Structure and neutralization mechanism of a human antibody targeting a complex Epitope on Zika virus.

We currently have an incomplete understanding of why only a fraction of human antibodies that bind to flaviviruses block infection of cells. Here we define the footprint of a strongly neutralizing human monoclonal antibody (mAb G9E) with Zika virus (ZIKV) by both X-ray crystallography and cryo-elect...

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Main Authors: Cameron Adams, Derek L Carbaugh, Bo Shu, Thiam-Seng Ng, Izabella N Castillo, Ryan Bhowmik, Bruno Segovia-Chumbez, Ana C Puhl, Stephen Graham, Sean A Diehl, Helen M Lazear, Shee-Mei Lok, Aravinda M de Silva, Lakshmanane Premkumar
Format: Article
Language:English
Published: Public Library of Science (PLoS) 2023-01-01
Series:PLoS Pathogens
Online Access:https://journals.plos.org/plospathogens/article/file?id=10.1371/journal.ppat.1010814&type=printable
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author Cameron Adams
Derek L Carbaugh
Bo Shu
Thiam-Seng Ng
Izabella N Castillo
Ryan Bhowmik
Bruno Segovia-Chumbez
Ana C Puhl
Stephen Graham
Sean A Diehl
Helen M Lazear
Shee-Mei Lok
Aravinda M de Silva
Lakshmanane Premkumar
author_facet Cameron Adams
Derek L Carbaugh
Bo Shu
Thiam-Seng Ng
Izabella N Castillo
Ryan Bhowmik
Bruno Segovia-Chumbez
Ana C Puhl
Stephen Graham
Sean A Diehl
Helen M Lazear
Shee-Mei Lok
Aravinda M de Silva
Lakshmanane Premkumar
author_sort Cameron Adams
collection DOAJ
description We currently have an incomplete understanding of why only a fraction of human antibodies that bind to flaviviruses block infection of cells. Here we define the footprint of a strongly neutralizing human monoclonal antibody (mAb G9E) with Zika virus (ZIKV) by both X-ray crystallography and cryo-electron microscopy. Flavivirus envelope (E) glycoproteins are present as homodimers on the virion surface, and G9E bound to a quaternary structure epitope spanning both E protomers forming a homodimer. As G9E mainly neutralized ZIKV by blocking a step after viral attachment to cells, we tested if the neutralization mechanism of G9E was dependent on the mAb cross-linking E molecules and blocking low-pH triggered conformational changes required for viral membrane fusion. We introduced targeted mutations to the G9E paratope to create recombinant antibodies that bound to the ZIKV envelope without cross-linking E protomers. The G9E paratope mutants that bound to a restricted epitope on one protomer poorly neutralized ZIKV compared to the wild-type mAb, demonstrating that the neutralization mechanism depended on the ability of G9E to cross-link E proteins. In cell-free low pH triggered viral fusion assay, both wild-type G9E, and epitope restricted paratope mutant G9E bound to ZIKV but only the wild-type G9E blocked fusion. We propose that, beyond antibody binding strength, the ability of human antibodies to cross-link E-proteins is a critical determinant of flavivirus neutralization potency.
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spelling doaj-art-470ce3319ca643cab15d968be35cdd932025-08-20T03:08:32ZengPublic Library of Science (PLoS)PLoS Pathogens1553-73661553-73742023-01-01191e101081410.1371/journal.ppat.1010814Structure and neutralization mechanism of a human antibody targeting a complex Epitope on Zika virus.Cameron AdamsDerek L CarbaughBo ShuThiam-Seng NgIzabella N CastilloRyan BhowmikBruno Segovia-ChumbezAna C PuhlStephen GrahamSean A DiehlHelen M LazearShee-Mei LokAravinda M de SilvaLakshmanane PremkumarWe currently have an incomplete understanding of why only a fraction of human antibodies that bind to flaviviruses block infection of cells. Here we define the footprint of a strongly neutralizing human monoclonal antibody (mAb G9E) with Zika virus (ZIKV) by both X-ray crystallography and cryo-electron microscopy. Flavivirus envelope (E) glycoproteins are present as homodimers on the virion surface, and G9E bound to a quaternary structure epitope spanning both E protomers forming a homodimer. As G9E mainly neutralized ZIKV by blocking a step after viral attachment to cells, we tested if the neutralization mechanism of G9E was dependent on the mAb cross-linking E molecules and blocking low-pH triggered conformational changes required for viral membrane fusion. We introduced targeted mutations to the G9E paratope to create recombinant antibodies that bound to the ZIKV envelope without cross-linking E protomers. The G9E paratope mutants that bound to a restricted epitope on one protomer poorly neutralized ZIKV compared to the wild-type mAb, demonstrating that the neutralization mechanism depended on the ability of G9E to cross-link E proteins. In cell-free low pH triggered viral fusion assay, both wild-type G9E, and epitope restricted paratope mutant G9E bound to ZIKV but only the wild-type G9E blocked fusion. We propose that, beyond antibody binding strength, the ability of human antibodies to cross-link E-proteins is a critical determinant of flavivirus neutralization potency.https://journals.plos.org/plospathogens/article/file?id=10.1371/journal.ppat.1010814&type=printable
spellingShingle Cameron Adams
Derek L Carbaugh
Bo Shu
Thiam-Seng Ng
Izabella N Castillo
Ryan Bhowmik
Bruno Segovia-Chumbez
Ana C Puhl
Stephen Graham
Sean A Diehl
Helen M Lazear
Shee-Mei Lok
Aravinda M de Silva
Lakshmanane Premkumar
Structure and neutralization mechanism of a human antibody targeting a complex Epitope on Zika virus.
PLoS Pathogens
title Structure and neutralization mechanism of a human antibody targeting a complex Epitope on Zika virus.
title_full Structure and neutralization mechanism of a human antibody targeting a complex Epitope on Zika virus.
title_fullStr Structure and neutralization mechanism of a human antibody targeting a complex Epitope on Zika virus.
title_full_unstemmed Structure and neutralization mechanism of a human antibody targeting a complex Epitope on Zika virus.
title_short Structure and neutralization mechanism of a human antibody targeting a complex Epitope on Zika virus.
title_sort structure and neutralization mechanism of a human antibody targeting a complex epitope on zika virus
url https://journals.plos.org/plospathogens/article/file?id=10.1371/journal.ppat.1010814&type=printable
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