A quantitative characterization of the heterogeneous response of glioblastoma U-87 MG cell line to temozolomide

Abstract Most cancers are genetically and phenotypically heterogeneous. This includes subpopulations of cells with different levels of sensitivity to chemotherapy, which may lead to treatment failure as the more resistant cells can survive drug treatment and continue to proliferate. While the geneti...

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Main Authors: Pragyesh Dixit, Ilyas Djafer-Cherif, Saumil Shah, Karolina Drabik, Arne Traulsen, Bartlomiej Waclaw
Format: Article
Language:English
Published: Nature Portfolio 2025-05-01
Series:Scientific Reports
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Online Access:https://doi.org/10.1038/s41598-025-99426-6
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author Pragyesh Dixit
Ilyas Djafer-Cherif
Saumil Shah
Karolina Drabik
Arne Traulsen
Bartlomiej Waclaw
author_facet Pragyesh Dixit
Ilyas Djafer-Cherif
Saumil Shah
Karolina Drabik
Arne Traulsen
Bartlomiej Waclaw
author_sort Pragyesh Dixit
collection DOAJ
description Abstract Most cancers are genetically and phenotypically heterogeneous. This includes subpopulations of cells with different levels of sensitivity to chemotherapy, which may lead to treatment failure as the more resistant cells can survive drug treatment and continue to proliferate. While the genetic basis of resistance to many drugs is relatively well characterised, non-genetic factors are much less understood. Here we investigate the role of non-genetic, phenotypic heterogeneity in the response of glioblastoma cancer cells to the drug temozolomide (TMZ) often used to treat this type of cancer. Using a combination of live imaging, machine-learning image analysis and agent-based modelling, we show that even if all cells share the same genetic background, individual cells respond differently to TMZ. We quantitatively characterise this response by measuring the doubling time, lifespan, cell cycle phase, area and motility of cells, and determine how these quantities correlate with each other as well as between the mother and daughter cell. We also show that these responses do not correlate with the cellular level of the enzyme MGMT which has been implicated in the response to TMZ.
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spelling doaj-art-446fd3612ba04a01be8c277e23bcb9ef2025-08-20T01:49:39ZengNature PortfolioScientific Reports2045-23222025-05-0115111310.1038/s41598-025-99426-6A quantitative characterization of the heterogeneous response of glioblastoma U-87 MG cell line to temozolomidePragyesh Dixit0Ilyas Djafer-Cherif1Saumil Shah2Karolina Drabik3Arne Traulsen4Bartlomiej Waclaw5Dioscuri Centre for Physics and Chemistry of Bacteria, Institute of Physical Chemistry, Polish Academy of SciencesDioscuri Centre for Physics and Chemistry of Bacteria, Institute of Physical Chemistry, Polish Academy of SciencesDepartment of Theoretical Biology, Max Planck Institute for Evolutionary BiologyDioscuri Centre for Physics and Chemistry of Bacteria, Institute of Physical Chemistry, Polish Academy of SciencesDepartment of Theoretical Biology, Max Planck Institute for Evolutionary BiologyDioscuri Centre for Physics and Chemistry of Bacteria, Institute of Physical Chemistry, Polish Academy of SciencesAbstract Most cancers are genetically and phenotypically heterogeneous. This includes subpopulations of cells with different levels of sensitivity to chemotherapy, which may lead to treatment failure as the more resistant cells can survive drug treatment and continue to proliferate. While the genetic basis of resistance to many drugs is relatively well characterised, non-genetic factors are much less understood. Here we investigate the role of non-genetic, phenotypic heterogeneity in the response of glioblastoma cancer cells to the drug temozolomide (TMZ) often used to treat this type of cancer. Using a combination of live imaging, machine-learning image analysis and agent-based modelling, we show that even if all cells share the same genetic background, individual cells respond differently to TMZ. We quantitatively characterise this response by measuring the doubling time, lifespan, cell cycle phase, area and motility of cells, and determine how these quantities correlate with each other as well as between the mother and daughter cell. We also show that these responses do not correlate with the cellular level of the enzyme MGMT which has been implicated in the response to TMZ.https://doi.org/10.1038/s41598-025-99426-6CancerGlioblastomaTemozolomidePhenotypic heterogeneityMathematical modelling
spellingShingle Pragyesh Dixit
Ilyas Djafer-Cherif
Saumil Shah
Karolina Drabik
Arne Traulsen
Bartlomiej Waclaw
A quantitative characterization of the heterogeneous response of glioblastoma U-87 MG cell line to temozolomide
Scientific Reports
Cancer
Glioblastoma
Temozolomide
Phenotypic heterogeneity
Mathematical modelling
title A quantitative characterization of the heterogeneous response of glioblastoma U-87 MG cell line to temozolomide
title_full A quantitative characterization of the heterogeneous response of glioblastoma U-87 MG cell line to temozolomide
title_fullStr A quantitative characterization of the heterogeneous response of glioblastoma U-87 MG cell line to temozolomide
title_full_unstemmed A quantitative characterization of the heterogeneous response of glioblastoma U-87 MG cell line to temozolomide
title_short A quantitative characterization of the heterogeneous response of glioblastoma U-87 MG cell line to temozolomide
title_sort quantitative characterization of the heterogeneous response of glioblastoma u 87 mg cell line to temozolomide
topic Cancer
Glioblastoma
Temozolomide
Phenotypic heterogeneity
Mathematical modelling
url https://doi.org/10.1038/s41598-025-99426-6
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