CAF-mediated regulation of prostate cancer stem cell stemness via the Wnt/β-catenin and SDF-1/CXCR4 pathways in castration-resistant prostate cancer

IntroductionThe role of cancer-associated fibroblasts (CAFs) in the progression, therapeutic resistance, and metastasis of castration-resistant prostate cancer (CRPC) remains incompletely understood. This study aimed to investigate how CAFs regulate the stemness of prostate cancer stem cells (PCSCs)...

Full description

Saved in:
Bibliographic Details
Main Authors: Haoran Chen, Zhen Li, Yuan Yue, Xudong Zhu, Jiazheng Wang, Yafei Chen, Yilin Wang, Zhanyang Luo, Hao Liu
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-07-01
Series:Frontiers in Cell and Developmental Biology
Subjects:
Online Access:https://www.frontiersin.org/articles/10.3389/fcell.2025.1617200/full
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849432425998843904
author Haoran Chen
Zhen Li
Yuan Yue
Xudong Zhu
Jiazheng Wang
Yafei Chen
Yilin Wang
Zhanyang Luo
Hao Liu
author_facet Haoran Chen
Zhen Li
Yuan Yue
Xudong Zhu
Jiazheng Wang
Yafei Chen
Yilin Wang
Zhanyang Luo
Hao Liu
author_sort Haoran Chen
collection DOAJ
description IntroductionThe role of cancer-associated fibroblasts (CAFs) in the progression, therapeutic resistance, and metastasis of castration-resistant prostate cancer (CRPC) remains incompletely understood. This study aimed to investigate how CAFs regulate the stemness of prostate cancer stem cells (PCSCs), with a focus on the Wnt/β-catenin and SDF-1/CXCR4 signaling pathways.MethodsWe assessed the expression of CAF and PCSC markers in xenograft tumor tissues from hormone-sensitive prostate cancer and CRPC mouse models using immunohistochemistry and immunofluorescence. The impact of CAFs on stemness markers, SDF-1, CXCR4, and Wnt pathway activation was evaluated both in vitro and in vivo.ResultsThe expression levels of CAF and PCSC markers were significantly elevated in CRPC tissues compared to hormone-sensitive tumors. Bioinformatics analysis indicated high expression of CXCR4 and CTNNB1 (β-catenin) in CRPC, with positive correlations to disease progression. CAFs enhanced PCSC stemness, while inhibition of Wnt3a or SDF-1 led to reduced stemness and pathway activity. In vivo, CAFs promoted CRPC tumor growth and significantly increased the expression of Wnt3a, β-catenin, TCF4, LEF1, SDF-1, and CXCR4, along with an elevated p-GSK-3β/GSK-3β ratio. Conversely, β-catenin and CXCR4 inhibitors suppressed tumor growth and downregulated Wnt signaling components.Discussionβ-Catenin and CXCR4 showed strong co-localization in xenograft tumors. These findings suggest that CAFs promote PCSC stemness and CRPC progression by activating the Wnt/β-catenin and SDF-1/CXCR4 pathways via Wnt3a and SDF-1 expression. These insights provide potential targets for managing CRPC.
format Article
id doaj-art-421ddc5ba5484f09b2027bd29b5b039b
institution Kabale University
issn 2296-634X
language English
publishDate 2025-07-01
publisher Frontiers Media S.A.
record_format Article
series Frontiers in Cell and Developmental Biology
spelling doaj-art-421ddc5ba5484f09b2027bd29b5b039b2025-08-20T03:27:22ZengFrontiers Media S.A.Frontiers in Cell and Developmental Biology2296-634X2025-07-011310.3389/fcell.2025.16172001617200CAF-mediated regulation of prostate cancer stem cell stemness via the Wnt/β-catenin and SDF-1/CXCR4 pathways in castration-resistant prostate cancerHaoran Chen0Zhen Li1Yuan Yue2Xudong Zhu3Jiazheng Wang4Yafei Chen5Yilin Wang6Zhanyang Luo7Hao Liu8Guang’anmen Hospital, China Academy of Chinese Medical Sciences, Beijing, ChinaCollege of Traditional Chinese Medicine, Anhui University of Chinese Medicine, Hefei, Anhui, ChinaThe Affiliated Hospital of Southwest Medical University, Luzhou, Sichuan, ChinaGuang’anmen Hospital, China Academy of Chinese Medical Sciences, Beijing, ChinaGuang’anmen Hospital, China Academy of Chinese Medical Sciences, Beijing, ChinaGraduate School, Beijing University of Chinese Medicine, Beijing, ChinaGraduate School, Beijing University of Chinese Medicine, Beijing, ChinaShanghai Pudong Hospital, Fudan University Pudong Medical Center, Shanghai, ChinaGuang’anmen Hospital, China Academy of Chinese Medical Sciences, Beijing, ChinaIntroductionThe role of cancer-associated fibroblasts (CAFs) in the progression, therapeutic resistance, and metastasis of castration-resistant prostate cancer (CRPC) remains incompletely understood. This study aimed to investigate how CAFs regulate the stemness of prostate cancer stem cells (PCSCs), with a focus on the Wnt/β-catenin and SDF-1/CXCR4 signaling pathways.MethodsWe assessed the expression of CAF and PCSC markers in xenograft tumor tissues from hormone-sensitive prostate cancer and CRPC mouse models using immunohistochemistry and immunofluorescence. The impact of CAFs on stemness markers, SDF-1, CXCR4, and Wnt pathway activation was evaluated both in vitro and in vivo.ResultsThe expression levels of CAF and PCSC markers were significantly elevated in CRPC tissues compared to hormone-sensitive tumors. Bioinformatics analysis indicated high expression of CXCR4 and CTNNB1 (β-catenin) in CRPC, with positive correlations to disease progression. CAFs enhanced PCSC stemness, while inhibition of Wnt3a or SDF-1 led to reduced stemness and pathway activity. In vivo, CAFs promoted CRPC tumor growth and significantly increased the expression of Wnt3a, β-catenin, TCF4, LEF1, SDF-1, and CXCR4, along with an elevated p-GSK-3β/GSK-3β ratio. Conversely, β-catenin and CXCR4 inhibitors suppressed tumor growth and downregulated Wnt signaling components.Discussionβ-Catenin and CXCR4 showed strong co-localization in xenograft tumors. These findings suggest that CAFs promote PCSC stemness and CRPC progression by activating the Wnt/β-catenin and SDF-1/CXCR4 pathways via Wnt3a and SDF-1 expression. These insights provide potential targets for managing CRPC.https://www.frontiersin.org/articles/10.3389/fcell.2025.1617200/fullcastration-resistant prostate cancercancer-associated fibroblastprostate cancer stem cellWnt/β-cateninSDF-1/CXCR4
spellingShingle Haoran Chen
Zhen Li
Yuan Yue
Xudong Zhu
Jiazheng Wang
Yafei Chen
Yilin Wang
Zhanyang Luo
Hao Liu
CAF-mediated regulation of prostate cancer stem cell stemness via the Wnt/β-catenin and SDF-1/CXCR4 pathways in castration-resistant prostate cancer
Frontiers in Cell and Developmental Biology
castration-resistant prostate cancer
cancer-associated fibroblast
prostate cancer stem cell
Wnt/β-catenin
SDF-1/CXCR4
title CAF-mediated regulation of prostate cancer stem cell stemness via the Wnt/β-catenin and SDF-1/CXCR4 pathways in castration-resistant prostate cancer
title_full CAF-mediated regulation of prostate cancer stem cell stemness via the Wnt/β-catenin and SDF-1/CXCR4 pathways in castration-resistant prostate cancer
title_fullStr CAF-mediated regulation of prostate cancer stem cell stemness via the Wnt/β-catenin and SDF-1/CXCR4 pathways in castration-resistant prostate cancer
title_full_unstemmed CAF-mediated regulation of prostate cancer stem cell stemness via the Wnt/β-catenin and SDF-1/CXCR4 pathways in castration-resistant prostate cancer
title_short CAF-mediated regulation of prostate cancer stem cell stemness via the Wnt/β-catenin and SDF-1/CXCR4 pathways in castration-resistant prostate cancer
title_sort caf mediated regulation of prostate cancer stem cell stemness via the wnt β catenin and sdf 1 cxcr4 pathways in castration resistant prostate cancer
topic castration-resistant prostate cancer
cancer-associated fibroblast
prostate cancer stem cell
Wnt/β-catenin
SDF-1/CXCR4
url https://www.frontiersin.org/articles/10.3389/fcell.2025.1617200/full
work_keys_str_mv AT haoranchen cafmediatedregulationofprostatecancerstemcellstemnessviathewntbcateninandsdf1cxcr4pathwaysincastrationresistantprostatecancer
AT zhenli cafmediatedregulationofprostatecancerstemcellstemnessviathewntbcateninandsdf1cxcr4pathwaysincastrationresistantprostatecancer
AT yuanyue cafmediatedregulationofprostatecancerstemcellstemnessviathewntbcateninandsdf1cxcr4pathwaysincastrationresistantprostatecancer
AT xudongzhu cafmediatedregulationofprostatecancerstemcellstemnessviathewntbcateninandsdf1cxcr4pathwaysincastrationresistantprostatecancer
AT jiazhengwang cafmediatedregulationofprostatecancerstemcellstemnessviathewntbcateninandsdf1cxcr4pathwaysincastrationresistantprostatecancer
AT yafeichen cafmediatedregulationofprostatecancerstemcellstemnessviathewntbcateninandsdf1cxcr4pathwaysincastrationresistantprostatecancer
AT yilinwang cafmediatedregulationofprostatecancerstemcellstemnessviathewntbcateninandsdf1cxcr4pathwaysincastrationresistantprostatecancer
AT zhanyangluo cafmediatedregulationofprostatecancerstemcellstemnessviathewntbcateninandsdf1cxcr4pathwaysincastrationresistantprostatecancer
AT haoliu cafmediatedregulationofprostatecancerstemcellstemnessviathewntbcateninandsdf1cxcr4pathwaysincastrationresistantprostatecancer