Increased infection risk in patients on preventive CGRP-targeting therapies– a meta-analysis and clinical effect assessment

Abstract Background Calcitonin gene related peptide (CGRP) pathway targeting therapies have proven efficacy, safety and tolerability. However, CGRP is also involved in immune responses, and reports of an increased risk of infection have emerged. This meta-analysis aims to verify whether CGRP-targeti...

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Main Authors: Marcin Straburzyński, Daria Kopyt, Karol Marschollek, Bartłomiej Błaszczyk, Ewa Kuca-Warnawin, Weronika Kurowska, Błażej Misiak, Kuan-Po Peng, Marta Waliszewska-Prosół, Arne May
Format: Article
Language:English
Published: BMC 2025-04-01
Series:The Journal of Headache and Pain
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Online Access:https://doi.org/10.1186/s10194-025-02040-0
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author Marcin Straburzyński
Daria Kopyt
Karol Marschollek
Bartłomiej Błaszczyk
Ewa Kuca-Warnawin
Weronika Kurowska
Błażej Misiak
Kuan-Po Peng
Marta Waliszewska-Prosół
Arne May
author_facet Marcin Straburzyński
Daria Kopyt
Karol Marschollek
Bartłomiej Błaszczyk
Ewa Kuca-Warnawin
Weronika Kurowska
Błażej Misiak
Kuan-Po Peng
Marta Waliszewska-Prosół
Arne May
author_sort Marcin Straburzyński
collection DOAJ
description Abstract Background Calcitonin gene related peptide (CGRP) pathway targeting therapies have proven efficacy, safety and tolerability. However, CGRP is also involved in immune responses, and reports of an increased risk of infection have emerged. This meta-analysis aims to verify whether CGRP-targeting therapies show evidence of increasing infection risk. Methods A systematic review was conducted according to PRISMA-Harms guidelines. A PubMed and Embase search result selection and extraction was performed. Risk of bias, sensitivity analysis, and fixed/random effects network meta-analyses were conducted for incidence of infectious adverse events in the studied populations with subsequent effect size assessment. An additional infectious serious adverse event search was performed in double-blind and open-label studies. Results The search and selection process yielded 37 randomized placebo-controlled trials. 22,518 patients (77.3% women) treated with erenumab, fremanezumab, galcanezumab, eptinezumab, atogepant and rimegepant participated in these studies. Preventive CGRP-targeting therapies appear to increase the infection relative risk (RR = 1.08 [1.01; 1.14], p = 0.016, Number Needed to Harm [NNH] = 287). However, in individual analyses only galcanezumab and eptinezumab showed an increase in risk of infections: galcanezumab at clinically used doses (RR 1.13 [1.02; 1.25], p = 0.024, NNH = 77); eptinezumab at higher doses (RR 1.23 [1.04; 1.45], p = 0.015, NNH = 24). Fremanezumab was associated with fewest infectious SAEs (n = 3 in 3 studies), while erenumab showed the highest incidence of these events (n = 36 in 11 studies). Conclusions CGRP has multiple and often potentially opposing effects on the immune system. In effect, preventive CGRP pathway antagonists (especially eptinezumab and galcanezumab) possibly only mildly increase the risk of infections. However, it is unlikely to affect most migraine patients considering relatively high NNH, low effect size and few infectious SAEs reported so far. The result of CGRP-targeting therapies potentially depends on the type of pathogen and patient’s immune status. Consequently, in immunocompromised patients or at public health levels the increased infection risk may have more pronounced effect.
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series The Journal of Headache and Pain
spelling doaj-art-31701e1116634367833bf08bcc0f2bde2025-08-20T03:53:32ZengBMCThe Journal of Headache and Pain1129-23772025-04-0126111710.1186/s10194-025-02040-0Increased infection risk in patients on preventive CGRP-targeting therapies– a meta-analysis and clinical effect assessmentMarcin Straburzyński0Daria Kopyt1Karol Marschollek2Bartłomiej Błaszczyk3Ewa Kuca-Warnawin4Weronika Kurowska5Błażej Misiak6Kuan-Po Peng7Marta Waliszewska-Prosół8Arne May9Department of Family Medicine and Infectious Diseases, University of Warmia and Mazury in OlsztynScientific Section of the Polish Society of Family MedicineDepartment of Neurology, Wroclaw Medical UniversityDepartment of Neurology, Wroclaw Medical UniversityDepartment of Pathophysiology and Immunology, National Institute of Geriatrics, Rheumatology and RehabilitationDepartment of Pathophysiology and Immunology, National Institute of Geriatrics, Rheumatology and RehabilitationDepartment of Psychiatry, Wroclaw Medical UniversityDepartment of Systems Neuroscience, University Medical Center Hamburg-EppendorfDepartment of Neurology, Wroclaw Medical UniversityDepartment of Systems Neuroscience, University Medical Center Hamburg-EppendorfAbstract Background Calcitonin gene related peptide (CGRP) pathway targeting therapies have proven efficacy, safety and tolerability. However, CGRP is also involved in immune responses, and reports of an increased risk of infection have emerged. This meta-analysis aims to verify whether CGRP-targeting therapies show evidence of increasing infection risk. Methods A systematic review was conducted according to PRISMA-Harms guidelines. A PubMed and Embase search result selection and extraction was performed. Risk of bias, sensitivity analysis, and fixed/random effects network meta-analyses were conducted for incidence of infectious adverse events in the studied populations with subsequent effect size assessment. An additional infectious serious adverse event search was performed in double-blind and open-label studies. Results The search and selection process yielded 37 randomized placebo-controlled trials. 22,518 patients (77.3% women) treated with erenumab, fremanezumab, galcanezumab, eptinezumab, atogepant and rimegepant participated in these studies. Preventive CGRP-targeting therapies appear to increase the infection relative risk (RR = 1.08 [1.01; 1.14], p = 0.016, Number Needed to Harm [NNH] = 287). However, in individual analyses only galcanezumab and eptinezumab showed an increase in risk of infections: galcanezumab at clinically used doses (RR 1.13 [1.02; 1.25], p = 0.024, NNH = 77); eptinezumab at higher doses (RR 1.23 [1.04; 1.45], p = 0.015, NNH = 24). Fremanezumab was associated with fewest infectious SAEs (n = 3 in 3 studies), while erenumab showed the highest incidence of these events (n = 36 in 11 studies). Conclusions CGRP has multiple and often potentially opposing effects on the immune system. In effect, preventive CGRP pathway antagonists (especially eptinezumab and galcanezumab) possibly only mildly increase the risk of infections. However, it is unlikely to affect most migraine patients considering relatively high NNH, low effect size and few infectious SAEs reported so far. The result of CGRP-targeting therapies potentially depends on the type of pathogen and patient’s immune status. Consequently, in immunocompromised patients or at public health levels the increased infection risk may have more pronounced effect.https://doi.org/10.1186/s10194-025-02040-0ErenumabFremanezumabGalcanezumabEptinezumabAtogepantRimegepant
spellingShingle Marcin Straburzyński
Daria Kopyt
Karol Marschollek
Bartłomiej Błaszczyk
Ewa Kuca-Warnawin
Weronika Kurowska
Błażej Misiak
Kuan-Po Peng
Marta Waliszewska-Prosół
Arne May
Increased infection risk in patients on preventive CGRP-targeting therapies– a meta-analysis and clinical effect assessment
The Journal of Headache and Pain
Erenumab
Fremanezumab
Galcanezumab
Eptinezumab
Atogepant
Rimegepant
title Increased infection risk in patients on preventive CGRP-targeting therapies– a meta-analysis and clinical effect assessment
title_full Increased infection risk in patients on preventive CGRP-targeting therapies– a meta-analysis and clinical effect assessment
title_fullStr Increased infection risk in patients on preventive CGRP-targeting therapies– a meta-analysis and clinical effect assessment
title_full_unstemmed Increased infection risk in patients on preventive CGRP-targeting therapies– a meta-analysis and clinical effect assessment
title_short Increased infection risk in patients on preventive CGRP-targeting therapies– a meta-analysis and clinical effect assessment
title_sort increased infection risk in patients on preventive cgrp targeting therapies a meta analysis and clinical effect assessment
topic Erenumab
Fremanezumab
Galcanezumab
Eptinezumab
Atogepant
Rimegepant
url https://doi.org/10.1186/s10194-025-02040-0
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