Acalypha indica aqueous leaf extract as potential nematicide against the root-knot nematode, Meloidogyne incognita: in vitro and molecular docking studies

Root-knot nematode (RKN) (Meloidogyne incognita) is a major plant parasitic nematode that severely damages crops, leading to significant yield losses and substantial economic impact globally. This study aims to investigate an environmentally sustainable biological strategy for mitigating parasitic p...

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Main Authors: Altaf Khan, Manar Fawzi Bani Mfarrej, Fohad Mabood Husain, Qamar Zia, Mohd Adil, Mohammed Arshad, Khalid Umar, Niraj Kumar Jha, Pieter Malan, Soumya Pandit, Faheem Ahmad
Format: Article
Language:English
Published: Taylor & Francis Group 2024-12-01
Series:Cogent Food & Agriculture
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Online Access:https://www.tandfonline.com/doi/10.1080/23311932.2024.2405027
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author Altaf Khan
Manar Fawzi Bani Mfarrej
Fohad Mabood Husain
Qamar Zia
Mohd Adil
Mohammed Arshad
Khalid Umar
Niraj Kumar Jha
Pieter Malan
Soumya Pandit
Faheem Ahmad
author_facet Altaf Khan
Manar Fawzi Bani Mfarrej
Fohad Mabood Husain
Qamar Zia
Mohd Adil
Mohammed Arshad
Khalid Umar
Niraj Kumar Jha
Pieter Malan
Soumya Pandit
Faheem Ahmad
author_sort Altaf Khan
collection DOAJ
description Root-knot nematode (RKN) (Meloidogyne incognita) is a major plant parasitic nematode that severely damages crops, leading to significant yield losses and substantial economic impact globally. This study aims to investigate an environmentally sustainable biological strategy for mitigating parasitic populations of the root-knot nematode, M. incognita. Specifically, the research focuses on assessing the nematicidal efficacy of Acalypha indica against M. incognita mortality and second-stage juveniles’ (J2) hatching under controlled in vitro conditions. A. indica leaf aqueous extract was applied at varying concentrations (250, 500, 750, and 1000 ppm) to J2s and egg masses of M. incognita. Notably, at 1000 ppm, a significant increase in J2 mortality and hatching inhibition was observed, while 250 ppm concentration showed the least favorable outcome; with mortality rates ranging from 22–82%. Chemical analysis via gas chromatography-mass spectroscopy (GC-MS) identified Benzoic acid, Cyclooctasiloxane, and 3-Isopropoxy-1,1,1,7,7,7-hexamethyl-3,5,5-tris (trimethylsiloxy) tetrasiloxane as predominant compounds. The nematicidal activity of A. indica leaf extract was further validated through in silico molecular docking, revealing that benzoic acid, Cyclooctasiloxane, and 3-Isopropoxy-1,1,1,7,7,7-hexamethyl-3,5,5-tris (trimethylsiloxy) tetrasiloxane bind to the ODR 3 protein of M. incognita with binding energies of −15.72, −8.91, and −7.35 kJ/mol, respectively. These findings hold promise for environmentally benign root-knot nematode management, contributing to improved soil health.
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spelling doaj-art-5a7edc0a56ad4346854cd8a0ce29afc62025-08-20T01:58:52ZengTaylor & Francis GroupCogent Food & Agriculture2331-19322024-12-0110110.1080/23311932.2024.2405027Acalypha indica aqueous leaf extract as potential nematicide against the root-knot nematode, Meloidogyne incognita: in vitro and molecular docking studiesAltaf Khan0Manar Fawzi Bani Mfarrej1Fohad Mabood Husain2Qamar Zia3Mohd Adil4Mohammed Arshad5Khalid Umar6Niraj Kumar Jha7Pieter Malan8Soumya Pandit9Faheem Ahmad10Department of Pharmacology, College of Pharmacy, King Saud University, Riyadh, KSADepartment of Life and Environmental Sciences, College of Natural and Health Sciences, Zayed University, United Arab EmiratesDepartment of Food Science and Nutrition, King Saud University, Riyadh, KSAInterdisciplinary Biotechnology Unit, Aligarh Muslim University, Aligarh, IndiaDepartment of Environmental Sciences, Dalhousie University, Truro, Nova Scotia, CanadaDental Health Department, College of Applied Medical Sciences, King Saud University, Riyadh, KSASchool of Chemical Sciences, Universiti Sains Malaysia, Gelugor, Pulau Pinang, MalaysiaCentre for Global Health Research, Saveetha Medical College, Saveetha Institute of Medical and Technical Sciences, Saveetha University, Chennai, IndiaUnit for Environmental Sciences and Management, Mafikeng Campus, North-West University, Mmabatho, South AfricaDepartment of Biotechnology, Graphic Era University, Dehradun, Uttarakhand, IndiaDepartment of Botany, Aligarh Muslim University, Aligarh, IndiaRoot-knot nematode (RKN) (Meloidogyne incognita) is a major plant parasitic nematode that severely damages crops, leading to significant yield losses and substantial economic impact globally. This study aims to investigate an environmentally sustainable biological strategy for mitigating parasitic populations of the root-knot nematode, M. incognita. Specifically, the research focuses on assessing the nematicidal efficacy of Acalypha indica against M. incognita mortality and second-stage juveniles’ (J2) hatching under controlled in vitro conditions. A. indica leaf aqueous extract was applied at varying concentrations (250, 500, 750, and 1000 ppm) to J2s and egg masses of M. incognita. Notably, at 1000 ppm, a significant increase in J2 mortality and hatching inhibition was observed, while 250 ppm concentration showed the least favorable outcome; with mortality rates ranging from 22–82%. Chemical analysis via gas chromatography-mass spectroscopy (GC-MS) identified Benzoic acid, Cyclooctasiloxane, and 3-Isopropoxy-1,1,1,7,7,7-hexamethyl-3,5,5-tris (trimethylsiloxy) tetrasiloxane as predominant compounds. The nematicidal activity of A. indica leaf extract was further validated through in silico molecular docking, revealing that benzoic acid, Cyclooctasiloxane, and 3-Isopropoxy-1,1,1,7,7,7-hexamethyl-3,5,5-tris (trimethylsiloxy) tetrasiloxane bind to the ODR 3 protein of M. incognita with binding energies of −15.72, −8.91, and −7.35 kJ/mol, respectively. These findings hold promise for environmentally benign root-knot nematode management, contributing to improved soil health.https://www.tandfonline.com/doi/10.1080/23311932.2024.2405027BotanicalsAcalypha indicamolecular dockingMeloidogyne incognitanematicidal activityPlant Pathology
spellingShingle Altaf Khan
Manar Fawzi Bani Mfarrej
Fohad Mabood Husain
Qamar Zia
Mohd Adil
Mohammed Arshad
Khalid Umar
Niraj Kumar Jha
Pieter Malan
Soumya Pandit
Faheem Ahmad
Acalypha indica aqueous leaf extract as potential nematicide against the root-knot nematode, Meloidogyne incognita: in vitro and molecular docking studies
Cogent Food & Agriculture
Botanicals
Acalypha indica
molecular docking
Meloidogyne incognita
nematicidal activity
Plant Pathology
title Acalypha indica aqueous leaf extract as potential nematicide against the root-knot nematode, Meloidogyne incognita: in vitro and molecular docking studies
title_full Acalypha indica aqueous leaf extract as potential nematicide against the root-knot nematode, Meloidogyne incognita: in vitro and molecular docking studies
title_fullStr Acalypha indica aqueous leaf extract as potential nematicide against the root-knot nematode, Meloidogyne incognita: in vitro and molecular docking studies
title_full_unstemmed Acalypha indica aqueous leaf extract as potential nematicide against the root-knot nematode, Meloidogyne incognita: in vitro and molecular docking studies
title_short Acalypha indica aqueous leaf extract as potential nematicide against the root-knot nematode, Meloidogyne incognita: in vitro and molecular docking studies
title_sort acalypha indica aqueous leaf extract as potential nematicide against the root knot nematode meloidogyne incognita in vitro and molecular docking studies
topic Botanicals
Acalypha indica
molecular docking
Meloidogyne incognita
nematicidal activity
Plant Pathology
url https://www.tandfonline.com/doi/10.1080/23311932.2024.2405027
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