A Convenient Synthesis of C-3-Aryloxymethyl Imidazo[1,2-a]Pyridine Derivatives

Imidazo[1,2-a]pyridine-based tosylhydrazone was prepared and treated with K2CO3 in dioxane at 110°C to generate the corresponding carbene in situ. It was coupled with a variety of aryl alcohols in one pot to obtain a series of imidazo[1,2-a]pyridine derivatives possessing aryl ether moiety at C-3 po...

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Main Authors: Sridevi Kona, Rama Suresh Ravi, Venkata N. R. Chava, Ramu Sridhar Perali
Format: Article
Language:English
Published: Wiley 2013-01-01
Series:Journal of Chemistry
Online Access:http://dx.doi.org/10.1155/2013/296792
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author Sridevi Kona
Rama Suresh Ravi
Venkata N. R. Chava
Ramu Sridhar Perali
author_facet Sridevi Kona
Rama Suresh Ravi
Venkata N. R. Chava
Ramu Sridhar Perali
author_sort Sridevi Kona
collection DOAJ
description Imidazo[1,2-a]pyridine-based tosylhydrazone was prepared and treated with K2CO3 in dioxane at 110°C to generate the corresponding carbene in situ. It was coupled with a variety of aryl alcohols in one pot to obtain a series of imidazo[1,2-a]pyridine derivatives possessing aryl ether moiety at C-3 position.
format Article
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publishDate 2013-01-01
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spelling doaj-art-572f243e7c9b4645bef99a5cb2554c392025-08-20T02:05:57ZengWileyJournal of Chemistry2090-90632090-90712013-01-01201310.1155/2013/296792296792A Convenient Synthesis of C-3-Aryloxymethyl Imidazo[1,2-a]Pyridine DerivativesSridevi Kona0Rama Suresh Ravi1Venkata N. R. Chava2Ramu Sridhar Perali3School of Chemistry, University of Hyderabad, Andhra Pradesh, Hyderabad 500046, IndiaSchool of Chemistry, University of Hyderabad, Andhra Pradesh, Hyderabad 500046, IndiaDepartment of Chemistry, AG & SG Siddhartha Arts and Science College, Andhra Pradesh, Vuyyuru 521165, IndiaSchool of Chemistry, University of Hyderabad, Andhra Pradesh, Hyderabad 500046, IndiaImidazo[1,2-a]pyridine-based tosylhydrazone was prepared and treated with K2CO3 in dioxane at 110°C to generate the corresponding carbene in situ. It was coupled with a variety of aryl alcohols in one pot to obtain a series of imidazo[1,2-a]pyridine derivatives possessing aryl ether moiety at C-3 position.http://dx.doi.org/10.1155/2013/296792
spellingShingle Sridevi Kona
Rama Suresh Ravi
Venkata N. R. Chava
Ramu Sridhar Perali
A Convenient Synthesis of C-3-Aryloxymethyl Imidazo[1,2-a]Pyridine Derivatives
Journal of Chemistry
title A Convenient Synthesis of C-3-Aryloxymethyl Imidazo[1,2-a]Pyridine Derivatives
title_full A Convenient Synthesis of C-3-Aryloxymethyl Imidazo[1,2-a]Pyridine Derivatives
title_fullStr A Convenient Synthesis of C-3-Aryloxymethyl Imidazo[1,2-a]Pyridine Derivatives
title_full_unstemmed A Convenient Synthesis of C-3-Aryloxymethyl Imidazo[1,2-a]Pyridine Derivatives
title_short A Convenient Synthesis of C-3-Aryloxymethyl Imidazo[1,2-a]Pyridine Derivatives
title_sort convenient synthesis of c 3 aryloxymethyl imidazo 1 2 a pyridine derivatives
url http://dx.doi.org/10.1155/2013/296792
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