AERIFY-1/2: two phase 3, randomised, controlled trials of itepekimab in former smokers with moderate-to-severe COPD

Background Accumulating data implicate interleukin (IL)-33, a proinflammatory cytokine released locally upon epithelial cell damage, in the pathogenesis of COPD. In a phase 2 study, itepekimab, a human monoclonal antibody against IL-33, reduced exacerbations and improved lung function in a subgroup...

Full description

Saved in:
Bibliographic Details
Main Authors: Klaus F. Rabe, Fernando J. Martinez, Surya P. Bhatt, Tomotaka Kawayama, Borja G. Cosio, Robert M. Mroz, Maarten M. Boomsma, Helene Goulaouic, Michael C. Nivens, Michel Djandji, Xavier Soler, Ying Liu, Matthew P. Kosloski, Christine R. Xu, Nikhil Amin, Heribert Staudinger, David J. Lederer, Raolat M. Abdulai
Format: Article
Language:English
Published: European Respiratory Society 2024-09-01
Series:ERJ Open Research
Online Access:http://openres.ersjournals.com/content/10/5/00718-2023.full
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850193671806255104
author Klaus F. Rabe
Fernando J. Martinez
Surya P. Bhatt
Tomotaka Kawayama
Borja G. Cosio
Robert M. Mroz
Maarten M. Boomsma
Helene Goulaouic
Michael C. Nivens
Michel Djandji
Xavier Soler
Ying Liu
Matthew P. Kosloski
Christine R. Xu
Nikhil Amin
Heribert Staudinger
David J. Lederer
Raolat M. Abdulai
author_facet Klaus F. Rabe
Fernando J. Martinez
Surya P. Bhatt
Tomotaka Kawayama
Borja G. Cosio
Robert M. Mroz
Maarten M. Boomsma
Helene Goulaouic
Michael C. Nivens
Michel Djandji
Xavier Soler
Ying Liu
Matthew P. Kosloski
Christine R. Xu
Nikhil Amin
Heribert Staudinger
David J. Lederer
Raolat M. Abdulai
author_sort Klaus F. Rabe
collection DOAJ
description Background Accumulating data implicate interleukin (IL)-33, a proinflammatory cytokine released locally upon epithelial cell damage, in the pathogenesis of COPD. In a phase 2 study, itepekimab, a human monoclonal antibody against IL-33, reduced exacerbations and improved lung function in a subgroup analysis of former smokers with COPD with an acceptable safety profile. Methods The study designs of AERIFY-1 and AERIFY-2 are described in this article. Discussion The primary objective of AERIFY-1/2 (NCT04701983/NCT04751487), two phase 3 randomised, double-blind, placebo-controlled trials, is to assess the efficacy and safety of itepekimab versus placebo in a population of former smokers with moderate-to-severe COPD over up to 52 weeks. An additional secondary population of current smokers are being enrolled in AERIFY-2. These two studies will enrol patients (aged 40–85 years) with COPD and chronic bronchitis who had ≥2 moderate or ≥ 1 severe exacerbations within the previous year despite standard-of-care triple or double background therapy. All participants are required to have ≥10-pack-year smoking history, and ≥6 months since smoking cessation for former smokers. The primary end-point is the annualised rate of moderate or severe acute exacerbation of COPD. Secondary end-points include change from baseline in pre- and post-bronchodilator forced expiratory volume in 1 s, and annualised frequency of severe exacerbations. Symptomatic end-points include Evaluating Respiratory Symptoms in COPD and St. George's Respiratory Questionnaire, safety and anti-drug antibody responses.
format Article
id doaj-art-3bd4edef6ab44bf1a5e1e7bec238bd0c
institution OA Journals
issn 2312-0541
language English
publishDate 2024-09-01
publisher European Respiratory Society
record_format Article
series ERJ Open Research
spelling doaj-art-3bd4edef6ab44bf1a5e1e7bec238bd0c2025-08-20T02:14:11ZengEuropean Respiratory SocietyERJ Open Research2312-05412024-09-0110510.1183/23120541.00718-202300718-2023AERIFY-1/2: two phase 3, randomised, controlled trials of itepekimab in former smokers with moderate-to-severe COPDKlaus F. Rabe0Fernando J. Martinez1Surya P. Bhatt2Tomotaka Kawayama3Borja G. Cosio4Robert M. Mroz5Maarten M. Boomsma6Helene Goulaouic7Michael C. Nivens8Michel Djandji9Xavier Soler10Ying Liu11Matthew P. Kosloski12Christine R. Xu13Nikhil Amin14Heribert Staudinger15David J. Lederer16Raolat M. Abdulai17 LungenClinic Grosshansdorf, Airway Research Center North, Grosshansdorf, Germany Weill Cornell Medical College, New York, NY, USA University of Alabama at Birmingham, Birmingham, AL, USA Kurume University School of Medicine, Fukuoka, Japan Hospital Universitario Son Espases-IdISBa-CIBERES, Palma de Mallorca, Spain Medical University of Bialystok, Bialystok, Poland Sanofi, Amsterdam, Netherlands Sanofi, Chilly-Mazarin, France Regeneron Pharmaceuticals, Inc., Tarrytown, NY, USA Sanofi, Cambridge, MA, USA Regeneron Pharmaceuticals, Inc., Tarrytown, NY, USA Sanofi, Bridgewater, NJ, USA Regeneron Pharmaceuticals, Inc., Tarrytown, NY, USA Sanofi, Bridgewater, NJ, USA Regeneron Pharmaceuticals, Inc., Tarrytown, NY, USA Sanofi, Bridgewater, NJ, USA Regeneron Pharmaceuticals, Inc., Tarrytown, NY, USA Former Sanofi employee Background Accumulating data implicate interleukin (IL)-33, a proinflammatory cytokine released locally upon epithelial cell damage, in the pathogenesis of COPD. In a phase 2 study, itepekimab, a human monoclonal antibody against IL-33, reduced exacerbations and improved lung function in a subgroup analysis of former smokers with COPD with an acceptable safety profile. Methods The study designs of AERIFY-1 and AERIFY-2 are described in this article. Discussion The primary objective of AERIFY-1/2 (NCT04701983/NCT04751487), two phase 3 randomised, double-blind, placebo-controlled trials, is to assess the efficacy and safety of itepekimab versus placebo in a population of former smokers with moderate-to-severe COPD over up to 52 weeks. An additional secondary population of current smokers are being enrolled in AERIFY-2. These two studies will enrol patients (aged 40–85 years) with COPD and chronic bronchitis who had ≥2 moderate or ≥ 1 severe exacerbations within the previous year despite standard-of-care triple or double background therapy. All participants are required to have ≥10-pack-year smoking history, and ≥6 months since smoking cessation for former smokers. The primary end-point is the annualised rate of moderate or severe acute exacerbation of COPD. Secondary end-points include change from baseline in pre- and post-bronchodilator forced expiratory volume in 1 s, and annualised frequency of severe exacerbations. Symptomatic end-points include Evaluating Respiratory Symptoms in COPD and St. George's Respiratory Questionnaire, safety and anti-drug antibody responses.http://openres.ersjournals.com/content/10/5/00718-2023.full
spellingShingle Klaus F. Rabe
Fernando J. Martinez
Surya P. Bhatt
Tomotaka Kawayama
Borja G. Cosio
Robert M. Mroz
Maarten M. Boomsma
Helene Goulaouic
Michael C. Nivens
Michel Djandji
Xavier Soler
Ying Liu
Matthew P. Kosloski
Christine R. Xu
Nikhil Amin
Heribert Staudinger
David J. Lederer
Raolat M. Abdulai
AERIFY-1/2: two phase 3, randomised, controlled trials of itepekimab in former smokers with moderate-to-severe COPD
ERJ Open Research
title AERIFY-1/2: two phase 3, randomised, controlled trials of itepekimab in former smokers with moderate-to-severe COPD
title_full AERIFY-1/2: two phase 3, randomised, controlled trials of itepekimab in former smokers with moderate-to-severe COPD
title_fullStr AERIFY-1/2: two phase 3, randomised, controlled trials of itepekimab in former smokers with moderate-to-severe COPD
title_full_unstemmed AERIFY-1/2: two phase 3, randomised, controlled trials of itepekimab in former smokers with moderate-to-severe COPD
title_short AERIFY-1/2: two phase 3, randomised, controlled trials of itepekimab in former smokers with moderate-to-severe COPD
title_sort aerify 1 2 two phase 3 randomised controlled trials of itepekimab in former smokers with moderate to severe copd
url http://openres.ersjournals.com/content/10/5/00718-2023.full
work_keys_str_mv AT klausfrabe aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT fernandojmartinez aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT suryapbhatt aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT tomotakakawayama aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT borjagcosio aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT robertmmroz aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT maartenmboomsma aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT helenegoulaouic aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT michaelcnivens aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT micheldjandji aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT xaviersoler aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT yingliu aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT matthewpkosloski aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT christinerxu aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT nikhilamin aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT heribertstaudinger aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT davidjlederer aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd
AT raolatmabdulai aerify12twophase3randomisedcontrolledtrialsofitepekimabinformersmokerswithmoderatetoseverecopd