Unveiling new features of the human pathogen Cryptococcus neoformans through the reconstruction and exploitation of a dedicated genome-scale metabolic model

Cryptococcus neoformans is notorious for causing severe pulmonary and central nervous system infections, particularly in immunocompromised patients. High mortality rates, associated with its tropism and adaptation to the brain microenvironment and its drug resistance profile, make this pathogen a pu...

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Main Authors: Romeu Viana, Diogo Couceiro, William Newton, Luís Coutinho, Oscar Dias, Carolina Coelho, Miguel Cacho Teixeira
Format: Article
Language:English
Published: Elsevier 2025-01-01
Series:Computational and Structural Biotechnology Journal
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Online Access:http://www.sciencedirect.com/science/article/pii/S2001037025001989
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author Romeu Viana
Diogo Couceiro
William Newton
Luís Coutinho
Oscar Dias
Carolina Coelho
Miguel Cacho Teixeira
author_facet Romeu Viana
Diogo Couceiro
William Newton
Luís Coutinho
Oscar Dias
Carolina Coelho
Miguel Cacho Teixeira
author_sort Romeu Viana
collection DOAJ
description Cryptococcus neoformans is notorious for causing severe pulmonary and central nervous system infections, particularly in immunocompromised patients. High mortality rates, associated with its tropism and adaptation to the brain microenvironment and its drug resistance profile, make this pathogen a public health threat and a World Health Organization (WHO) priority. This study presents the first reconstructed genome-scale metabolic model (GSMM), iRV890, for C. neoformans var. grubii, which comprises 890 genes, 2598 reactions, and 2047 metabolites across four compartments. The GSMM iRV890 model was reconstructed using the open-source software tool merlin 4.0.2, is openly available in the well-established systems biology markup language (SBML) format and underwent validation using experimental data for specific growth and glucose consumption rates, and 222 nitrogen and carbon assimilation sources, with a 85 % prediction rate. Based on the comparison with GSMMs available for other pathogenic yeasts, unique metabolic features were predicted for C. neoformans, including key pathways shaping dynamics between C. neoformans and human host, as well as its underlying adaptions to the brain environment. Finally, the 96 predicted essential genes from the validated model are investigated as potential novel antifungal drug targets—including Erg4, Chs1, Fol1, and Fas1—which represent promising candidates for targeted drug development due to their absence in human cells.
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spelling doaj-art-5aa1ff1baa9248ee8f528f74dcf1d8472025-08-20T03:07:24ZengElsevierComputational and Structural Biotechnology Journal2001-03702025-01-01272336234610.1016/j.csbj.2025.05.034Unveiling new features of the human pathogen Cryptococcus neoformans through the reconstruction and exploitation of a dedicated genome-scale metabolic modelRomeu Viana0Diogo Couceiro1William Newton2Luís Coutinho3Oscar Dias4Carolina Coelho5Miguel Cacho Teixeira6Department of Bioengineering, Instituto Superior Técnico, University of Lisbon, Lisboa 1049-001, Portugal; iBB - Institute for Bioengineering and Biosciences, Associate Laboratory Institute for Health and Bioeconomy - i4HB, Lisboa 1049-001, PortugalDepartment of Bioengineering, Instituto Superior Técnico, University of Lisbon, Lisboa 1049-001, Portugal; iBB - Institute for Bioengineering and Biosciences, Associate Laboratory Institute for Health and Bioeconomy - i4HB, Lisboa 1049-001, Portugal; INESC-ID, R. Alves Redol, 9, Lisbon 1000-029, PortugalMRC Centre for Medical Mycology at University of Exeter, University of Exeter, Exeter, United KingdomDepartment of Bioengineering, Instituto Superior Técnico, University of Lisbon, Lisboa 1049-001, Portugal; iBB - Institute for Bioengineering and Biosciences, Associate Laboratory Institute for Health and Bioeconomy - i4HB, Lisboa 1049-001, PortugalCEB - Centre of Biological Engineering, Universidade do Minho, Braga 4710-057, PortugalMRC Centre for Medical Mycology at University of Exeter, University of Exeter, Exeter, United KingdomDepartment of Bioengineering, Instituto Superior Técnico, University of Lisbon, Lisboa 1049-001, Portugal; iBB - Institute for Bioengineering and Biosciences, Associate Laboratory Institute for Health and Bioeconomy - i4HB, Lisboa 1049-001, Portugal; Corresponding author at: Department of Bioengineering, Instituto Superior Técnico, University of Lisbon, Lisboa 1049-001, Portugal.Cryptococcus neoformans is notorious for causing severe pulmonary and central nervous system infections, particularly in immunocompromised patients. High mortality rates, associated with its tropism and adaptation to the brain microenvironment and its drug resistance profile, make this pathogen a public health threat and a World Health Organization (WHO) priority. This study presents the first reconstructed genome-scale metabolic model (GSMM), iRV890, for C. neoformans var. grubii, which comprises 890 genes, 2598 reactions, and 2047 metabolites across four compartments. The GSMM iRV890 model was reconstructed using the open-source software tool merlin 4.0.2, is openly available in the well-established systems biology markup language (SBML) format and underwent validation using experimental data for specific growth and glucose consumption rates, and 222 nitrogen and carbon assimilation sources, with a 85 % prediction rate. Based on the comparison with GSMMs available for other pathogenic yeasts, unique metabolic features were predicted for C. neoformans, including key pathways shaping dynamics between C. neoformans and human host, as well as its underlying adaptions to the brain environment. Finally, the 96 predicted essential genes from the validated model are investigated as potential novel antifungal drug targets—including Erg4, Chs1, Fol1, and Fas1—which represent promising candidates for targeted drug development due to their absence in human cells.http://www.sciencedirect.com/science/article/pii/S2001037025001989C. neoformansGlobal stoichiometric modelDrug targetsMetabolic featuresNeurotropism
spellingShingle Romeu Viana
Diogo Couceiro
William Newton
Luís Coutinho
Oscar Dias
Carolina Coelho
Miguel Cacho Teixeira
Unveiling new features of the human pathogen Cryptococcus neoformans through the reconstruction and exploitation of a dedicated genome-scale metabolic model
Computational and Structural Biotechnology Journal
C. neoformans
Global stoichiometric model
Drug targets
Metabolic features
Neurotropism
title Unveiling new features of the human pathogen Cryptococcus neoformans through the reconstruction and exploitation of a dedicated genome-scale metabolic model
title_full Unveiling new features of the human pathogen Cryptococcus neoformans through the reconstruction and exploitation of a dedicated genome-scale metabolic model
title_fullStr Unveiling new features of the human pathogen Cryptococcus neoformans through the reconstruction and exploitation of a dedicated genome-scale metabolic model
title_full_unstemmed Unveiling new features of the human pathogen Cryptococcus neoformans through the reconstruction and exploitation of a dedicated genome-scale metabolic model
title_short Unveiling new features of the human pathogen Cryptococcus neoformans through the reconstruction and exploitation of a dedicated genome-scale metabolic model
title_sort unveiling new features of the human pathogen cryptococcus neoformans through the reconstruction and exploitation of a dedicated genome scale metabolic model
topic C. neoformans
Global stoichiometric model
Drug targets
Metabolic features
Neurotropism
url http://www.sciencedirect.com/science/article/pii/S2001037025001989
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