Innovative evaluation of selinexor and JQ1 synergy in leukemia therapy via C-MYC inhibition

Abstract Background Acute myeloid leukemia (AML) remains a therapeutic challenge due to drug resistance and relapse. Selinexor, an XPO1 inhibitor, shows limited efficacy as monotherapy, necessitating combination strategies. JQ1, a BET inhibitor targeting MYC, may synergize with Selinexor to enhance...

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Bibliographic Details
Main Authors: Pei-Hong Wang, Chu-Hong Hu, Jia-Qi Fan, Jia-Jun He, Ting-Fen Deng, Yan-Li Xu, Yu-Jun Dai, Shun-Qing Wang
Format: Article
Language:English
Published: BMC 2025-05-01
Series:Journal of Translational Medicine
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Online Access:https://doi.org/10.1186/s12967-025-06525-z
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