Pathogenesis of drug resistant epilepsy

Pharmacotherapy is the first-line treatment modality for epilepsy. However, in 20-40% of patients, epilepsy is resistant to pharmacotherapy. These numbers have not changed for decades despite the development and use of antiepileptic drugs with novel mechanisms of action. Drug-resistant epilepsy is n...

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Main Authors: S. M. Malyshev, T. M. Alekseeva, W. A. Khachatryan, M. M. Galagudza
Format: Article
Language:Russian
Published: IRBIS LLC 2019-04-01
Series:Эпилепсия и пароксизмальные состояния
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Online Access:https://www.epilepsia.su/jour/article/view/460
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author S. M. Malyshev
T. M. Alekseeva
W. A. Khachatryan
M. M. Galagudza
author_facet S. M. Malyshev
T. M. Alekseeva
W. A. Khachatryan
M. M. Galagudza
author_sort S. M. Malyshev
collection DOAJ
description Pharmacotherapy is the first-line treatment modality for epilepsy. However, in 20-40% of patients, epilepsy is resistant to pharmacotherapy. These numbers have not changed for decades despite the development and use of antiepileptic drugs with novel mechanisms of action. Drug-resistant epilepsy is now considered a separate pathophysiologic and clinical entity. The existing hypotheses on its pathogenesis could be divided in two groups. Firstly, drug-resistance might be caused by an abnormal pharmacokinetics or pharmacodynamics of antiepileptic drugs as a result of congenital or acquired dysfunction of the transporter or receptor proteins. Secondly, it might be a consequence of inherent features of epilepsy per se, such as the so-called “intrinsic severity” or some disorder of the connectome. Taking into account the complexity of this phenomenon, the issue of drug resistance continues to remain in the focus of the current research efforts.
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institution Kabale University
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publisher IRBIS LLC
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series Эпилепсия и пароксизмальные состояния
spelling doaj-art-3e516ade19504db7adfb6e05aa2509742025-08-20T03:39:32ZrusIRBIS LLCЭпилепсия и пароксизмальные состояния2077-83332311-40882019-04-01111798710.17749/2077-8333.2019.11.1.79-87436Pathogenesis of drug resistant epilepsyS. M. Malyshev0T. M. Alekseeva1W. A. Khachatryan2M. M. Galagudza3VA Almazov National Medical Research CenterVA Almazov National Medical Research CenterVA Almazov National Medical Research CenterVA Almazov National Medical Research CenterPharmacotherapy is the first-line treatment modality for epilepsy. However, in 20-40% of patients, epilepsy is resistant to pharmacotherapy. These numbers have not changed for decades despite the development and use of antiepileptic drugs with novel mechanisms of action. Drug-resistant epilepsy is now considered a separate pathophysiologic and clinical entity. The existing hypotheses on its pathogenesis could be divided in two groups. Firstly, drug-resistance might be caused by an abnormal pharmacokinetics or pharmacodynamics of antiepileptic drugs as a result of congenital or acquired dysfunction of the transporter or receptor proteins. Secondly, it might be a consequence of inherent features of epilepsy per se, such as the so-called “intrinsic severity” or some disorder of the connectome. Taking into account the complexity of this phenomenon, the issue of drug resistance continues to remain in the focus of the current research efforts.https://www.epilepsia.su/jour/article/view/460drug resistant epilepsyantiepileptic drugsconnectomicstranslational medicine
spellingShingle S. M. Malyshev
T. M. Alekseeva
W. A. Khachatryan
M. M. Galagudza
Pathogenesis of drug resistant epilepsy
Эпилепсия и пароксизмальные состояния
drug resistant epilepsy
antiepileptic drugs
connectomics
translational medicine
title Pathogenesis of drug resistant epilepsy
title_full Pathogenesis of drug resistant epilepsy
title_fullStr Pathogenesis of drug resistant epilepsy
title_full_unstemmed Pathogenesis of drug resistant epilepsy
title_short Pathogenesis of drug resistant epilepsy
title_sort pathogenesis of drug resistant epilepsy
topic drug resistant epilepsy
antiepileptic drugs
connectomics
translational medicine
url https://www.epilepsia.su/jour/article/view/460
work_keys_str_mv AT smmalyshev pathogenesisofdrugresistantepilepsy
AT tmalekseeva pathogenesisofdrugresistantepilepsy
AT wakhachatryan pathogenesisofdrugresistantepilepsy
AT mmgalagudza pathogenesisofdrugresistantepilepsy