Osthole: A Coumarin with Dual Roles in Biology and Chemistry

Osthole is a natural coumarin-like compound isolated from the <i>Fructus cnidii</i>. In the last few years, this plant-derived product and its derivatives have aroused much attention for their interesting biological activities, including anticancer, anti-inflammatory, neuroprotective, an...

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Bibliographic Details
Main Authors: Min Lv, Haixia Ding, Hui Xu
Format: Article
Language:English
Published: MDPI AG 2025-05-01
Series:Biology
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Online Access:https://www.mdpi.com/2079-7737/14/6/588
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Summary:Osthole is a natural coumarin-like compound isolated from the <i>Fructus cnidii</i>. In the last few years, this plant-derived product and its derivatives have aroused much attention for their interesting biological activities, including anticancer, anti-inflammatory, neuroprotective, and insecticidal effects. This review summarizes the recent progress on the biological activities of osthole and its derivatives from 2018 to early 2025, with a focus on their total synthesis, structural modifications, and mechanisms of action. Additionally, structure–activity relationships (SARs) of osthole derivatives are presented. This review aims to serve as a comprehensive reference for future research on osthole and its derivatives in both medicinal and agricultural applications.
ISSN:2079-7737