Synthesis, Characterization and study biologicalactivity of several 1-cyclopentene-1,2-dicarboxylimidyl Containing oxadiazole and Benzothiazole
In this work involved prepared of several new 1-cyclopentene-1,2-dicarboxylimide linked to oxadiazole and benzothiazole moiety were synthesized by two steps: The first step 2-amino-substituted-1,3,4-oxadiazoles and substituted-2-aminobenzothiazole were reaction with 1-cyclopentene-1,2-dicarboxyl anh...
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University of Baghdad, College of Science for Women
2014-06-01
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| Series: | مجلة بغداد للعلوم |
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| Online Access: | http://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/2647 |
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| author | Baghdad Science Journal |
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| description | In this work involved prepared of several new 1-cyclopentene-1,2-dicarboxylimide linked to oxadiazole and benzothiazole moiety were synthesized by two steps:
The first step 2-amino-substituted-1,3,4-oxadiazoles and substituted-2-aminobenzothiazole were reaction with 1-cyclopentene-1,2-dicarboxyl anhydride producing N-( 5- substituted-1,3,4-oxadiazole-2-yl)-1-cyclopentene-1,2-dicarboxyl amic acids and N-(Substitutedbenzothiazole-2-yl)-1-cyclopentene-1,2-dicarboxyl amic acids which in turn were dehydrated in the second step via fusion method to afford he desirable N-(5-substituted-1,3,4-oxadiazole-2-yl)-1-cyclopentene-1,2-dicarboxylimides and N-(Substituted benzothiazole-2-yl)1-cyclopentene-1,2-dicarboxylimides respectively. Structures of the prepared compounds were characterized by depending on FTIR, U.V spectral data which were in agreement with the proposed ones. Finally antibacterial activity of some of the prepared new cyclic imides were studied by two types of bacteria and the results showed that the most of the tested imides posses good biological activity against these bacteria. |
| format | Article |
| id | doaj-art-5283f6ac0d144991acb3871b08a3da68 |
| institution | Kabale University |
| issn | 2078-8665 2411-7986 |
| language | English |
| publishDate | 2014-06-01 |
| publisher | University of Baghdad, College of Science for Women |
| record_format | Article |
| series | مجلة بغداد للعلوم |
| spelling | doaj-art-5283f6ac0d144991acb3871b08a3da682025-08-20T03:33:32ZengUniversity of Baghdad, College of Science for Womenمجلة بغداد للعلوم2078-86652411-79862014-06-0111210.21123/bsj.11.2.429-437Synthesis, Characterization and study biologicalactivity of several 1-cyclopentene-1,2-dicarboxylimidyl Containing oxadiazole and BenzothiazoleBaghdad Science JournalIn this work involved prepared of several new 1-cyclopentene-1,2-dicarboxylimide linked to oxadiazole and benzothiazole moiety were synthesized by two steps: The first step 2-amino-substituted-1,3,4-oxadiazoles and substituted-2-aminobenzothiazole were reaction with 1-cyclopentene-1,2-dicarboxyl anhydride producing N-( 5- substituted-1,3,4-oxadiazole-2-yl)-1-cyclopentene-1,2-dicarboxyl amic acids and N-(Substitutedbenzothiazole-2-yl)-1-cyclopentene-1,2-dicarboxyl amic acids which in turn were dehydrated in the second step via fusion method to afford he desirable N-(5-substituted-1,3,4-oxadiazole-2-yl)-1-cyclopentene-1,2-dicarboxylimides and N-(Substituted benzothiazole-2-yl)1-cyclopentene-1,2-dicarboxylimides respectively. Structures of the prepared compounds were characterized by depending on FTIR, U.V spectral data which were in agreement with the proposed ones. Finally antibacterial activity of some of the prepared new cyclic imides were studied by two types of bacteria and the results showed that the most of the tested imides posses good biological activity against these bacteria.http://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/26471-cyclopentene-1,2-dicarboxylimidyl, oxadiazol, benzothiazol. |
| spellingShingle | Baghdad Science Journal Synthesis, Characterization and study biologicalactivity of several 1-cyclopentene-1,2-dicarboxylimidyl Containing oxadiazole and Benzothiazole مجلة بغداد للعلوم 1-cyclopentene-1,2-dicarboxylimidyl, oxadiazol, benzothiazol. |
| title | Synthesis, Characterization and study biologicalactivity of several 1-cyclopentene-1,2-dicarboxylimidyl Containing oxadiazole and Benzothiazole |
| title_full | Synthesis, Characterization and study biologicalactivity of several 1-cyclopentene-1,2-dicarboxylimidyl Containing oxadiazole and Benzothiazole |
| title_fullStr | Synthesis, Characterization and study biologicalactivity of several 1-cyclopentene-1,2-dicarboxylimidyl Containing oxadiazole and Benzothiazole |
| title_full_unstemmed | Synthesis, Characterization and study biologicalactivity of several 1-cyclopentene-1,2-dicarboxylimidyl Containing oxadiazole and Benzothiazole |
| title_short | Synthesis, Characterization and study biologicalactivity of several 1-cyclopentene-1,2-dicarboxylimidyl Containing oxadiazole and Benzothiazole |
| title_sort | synthesis characterization and study biologicalactivity of several 1 cyclopentene 1 2 dicarboxylimidyl containing oxadiazole and benzothiazole |
| topic | 1-cyclopentene-1,2-dicarboxylimidyl, oxadiazol, benzothiazol. |
| url | http://bsj.uobaghdad.edu.iq/index.php/BSJ/article/view/2647 |
| work_keys_str_mv | AT baghdadsciencejournal synthesischaracterizationandstudybiologicalactivityofseveral1cyclopentene12dicarboxylimidylcontainingoxadiazoleandbenzothiazole |