Synthesis and antibacterial activity of some new 3-hydroxy-2-naphthoic acid hydrazide derivatives for dyeing polyester fabrics
Dibenzobarallene was used as a key intermediate for the synthesis of 2-(3-hydroxy-2-naphthoyl)-3,4,4a,5,10,10a-hexahydro-1H-5,10-benzenobenzo[g]phthalazine-1,4-dione (2). The previous compound was coupled with the appropriate diazonium chloride to give the corresponding 4-arylazo-2-naphthol derivati...
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| Language: | English |
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2016-03-01
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| Series: | Journal of Saudi Chemical Society |
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| Online Access: | http://www.sciencedirect.com/science/article/pii/S131961031200083X |
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| author | Abd El-Galil M. Khalil Moged A. Berghot Moustafa A. Gouda |
| author_facet | Abd El-Galil M. Khalil Moged A. Berghot Moustafa A. Gouda |
| author_sort | Abd El-Galil M. Khalil |
| collection | DOAJ |
| description | Dibenzobarallene was used as a key intermediate for the synthesis of 2-(3-hydroxy-2-naphthoyl)-3,4,4a,5,10,10a-hexahydro-1H-5,10-benzenobenzo[g]phthalazine-1,4-dione (2). The previous compound was coupled with the appropriate diazonium chloride to give the corresponding 4-arylazo-2-naphthol derivatives 3a–l. Also, nitration, nitrosation and bromination of compound 2 afforded the corresponding nitro, nitroso and bromo derivatives 4–6, respectively. The synthesized compounds were established and evaluated as antibacterial agents. The results showed clearly that compounds 2, 3a, 3c, 3d, 3g, 3i, 4, 5 and 6 exhibited interesting high activities compared with reference drugs. Also, these compounds were applied to polyester as disperse dyes in which their color measurement and fastness properties were evaluated. |
| format | Article |
| id | doaj-art-3fb08bcccda645b6af5213157cf90fd9 |
| institution | Kabale University |
| issn | 1319-6103 |
| language | English |
| publishDate | 2016-03-01 |
| publisher | Springer |
| record_format | Article |
| series | Journal of Saudi Chemical Society |
| spelling | doaj-art-3fb08bcccda645b6af5213157cf90fd92025-08-20T03:52:25ZengSpringerJournal of Saudi Chemical Society1319-61032016-03-0120216517210.1016/j.jscs.2012.06.007Synthesis and antibacterial activity of some new 3-hydroxy-2-naphthoic acid hydrazide derivatives for dyeing polyester fabricsAbd El-Galil M. KhalilMoged A. BerghotMoustafa A. GoudaDibenzobarallene was used as a key intermediate for the synthesis of 2-(3-hydroxy-2-naphthoyl)-3,4,4a,5,10,10a-hexahydro-1H-5,10-benzenobenzo[g]phthalazine-1,4-dione (2). The previous compound was coupled with the appropriate diazonium chloride to give the corresponding 4-arylazo-2-naphthol derivatives 3a–l. Also, nitration, nitrosation and bromination of compound 2 afforded the corresponding nitro, nitroso and bromo derivatives 4–6, respectively. The synthesized compounds were established and evaluated as antibacterial agents. The results showed clearly that compounds 2, 3a, 3c, 3d, 3g, 3i, 4, 5 and 6 exhibited interesting high activities compared with reference drugs. Also, these compounds were applied to polyester as disperse dyes in which their color measurement and fastness properties were evaluated.http://www.sciencedirect.com/science/article/pii/S131961031200083XNaphthoic acid hydrazideNaphthol dyesPolyester fabricsAntibacterialColor measurementsFastness properties |
| spellingShingle | Abd El-Galil M. Khalil Moged A. Berghot Moustafa A. Gouda Synthesis and antibacterial activity of some new 3-hydroxy-2-naphthoic acid hydrazide derivatives for dyeing polyester fabrics Journal of Saudi Chemical Society Naphthoic acid hydrazide Naphthol dyes Polyester fabrics Antibacterial Color measurements Fastness properties |
| title | Synthesis and antibacterial activity of some new 3-hydroxy-2-naphthoic acid hydrazide derivatives for dyeing polyester fabrics |
| title_full | Synthesis and antibacterial activity of some new 3-hydroxy-2-naphthoic acid hydrazide derivatives for dyeing polyester fabrics |
| title_fullStr | Synthesis and antibacterial activity of some new 3-hydroxy-2-naphthoic acid hydrazide derivatives for dyeing polyester fabrics |
| title_full_unstemmed | Synthesis and antibacterial activity of some new 3-hydroxy-2-naphthoic acid hydrazide derivatives for dyeing polyester fabrics |
| title_short | Synthesis and antibacterial activity of some new 3-hydroxy-2-naphthoic acid hydrazide derivatives for dyeing polyester fabrics |
| title_sort | synthesis and antibacterial activity of some new 3 hydroxy 2 naphthoic acid hydrazide derivatives for dyeing polyester fabrics |
| topic | Naphthoic acid hydrazide Naphthol dyes Polyester fabrics Antibacterial Color measurements Fastness properties |
| url | http://www.sciencedirect.com/science/article/pii/S131961031200083X |
| work_keys_str_mv | AT abdelgalilmkhalil synthesisandantibacterialactivityofsomenew3hydroxy2naphthoicacidhydrazidederivativesfordyeingpolyesterfabrics AT mogedaberghot synthesisandantibacterialactivityofsomenew3hydroxy2naphthoicacidhydrazidederivativesfordyeingpolyesterfabrics AT moustafaagouda synthesisandantibacterialactivityofsomenew3hydroxy2naphthoicacidhydrazidederivativesfordyeingpolyesterfabrics |