Statins and their impact on epigenetic regulation: insights into disease

Statins have been primarily used for the management of low-density lipoprotein cholesterol and cardiovascular diseases However, in recent years, research has identified potential applications beyond cholesterol regulation. Statins exhibit pleiotropic effects, due to their ability to modulate gene ex...

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Main Authors: Rafael Tamayo-Trujillo, Patricia Guevara-Ramírez, Santiago Cadena-Ullauri, Viviana A. Ruiz Pozo, Elius Paz-Cruz, Ana Karina Zambrano
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-07-01
Series:Frontiers in Pharmacology
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Online Access:https://www.frontiersin.org/articles/10.3389/fphar.2025.1621163/full
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author Rafael Tamayo-Trujillo
Patricia Guevara-Ramírez
Santiago Cadena-Ullauri
Viviana A. Ruiz Pozo
Elius Paz-Cruz
Ana Karina Zambrano
author_facet Rafael Tamayo-Trujillo
Patricia Guevara-Ramírez
Santiago Cadena-Ullauri
Viviana A. Ruiz Pozo
Elius Paz-Cruz
Ana Karina Zambrano
author_sort Rafael Tamayo-Trujillo
collection DOAJ
description Statins have been primarily used for the management of low-density lipoprotein cholesterol and cardiovascular diseases However, in recent years, research has identified potential applications beyond cholesterol regulation. Statins exhibit pleiotropic effects, due to their ability to modulate gene expression via epigenetic mechanisms, including DNA methylation, histone acetylation, and microRNA regulation. Clinical studies have correlated these epigenetic changes with various pathological conditions, such as inflammation, atherosclerosis, cancer, diabetes, and autoimmune disorders. Despite encouraging findings, further research is required to fully understand the molecular pathways associated with the epigenetic actions of statins and disease pathogenesis. This review describes the potential role of statins as epigenetic modulators and their relevance in human disease management.
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publisher Frontiers Media S.A.
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spelling doaj-art-449bf2fd1f8f43a4805c3ef0f5290fe52025-08-20T03:51:02ZengFrontiers Media S.A.Frontiers in Pharmacology1663-98122025-07-011610.3389/fphar.2025.16211631621163Statins and their impact on epigenetic regulation: insights into diseaseRafael Tamayo-TrujilloPatricia Guevara-RamírezSantiago Cadena-UllauriViviana A. Ruiz PozoElius Paz-CruzAna Karina ZambranoStatins have been primarily used for the management of low-density lipoprotein cholesterol and cardiovascular diseases However, in recent years, research has identified potential applications beyond cholesterol regulation. Statins exhibit pleiotropic effects, due to their ability to modulate gene expression via epigenetic mechanisms, including DNA methylation, histone acetylation, and microRNA regulation. Clinical studies have correlated these epigenetic changes with various pathological conditions, such as inflammation, atherosclerosis, cancer, diabetes, and autoimmune disorders. Despite encouraging findings, further research is required to fully understand the molecular pathways associated with the epigenetic actions of statins and disease pathogenesis. This review describes the potential role of statins as epigenetic modulators and their relevance in human disease management.https://www.frontiersin.org/articles/10.3389/fphar.2025.1621163/fullpharmacologypharmacoepigeneticsepigeneticsstatinsmolecular biologyhealthcare and well-being
spellingShingle Rafael Tamayo-Trujillo
Patricia Guevara-Ramírez
Santiago Cadena-Ullauri
Viviana A. Ruiz Pozo
Elius Paz-Cruz
Ana Karina Zambrano
Statins and their impact on epigenetic regulation: insights into disease
Frontiers in Pharmacology
pharmacology
pharmacoepigenetics
epigenetics
statins
molecular biology
healthcare and well-being
title Statins and their impact on epigenetic regulation: insights into disease
title_full Statins and their impact on epigenetic regulation: insights into disease
title_fullStr Statins and their impact on epigenetic regulation: insights into disease
title_full_unstemmed Statins and their impact on epigenetic regulation: insights into disease
title_short Statins and their impact on epigenetic regulation: insights into disease
title_sort statins and their impact on epigenetic regulation insights into disease
topic pharmacology
pharmacoepigenetics
epigenetics
statins
molecular biology
healthcare and well-being
url https://www.frontiersin.org/articles/10.3389/fphar.2025.1621163/full
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