The DRN-VLO pathway via distinct 5-HT synaptic mechanisms modulates neuropathic pain–induced depressive-like behaviors in mice

Abstract Background The neuronal activities within the dorsal raphe nucleus (DRN) and the ventrolateral orbital cortex (VLO) are strongly implicated in the development of depression, a condition comorbid with chronic pain. The goal of the present study was to determine whether and how the DRN-VLO pa...

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Main Authors: Hai-Yan Sheng, Wei-Zhen Liu, Yan-Kai Liu, Qing-Rong Han, Dong-Yang Chen, Li-Bin Zhang, Xin-Ru Chu, Si-Han He, Jia-Xin Li, Zi-Qing Zhang, Bo-Han Duanmu, Ya-Ling Yin, Lin-Hua Jiang
Format: Article
Language:English
Published: BMC 2025-07-01
Series:The Journal of Headache and Pain
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Online Access:https://doi.org/10.1186/s10194-025-02110-3
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author Hai-Yan Sheng
Wei-Zhen Liu
Yan-Kai Liu
Qing-Rong Han
Dong-Yang Chen
Li-Bin Zhang
Xin-Ru Chu
Si-Han He
Jia-Xin Li
Zi-Qing Zhang
Bo-Han Duanmu
Ya-Ling Yin
Lin-Hua Jiang
author_facet Hai-Yan Sheng
Wei-Zhen Liu
Yan-Kai Liu
Qing-Rong Han
Dong-Yang Chen
Li-Bin Zhang
Xin-Ru Chu
Si-Han He
Jia-Xin Li
Zi-Qing Zhang
Bo-Han Duanmu
Ya-Ling Yin
Lin-Hua Jiang
author_sort Hai-Yan Sheng
collection DOAJ
description Abstract Background The neuronal activities within the dorsal raphe nucleus (DRN) and the ventrolateral orbital cortex (VLO) are strongly implicated in the development of depression, a condition comorbid with chronic pain. The goal of the present study was to determine whether and how the DRN-VLO pathway mediates chronic pain-induced depression. Methods Trigeminal neuralgia was induced unilaterally by chronic constriction injury of the infraorbital nerve. Depressive-like behaviors were assessed by the open field test, forced swimming test and tail suspension test. Neuronal projection tracing, chemogenetic manipulations and pharmacological interventions were performed to determine the DRN-VLO pathway projection activity and pathway-mediated anti-depressant mechanism in mice with trigeminal neuralgia. The neuronal activity was assessed by measuring the c-Fos level using immunofluorescence imaging. Results The VLO receives direct projection of the serotonergic neurons from the DRN. Anterograde or retrograde activation of the DRN-VLO pathway consistently produced anti-depressant effects in mice with neuropathic pain, whereas sustained inhibition of this pathway in healthy mice induced depressive-like behaviors. Activation of the 5-HT1A or 5-HT2A receptor in the VLO produced anti-depressant effects. Activation of the GABAA receptors in the VLO weakened 5-HT1A receptor-mediated anti-depressant effect. Conclusions The present study has revealed that activation of the DRN-VLO pathway exerts an anti-depressant effect in mice with neuropathic pain, through stimulating the 5-HT2A receptors in the excitatory neurons and also the 5-HT1A receptors in the GABAergic interneurons via a dis-inhibition mechanism, to enhance neuronal activity of the VLO.
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issn 1129-2377
language English
publishDate 2025-07-01
publisher BMC
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series The Journal of Headache and Pain
spelling doaj-art-46ed83e4d25a403bbd5d2a31990cec732025-08-20T03:46:25ZengBMCThe Journal of Headache and Pain1129-23772025-07-0126111710.1186/s10194-025-02110-3The DRN-VLO pathway via distinct 5-HT synaptic mechanisms modulates neuropathic pain–induced depressive-like behaviors in miceHai-Yan Sheng0Wei-Zhen Liu1Yan-Kai Liu2Qing-Rong Han3Dong-Yang Chen4Li-Bin Zhang5Xin-Ru Chu6Si-Han He7Jia-Xin Li8Zi-Qing Zhang9Bo-Han Duanmu10Ya-Ling Yin11Lin-Hua Jiang12Sino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversitySino-UK Joint Laboratory of Brain Function and Injury of Henan Province, Department of Physiology and Pathophysiology, School of Basic Medical Sciences, Xinxiang Medical UniversityAbstract Background The neuronal activities within the dorsal raphe nucleus (DRN) and the ventrolateral orbital cortex (VLO) are strongly implicated in the development of depression, a condition comorbid with chronic pain. The goal of the present study was to determine whether and how the DRN-VLO pathway mediates chronic pain-induced depression. Methods Trigeminal neuralgia was induced unilaterally by chronic constriction injury of the infraorbital nerve. Depressive-like behaviors were assessed by the open field test, forced swimming test and tail suspension test. Neuronal projection tracing, chemogenetic manipulations and pharmacological interventions were performed to determine the DRN-VLO pathway projection activity and pathway-mediated anti-depressant mechanism in mice with trigeminal neuralgia. The neuronal activity was assessed by measuring the c-Fos level using immunofluorescence imaging. Results The VLO receives direct projection of the serotonergic neurons from the DRN. Anterograde or retrograde activation of the DRN-VLO pathway consistently produced anti-depressant effects in mice with neuropathic pain, whereas sustained inhibition of this pathway in healthy mice induced depressive-like behaviors. Activation of the 5-HT1A or 5-HT2A receptor in the VLO produced anti-depressant effects. Activation of the GABAA receptors in the VLO weakened 5-HT1A receptor-mediated anti-depressant effect. Conclusions The present study has revealed that activation of the DRN-VLO pathway exerts an anti-depressant effect in mice with neuropathic pain, through stimulating the 5-HT2A receptors in the excitatory neurons and also the 5-HT1A receptors in the GABAergic interneurons via a dis-inhibition mechanism, to enhance neuronal activity of the VLO.https://doi.org/10.1186/s10194-025-02110-3Neuropathic painDepressionDRN-VLO pathway5-HT1A/5-HT2A receptorsGABAA receptor
spellingShingle Hai-Yan Sheng
Wei-Zhen Liu
Yan-Kai Liu
Qing-Rong Han
Dong-Yang Chen
Li-Bin Zhang
Xin-Ru Chu
Si-Han He
Jia-Xin Li
Zi-Qing Zhang
Bo-Han Duanmu
Ya-Ling Yin
Lin-Hua Jiang
The DRN-VLO pathway via distinct 5-HT synaptic mechanisms modulates neuropathic pain–induced depressive-like behaviors in mice
The Journal of Headache and Pain
Neuropathic pain
Depression
DRN-VLO pathway
5-HT1A/5-HT2A receptors
GABAA receptor
title The DRN-VLO pathway via distinct 5-HT synaptic mechanisms modulates neuropathic pain–induced depressive-like behaviors in mice
title_full The DRN-VLO pathway via distinct 5-HT synaptic mechanisms modulates neuropathic pain–induced depressive-like behaviors in mice
title_fullStr The DRN-VLO pathway via distinct 5-HT synaptic mechanisms modulates neuropathic pain–induced depressive-like behaviors in mice
title_full_unstemmed The DRN-VLO pathway via distinct 5-HT synaptic mechanisms modulates neuropathic pain–induced depressive-like behaviors in mice
title_short The DRN-VLO pathway via distinct 5-HT synaptic mechanisms modulates neuropathic pain–induced depressive-like behaviors in mice
title_sort drn vlo pathway via distinct 5 ht synaptic mechanisms modulates neuropathic pain induced depressive like behaviors in mice
topic Neuropathic pain
Depression
DRN-VLO pathway
5-HT1A/5-HT2A receptors
GABAA receptor
url https://doi.org/10.1186/s10194-025-02110-3
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