Mathematical modeling of pharmacokinetics and pharmacodynamics of losartan in relation to CYP2C9 allele variants

Losartan is a selective angiotensin II AT1-receptor antagonist for the treatment of arterial hypertension and heart failure. It is converted to a pharmacologically active metabolite carboxylosartan (E-3174) in the liver mainly by CYP2C9 enzyme, a member of the cytochrome P450 superfamily. The gene e...

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Bibliographic Details
Main Authors: Dmitry Babaev, Elena Kutumova, Fedor Kolpakov
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-05-01
Series:Frontiers in Systems Biology
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Online Access:https://www.frontiersin.org/articles/10.3389/fsysb.2025.1504077/full
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