STK11 mutation impacts CD1E expression to regulate the differentiation of macrophages in lung adenocarcinoma

Abstract Background The deficiency of serine/threonine protein kinase 11 (STK11), one of the most common tumor suppressor genes in non‐small‐cell lung cancer, is a crucial player in tumor immune microenvironment regulation. This study attempted to unveil how mutated STK11 impact the differentiation...

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Main Authors: Qingfeng Zhang, Juan Feng, Kui Liu, Xiaoyan Yang, Yun Huang, Bo Tang
Format: Article
Language:English
Published: Wiley 2023-07-01
Series:Immunity, Inflammation and Disease
Subjects:
Online Access:https://doi.org/10.1002/iid3.958
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author Qingfeng Zhang
Juan Feng
Kui Liu
Xiaoyan Yang
Yun Huang
Bo Tang
author_facet Qingfeng Zhang
Juan Feng
Kui Liu
Xiaoyan Yang
Yun Huang
Bo Tang
author_sort Qingfeng Zhang
collection DOAJ
description Abstract Background The deficiency of serine/threonine protein kinase 11 (STK11), one of the most common tumor suppressor genes in non‐small‐cell lung cancer, is a crucial player in tumor immune microenvironment regulation. This study attempted to unveil how mutated STK11 impact the differentiation of macrophages in lung adenocarcinoma (LUAD). Methods STK11 and CD1E expression levels in different cell models were assessed by quantitative reverse transcription polymerase chain reaction. Western blot was utilized to detect the protein expression levels of STK11, CD1E, apoptosis markers, and AMPK signaling pathway markers after transfection treatment. Cell viability and macrophage differentiation were detected by CCK‐8 and flow cytometry. Immunohistochemistry and immunofluorescence were employed to detect the expression of related genes and macrophage markers, respectively. Results This study found that STK11 mutations promoted the proliferation of LUAD cells and inhibited the differentiation of M1 macrophages, apoptosis, and the AMPK signaling pathway. Mutated STK11 led to CD1E downregulation, which curbed the differentiation of M1 macrophages and hence promoted LUAD progression. It was further validated by the in vivo experimental results that STK11 mutation significantly decreased the immune infiltration of M1 macrophages and promoted LUAD progression. Conclusion It was revealed that STK11 mutation affected CD1E expression to regulate macrophage differentiation in LUAD and then promote tumor progression. In this way, CD1E could be a potential biological target for the therapeutic interventions of STK11‐mutant LUAD patients. These findings also threw new light on a new therapeutic strategy for STK11‐mutant tumor patients that assisted the macrophage polarization pathway.
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spelling doaj-art-309d74cf889c4863a63b6960e2b091502025-08-20T03:56:09ZengWileyImmunity, Inflammation and Disease2050-45272023-07-01117n/an/a10.1002/iid3.958STK11 mutation impacts CD1E expression to regulate the differentiation of macrophages in lung adenocarcinomaQingfeng Zhang0Juan Feng1Kui Liu2Xiaoyan Yang3Yun Huang4Bo Tang5Department of Cardio‐Thoracic Surgery Zigong Fourth People's Hospital Zigong ChinaDepartment of Operating Room Zigong Fourth People's Hospital Zigong ChinaDepartment of Cardio‐Thoracic Surgery Zigong Fourth People's Hospital Zigong ChinaDepartment of Cardio‐Thoracic Surgery Zigong Fourth People's Hospital Zigong ChinaDepartment of Cardio‐Thoracic Surgery Zigong Fourth People's Hospital Zigong ChinaDepartment of Cardio‐Thoracic Surgery Zigong Fourth People's Hospital Zigong ChinaAbstract Background The deficiency of serine/threonine protein kinase 11 (STK11), one of the most common tumor suppressor genes in non‐small‐cell lung cancer, is a crucial player in tumor immune microenvironment regulation. This study attempted to unveil how mutated STK11 impact the differentiation of macrophages in lung adenocarcinoma (LUAD). Methods STK11 and CD1E expression levels in different cell models were assessed by quantitative reverse transcription polymerase chain reaction. Western blot was utilized to detect the protein expression levels of STK11, CD1E, apoptosis markers, and AMPK signaling pathway markers after transfection treatment. Cell viability and macrophage differentiation were detected by CCK‐8 and flow cytometry. Immunohistochemistry and immunofluorescence were employed to detect the expression of related genes and macrophage markers, respectively. Results This study found that STK11 mutations promoted the proliferation of LUAD cells and inhibited the differentiation of M1 macrophages, apoptosis, and the AMPK signaling pathway. Mutated STK11 led to CD1E downregulation, which curbed the differentiation of M1 macrophages and hence promoted LUAD progression. It was further validated by the in vivo experimental results that STK11 mutation significantly decreased the immune infiltration of M1 macrophages and promoted LUAD progression. Conclusion It was revealed that STK11 mutation affected CD1E expression to regulate macrophage differentiation in LUAD and then promote tumor progression. In this way, CD1E could be a potential biological target for the therapeutic interventions of STK11‐mutant LUAD patients. These findings also threw new light on a new therapeutic strategy for STK11‐mutant tumor patients that assisted the macrophage polarization pathway.https://doi.org/10.1002/iid3.958CD1Elung adenocarcinomamacrophagesproliferationSTK11 mutation
spellingShingle Qingfeng Zhang
Juan Feng
Kui Liu
Xiaoyan Yang
Yun Huang
Bo Tang
STK11 mutation impacts CD1E expression to regulate the differentiation of macrophages in lung adenocarcinoma
Immunity, Inflammation and Disease
CD1E
lung adenocarcinoma
macrophages
proliferation
STK11 mutation
title STK11 mutation impacts CD1E expression to regulate the differentiation of macrophages in lung adenocarcinoma
title_full STK11 mutation impacts CD1E expression to regulate the differentiation of macrophages in lung adenocarcinoma
title_fullStr STK11 mutation impacts CD1E expression to regulate the differentiation of macrophages in lung adenocarcinoma
title_full_unstemmed STK11 mutation impacts CD1E expression to regulate the differentiation of macrophages in lung adenocarcinoma
title_short STK11 mutation impacts CD1E expression to regulate the differentiation of macrophages in lung adenocarcinoma
title_sort stk11 mutation impacts cd1e expression to regulate the differentiation of macrophages in lung adenocarcinoma
topic CD1E
lung adenocarcinoma
macrophages
proliferation
STK11 mutation
url https://doi.org/10.1002/iid3.958
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