Lysine crotonylation in disease: mechanisms, biological functions and therapeutic targets

Abstract Lysine crotonylation (Kcr), a previously unknown post-translational modification (PTM), plays crucial roles in regulating cellular processes, including gene expression, chromatin remodeling, and cellular metabolism. Kcr is associated with various diseases, including neurodegenerative disord...

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Main Authors: Yu Ji, Shanshan Liu, Yiqiao Zhang, Yiyang Min, Luyang Wei, Chengjian Guan, Huajing Yu, Zhongtao Zhang
Format: Article
Language:English
Published: BMC 2025-03-01
Series:Epigenetics & Chromatin
Online Access:https://doi.org/10.1186/s13072-025-00577-7
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author Yu Ji
Shanshan Liu
Yiqiao Zhang
Yiyang Min
Luyang Wei
Chengjian Guan
Huajing Yu
Zhongtao Zhang
author_facet Yu Ji
Shanshan Liu
Yiqiao Zhang
Yiyang Min
Luyang Wei
Chengjian Guan
Huajing Yu
Zhongtao Zhang
author_sort Yu Ji
collection DOAJ
description Abstract Lysine crotonylation (Kcr), a previously unknown post-translational modification (PTM), plays crucial roles in regulating cellular processes, including gene expression, chromatin remodeling, and cellular metabolism. Kcr is associated with various diseases, including neurodegenerative disorders, cancer, cardiovascular conditions, and metabolic syndromes. Despite advances in identifying crotonylation sites and their regulatory enzymes, the molecular mechanisms by which Kcr influences disease progression remain poorly understood. Understanding the interplay between Kcr and other acylation modifications may reveal opportunities for developing targeted therapies. This review synthesizes current research on Kcr, focusing on its regulatory mechanisms and disease associations, and highlights insights into future exploration in epigenetics and therapeutic interventions.
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institution Kabale University
issn 1756-8935
language English
publishDate 2025-03-01
publisher BMC
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series Epigenetics & Chromatin
spelling doaj-art-3c6d08becc744d87b04dde9ee11046b92025-08-20T03:41:50ZengBMCEpigenetics & Chromatin1756-89352025-03-0118112210.1186/s13072-025-00577-7Lysine crotonylation in disease: mechanisms, biological functions and therapeutic targetsYu Ji0Shanshan Liu1Yiqiao Zhang2Yiyang Min3Luyang Wei4Chengjian Guan5Huajing Yu6Zhongtao Zhang7Department of General Surgery, Beijing Friendship Hospital, Capital Medical University & State Key Lab of Digestive Health & National Clinical Research Center for Digestive DiseasesDepartment of General Surgery, Beijing Friendship Hospital, Capital Medical University & State Key Lab of Digestive Health & National Clinical Research Center for Digestive DiseasesDepartment of General Surgery, Beijing Friendship Hospital, Capital Medical University & State Key Lab of Digestive Health & National Clinical Research Center for Digestive DiseasesDepartment of General Surgery, Beijing Friendship Hospital, Capital Medical University & State Key Lab of Digestive Health & National Clinical Research Center for Digestive DiseasesDepartment of General Surgery, Beijing Friendship Hospital, Capital Medical University & State Key Lab of Digestive Health & National Clinical Research Center for Digestive DiseasesDepartment of General Surgery, Beijing Friendship Hospital, Capital Medical University & State Key Lab of Digestive Health & National Clinical Research Center for Digestive DiseasesDepartment of General Surgery, Beijing Friendship Hospital, Capital Medical University & State Key Lab of Digestive Health & National Clinical Research Center for Digestive DiseasesDepartment of General Surgery, Beijing Friendship Hospital, Capital Medical University & State Key Lab of Digestive Health & National Clinical Research Center for Digestive DiseasesAbstract Lysine crotonylation (Kcr), a previously unknown post-translational modification (PTM), plays crucial roles in regulating cellular processes, including gene expression, chromatin remodeling, and cellular metabolism. Kcr is associated with various diseases, including neurodegenerative disorders, cancer, cardiovascular conditions, and metabolic syndromes. Despite advances in identifying crotonylation sites and their regulatory enzymes, the molecular mechanisms by which Kcr influences disease progression remain poorly understood. Understanding the interplay between Kcr and other acylation modifications may reveal opportunities for developing targeted therapies. This review synthesizes current research on Kcr, focusing on its regulatory mechanisms and disease associations, and highlights insights into future exploration in epigenetics and therapeutic interventions.https://doi.org/10.1186/s13072-025-00577-7
spellingShingle Yu Ji
Shanshan Liu
Yiqiao Zhang
Yiyang Min
Luyang Wei
Chengjian Guan
Huajing Yu
Zhongtao Zhang
Lysine crotonylation in disease: mechanisms, biological functions and therapeutic targets
Epigenetics & Chromatin
title Lysine crotonylation in disease: mechanisms, biological functions and therapeutic targets
title_full Lysine crotonylation in disease: mechanisms, biological functions and therapeutic targets
title_fullStr Lysine crotonylation in disease: mechanisms, biological functions and therapeutic targets
title_full_unstemmed Lysine crotonylation in disease: mechanisms, biological functions and therapeutic targets
title_short Lysine crotonylation in disease: mechanisms, biological functions and therapeutic targets
title_sort lysine crotonylation in disease mechanisms biological functions and therapeutic targets
url https://doi.org/10.1186/s13072-025-00577-7
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