DEVELOPMENT AND VALIDATION OF A SPECTROFLUORIMETRIC METHOD FOR THE DETERMINATION OF PHENIBUT IN TABLET DRUGS

The developed method for the quantitative determination of phenibut in tablet drugs is based on the dansylation reaction in an alkaline medium (pH 9.18). The reaction results in the formation of a fluorescent derivative with λem=505 nm and λex=335 nm. Optimal conditions were selected to complete the...

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Main Authors: O. I. Lazovskaya, V. N. Leontiev, E. V. Litvinova
Format: Article
Language:Russian
Published: LLC Center of Pharmaceutical Analytics (LLC «CPHA») 2019-01-01
Series:Разработка и регистрация лекарственных средств
Subjects:
Online Access:https://www.pharmjournal.ru/jour/article/view/504
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author O. I. Lazovskaya
V. N. Leontiev
E. V. Litvinova
author_facet O. I. Lazovskaya
V. N. Leontiev
E. V. Litvinova
author_sort O. I. Lazovskaya
collection DOAJ
description The developed method for the quantitative determination of phenibut in tablet drugs is based on the dansylation reaction in an alkaline medium (pH 9.18). The reaction results in the formation of a fluorescent derivative with λem=505 nm and λex=335 nm. Optimal conditions were selected to complete the reaction: temperature and time of thermostatting (40 °C and 15 min), molar ratio of phenibut and dansyl chloride (1:1.4). The method was validated in parameters of specificity, linearity, precision and accuracy. A plot of fluorescence intensity versus concentration of phenibut over the range of 800-1200 ng/ml is described by the regression equation y =0.1003x+1.4685 ( r =0.9999). The limit of detection and limit of quantification were 29.55 и 89.54 ng/ml respectively.
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institution Kabale University
issn 2305-2066
2658-5049
language Russian
publishDate 2019-01-01
publisher LLC Center of Pharmaceutical Analytics (LLC «CPHA»)
record_format Article
series Разработка и регистрация лекарственных средств
spelling doaj-art-52c0d70462a64c8288f6e273c87f9b522025-08-20T03:59:20ZrusLLC Center of Pharmaceutical Analytics (LLC «CPHA»)Разработка и регистрация лекарственных средств2305-20662658-50492019-01-0104104107504DEVELOPMENT AND VALIDATION OF A SPECTROFLUORIMETRIC METHOD FOR THE DETERMINATION OF PHENIBUT IN TABLET DRUGSO. I. Lazovskaya0V. N. Leontiev1E. V. Litvinova2Belarusian State Technological UniversityBelarusian State Technological UniversityRUE «Belmedpreparaty»The developed method for the quantitative determination of phenibut in tablet drugs is based on the dansylation reaction in an alkaline medium (pH 9.18). The reaction results in the formation of a fluorescent derivative with λem=505 nm and λex=335 nm. Optimal conditions were selected to complete the reaction: temperature and time of thermostatting (40 °C and 15 min), molar ratio of phenibut and dansyl chloride (1:1.4). The method was validated in parameters of specificity, linearity, precision and accuracy. A plot of fluorescence intensity versus concentration of phenibut over the range of 800-1200 ng/ml is described by the regression equation y =0.1003x+1.4685 ( r =0.9999). The limit of detection and limit of quantification were 29.55 и 89.54 ng/ml respectively.https://www.pharmjournal.ru/jour/article/view/504fluorescence spectroscopydansyl chloridephenibuttablet drugvalidation
spellingShingle O. I. Lazovskaya
V. N. Leontiev
E. V. Litvinova
DEVELOPMENT AND VALIDATION OF A SPECTROFLUORIMETRIC METHOD FOR THE DETERMINATION OF PHENIBUT IN TABLET DRUGS
Разработка и регистрация лекарственных средств
fluorescence spectroscopy
dansyl chloride
phenibut
tablet drug
validation
title DEVELOPMENT AND VALIDATION OF A SPECTROFLUORIMETRIC METHOD FOR THE DETERMINATION OF PHENIBUT IN TABLET DRUGS
title_full DEVELOPMENT AND VALIDATION OF A SPECTROFLUORIMETRIC METHOD FOR THE DETERMINATION OF PHENIBUT IN TABLET DRUGS
title_fullStr DEVELOPMENT AND VALIDATION OF A SPECTROFLUORIMETRIC METHOD FOR THE DETERMINATION OF PHENIBUT IN TABLET DRUGS
title_full_unstemmed DEVELOPMENT AND VALIDATION OF A SPECTROFLUORIMETRIC METHOD FOR THE DETERMINATION OF PHENIBUT IN TABLET DRUGS
title_short DEVELOPMENT AND VALIDATION OF A SPECTROFLUORIMETRIC METHOD FOR THE DETERMINATION OF PHENIBUT IN TABLET DRUGS
title_sort development and validation of a spectrofluorimetric method for the determination of phenibut in tablet drugs
topic fluorescence spectroscopy
dansyl chloride
phenibut
tablet drug
validation
url https://www.pharmjournal.ru/jour/article/view/504
work_keys_str_mv AT oilazovskaya developmentandvalidationofaspectrofluorimetricmethodforthedeterminationofphenibutintabletdrugs
AT vnleontiev developmentandvalidationofaspectrofluorimetricmethodforthedeterminationofphenibutintabletdrugs
AT evlitvinova developmentandvalidationofaspectrofluorimetricmethodforthedeterminationofphenibutintabletdrugs