholine Derivatives
title_full_unstemmed Synthesis and Characterization of Some New Morpholine Derivatives
title_short Synthesis and Characterization of Some New Morpholine Derivatives
title_sort synthesis and characterization of some new morpholine derivatives
topic "Morpholine , 1,2,4-triazole and Mannich Reaction"
url http://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/2771
work_keys_str_mv AT baghdadsciencejournal synthesisandcharacterizationofsomenewmorpholinederivatives