Ellagitannin Oligomers from <i>Eucalyptus camaldulensis</i> Leaves and Their Role in the Detoxification of Aluminum

<i>Eucalyptus camaldulensis</i> of the Myrtaceae family shows high resistance to aluminum (Al) ions and contains various compounds such as steroids, terpenoids, saponins, flavonoids, glycosides, alkaloids, and tannins. Although the ellagitannin oenothein B (<b>12</b>) isolate...

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Main Authors: Haruna Uemori, Ayano Inoue, Shoichi Suzuki, Yuji Iwaoka, Tsutomu Hatano, Morio Yoshimura, Yoshiaki Amakura, Toshiyuki Murakami, Ko Tahara, Hideyuki Ito
Format: Article
Language:English
Published: MDPI AG 2025-05-01
Series:Molecules
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Online Access:https://www.mdpi.com/1420-3049/30/10/2216
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author Haruna Uemori
Ayano Inoue
Shoichi Suzuki
Yuji Iwaoka
Tsutomu Hatano
Morio Yoshimura
Yoshiaki Amakura
Toshiyuki Murakami
Ko Tahara
Hideyuki Ito
author_facet Haruna Uemori
Ayano Inoue
Shoichi Suzuki
Yuji Iwaoka
Tsutomu Hatano
Morio Yoshimura
Yoshiaki Amakura
Toshiyuki Murakami
Ko Tahara
Hideyuki Ito
author_sort Haruna Uemori
collection DOAJ
description <i>Eucalyptus camaldulensis</i> of the Myrtaceae family shows high resistance to aluminum (Al) ions and contains various compounds such as steroids, terpenoids, saponins, flavonoids, glycosides, alkaloids, and tannins. Although the ellagitannin oenothein B (<b>12</b>) isolated from <i>E. camaldulensis</i> exhibits remarkable properties for Al detoxification, likely contributing to its Al resistance, other ellagitannin oligomers present in <i>E. camaldulensis</i> have not been investigated in detail. In this study, novel dimeric and trimeric ellagitannin oligomers eucarpanin D<sub>2</sub> (<b>1</b>) and eucamalin A (<b>2</b>), together with known gallotannins (<b>7</b>, <b>8</b>, and <b>10</b>), monomeric ellagitannins (<b>4</b>–<b>6</b>, and <b>11</b>), and dimeric ellagitannins (<b>3</b>, <b>9</b>, and <b>12</b>–<b>14</b>), were isolated from <i>E. camaldulensis</i> leaves. The structures of these novel compounds were elucidated based on their chemical and physicochemical properties, including the orientations of tergalloyl groups in compounds <b>1</b> and <b>2</b>. Similar to compound <b>12</b>, previously isolated from the roots of <i>E. camaldulensis</i>, the ellagitannins demonstrated good Al detoxification properties. Hence, these tannins may play a critical role in the high Al resistance of <i>E. camaldulensis</i> in acidic soils. This paper reports for the first time the isolation of ellagitannin oligomers from the leaves of <i>E. camaldulensis</i>.
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spelling doaj-art-5396f16647c245ee8ecc3452bc1580f32025-08-20T03:48:02ZengMDPI AGMolecules1420-30492025-05-013010221610.3390/molecules30102216Ellagitannin Oligomers from <i>Eucalyptus camaldulensis</i> Leaves and Their Role in the Detoxification of AluminumHaruna Uemori0Ayano Inoue1Shoichi Suzuki2Yuji Iwaoka3Tsutomu Hatano4Morio Yoshimura5Yoshiaki Amakura6Toshiyuki Murakami7Ko Tahara8Hideyuki Ito9Doctorate Course of Health and Welfare Science, Graduate School of Okayama Prefectural University, 111 Kuboki, Soja 719-1197, Okayama, JapanFaculty of Health and Welfare Science, Okayama Prefectural University, 111 Kuboki, Soja 719-1197, Okayama, JapanFaculty of Health and Welfare Science, Okayama Prefectural University, 111 Kuboki, Soja 719-1197, Okayama, JapanDoctorate Course of Health and Welfare Science, Graduate School of Okayama Prefectural University, 111 Kuboki, Soja 719-1197, Okayama, JapanDivision of Pharmaceutical Sciences, Graduate School of Medicine, Dentistry, Pharmaceutical Sciences, Okayama University, 1-1-1 Tsushima-Naka, Kita-ku 700-8530, Okayama, JapanPharmaceutical Sciences, Matsuyama University, 4-2 Bunkyo-cho, Matsuyama 790-8578, Ehime, JapanPharmaceutical Sciences, Matsuyama University, 4-2 Bunkyo-cho, Matsuyama 790-8578, Ehime, JapanResearch Center, Maruzen Pharmaceuticals, Co., Ltd., 1089-8 Sagata, Shinnichi-Cho, Fukuyama 729-3102, Hiroshima, JapanForestry and Forest Products Research Institute, 1 Matunosato, Tsukuba 305-8687, Ibaraki, JapanDoctorate Course of Health and Welfare Science, Graduate School of Okayama Prefectural University, 111 Kuboki, Soja 719-1197, Okayama, Japan<i>Eucalyptus camaldulensis</i> of the Myrtaceae family shows high resistance to aluminum (Al) ions and contains various compounds such as steroids, terpenoids, saponins, flavonoids, glycosides, alkaloids, and tannins. Although the ellagitannin oenothein B (<b>12</b>) isolated from <i>E. camaldulensis</i> exhibits remarkable properties for Al detoxification, likely contributing to its Al resistance, other ellagitannin oligomers present in <i>E. camaldulensis</i> have not been investigated in detail. In this study, novel dimeric and trimeric ellagitannin oligomers eucarpanin D<sub>2</sub> (<b>1</b>) and eucamalin A (<b>2</b>), together with known gallotannins (<b>7</b>, <b>8</b>, and <b>10</b>), monomeric ellagitannins (<b>4</b>–<b>6</b>, and <b>11</b>), and dimeric ellagitannins (<b>3</b>, <b>9</b>, and <b>12</b>–<b>14</b>), were isolated from <i>E. camaldulensis</i> leaves. The structures of these novel compounds were elucidated based on their chemical and physicochemical properties, including the orientations of tergalloyl groups in compounds <b>1</b> and <b>2</b>. Similar to compound <b>12</b>, previously isolated from the roots of <i>E. camaldulensis</i>, the ellagitannins demonstrated good Al detoxification properties. Hence, these tannins may play a critical role in the high Al resistance of <i>E. camaldulensis</i> in acidic soils. This paper reports for the first time the isolation of ellagitannin oligomers from the leaves of <i>E. camaldulensis</i>.https://www.mdpi.com/1420-3049/30/10/2216<i>Eucalyptus camaldulensis</i> Dehnh.ellagitannin oligomereucamalin Aeucarpanin D<sub>2</sub>eurobustin CAl detoxification
spellingShingle Haruna Uemori
Ayano Inoue
Shoichi Suzuki
Yuji Iwaoka
Tsutomu Hatano
Morio Yoshimura
Yoshiaki Amakura
Toshiyuki Murakami
Ko Tahara
Hideyuki Ito
Ellagitannin Oligomers from <i>Eucalyptus camaldulensis</i> Leaves and Their Role in the Detoxification of Aluminum
Molecules
<i>Eucalyptus camaldulensis</i> Dehnh.
ellagitannin oligomer
eucamalin A
eucarpanin D<sub>2</sub>
eurobustin C
Al detoxification
title Ellagitannin Oligomers from <i>Eucalyptus camaldulensis</i> Leaves and Their Role in the Detoxification of Aluminum
title_full Ellagitannin Oligomers from <i>Eucalyptus camaldulensis</i> Leaves and Their Role in the Detoxification of Aluminum
title_fullStr Ellagitannin Oligomers from <i>Eucalyptus camaldulensis</i> Leaves and Their Role in the Detoxification of Aluminum
title_full_unstemmed Ellagitannin Oligomers from <i>Eucalyptus camaldulensis</i> Leaves and Their Role in the Detoxification of Aluminum
title_short Ellagitannin Oligomers from <i>Eucalyptus camaldulensis</i> Leaves and Their Role in the Detoxification of Aluminum
title_sort ellagitannin oligomers from i eucalyptus camaldulensis i leaves and their role in the detoxification of aluminum
topic <i>Eucalyptus camaldulensis</i> Dehnh.
ellagitannin oligomer
eucamalin A
eucarpanin D<sub>2</sub>
eurobustin C
Al detoxification
url https://www.mdpi.com/1420-3049/30/10/2216
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