SDA, a DNA aptamer inhibiting E- and P-selectin mediated adhesion of cancer and leukemia cells, the first and pivotal step in transendothelial migration during metastasis formation.

Endothelial (E-) and platelet (P-) selectin mediated adhesion of tumor cells to vascular endothelium is a pivotal step of hematogenous metastasis formation. Recent studies have demonstrated that selectin deficiency significantly reduces metastasis formation in vivo. We selected an E- and P-Selectin...

Full description

Saved in:
Bibliographic Details
Main Authors: Rassa Faryammanesh, Tobias Lange, Eileen Magbanua, Sina Haas, Cindy Meyer, Daniel Wicklein, Udo Schumacher, Ulrich Hahn
Format: Article
Language:English
Published: Public Library of Science (PLoS) 2014-01-01
Series:PLoS ONE
Online Access:https://journals.plos.org/plosone/article/file?id=10.1371/journal.pone.0093173&type=printable
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850026534570557440
author Rassa Faryammanesh
Tobias Lange
Eileen Magbanua
Sina Haas
Cindy Meyer
Daniel Wicklein
Udo Schumacher
Ulrich Hahn
author_facet Rassa Faryammanesh
Tobias Lange
Eileen Magbanua
Sina Haas
Cindy Meyer
Daniel Wicklein
Udo Schumacher
Ulrich Hahn
author_sort Rassa Faryammanesh
collection DOAJ
description Endothelial (E-) and platelet (P-) selectin mediated adhesion of tumor cells to vascular endothelium is a pivotal step of hematogenous metastasis formation. Recent studies have demonstrated that selectin deficiency significantly reduces metastasis formation in vivo. We selected an E- and P-Selectin specific DNA Aptamer (SDA) via SELEX (Systematic Evolution of Ligands by EXponential enrichment) with a K(d) value of approximately 100 nM and the capability of inhibiting the interaction between selectin and its ligands. Employing human colorectal cancer (HT29) and leukemia (EOL-1) cell lines we could demonstrate an anti-adhesive effect for SDA in vitro. Under physiological shear stress conditions in a laminar flow adhesion assay, SDA inhibited dynamic tumor cell adhesion to immobilized E- or P-selectin. The stability of SDA for more than two hours allowed its application in cell-cell adhesion assays in cell culture medium. When adhesion of HT29 cells to TNFα-stimulated E-selectin presenting human pulmonary microvascular endothelial cells was analyzed, inhibition via SDA could be demonstrated as well. In conclusion, SDA is a potential new therapeutic agent that antagonizes selectin-mediated adhesion during metastasis formation in human malignancies.
format Article
id doaj-art-300bac2634c745188924c6d0df3fcf6d
institution DOAJ
issn 1932-6203
language English
publishDate 2014-01-01
publisher Public Library of Science (PLoS)
record_format Article
series PLoS ONE
spelling doaj-art-300bac2634c745188924c6d0df3fcf6d2025-08-20T03:00:31ZengPublic Library of Science (PLoS)PLoS ONE1932-62032014-01-0194e9317310.1371/journal.pone.0093173SDA, a DNA aptamer inhibiting E- and P-selectin mediated adhesion of cancer and leukemia cells, the first and pivotal step in transendothelial migration during metastasis formation.Rassa FaryammaneshTobias LangeEileen MagbanuaSina HaasCindy MeyerDaniel WickleinUdo SchumacherUlrich HahnEndothelial (E-) and platelet (P-) selectin mediated adhesion of tumor cells to vascular endothelium is a pivotal step of hematogenous metastasis formation. Recent studies have demonstrated that selectin deficiency significantly reduces metastasis formation in vivo. We selected an E- and P-Selectin specific DNA Aptamer (SDA) via SELEX (Systematic Evolution of Ligands by EXponential enrichment) with a K(d) value of approximately 100 nM and the capability of inhibiting the interaction between selectin and its ligands. Employing human colorectal cancer (HT29) and leukemia (EOL-1) cell lines we could demonstrate an anti-adhesive effect for SDA in vitro. Under physiological shear stress conditions in a laminar flow adhesion assay, SDA inhibited dynamic tumor cell adhesion to immobilized E- or P-selectin. The stability of SDA for more than two hours allowed its application in cell-cell adhesion assays in cell culture medium. When adhesion of HT29 cells to TNFα-stimulated E-selectin presenting human pulmonary microvascular endothelial cells was analyzed, inhibition via SDA could be demonstrated as well. In conclusion, SDA is a potential new therapeutic agent that antagonizes selectin-mediated adhesion during metastasis formation in human malignancies.https://journals.plos.org/plosone/article/file?id=10.1371/journal.pone.0093173&type=printable
spellingShingle Rassa Faryammanesh
Tobias Lange
Eileen Magbanua
Sina Haas
Cindy Meyer
Daniel Wicklein
Udo Schumacher
Ulrich Hahn
SDA, a DNA aptamer inhibiting E- and P-selectin mediated adhesion of cancer and leukemia cells, the first and pivotal step in transendothelial migration during metastasis formation.
PLoS ONE
title SDA, a DNA aptamer inhibiting E- and P-selectin mediated adhesion of cancer and leukemia cells, the first and pivotal step in transendothelial migration during metastasis formation.
title_full SDA, a DNA aptamer inhibiting E- and P-selectin mediated adhesion of cancer and leukemia cells, the first and pivotal step in transendothelial migration during metastasis formation.
title_fullStr SDA, a DNA aptamer inhibiting E- and P-selectin mediated adhesion of cancer and leukemia cells, the first and pivotal step in transendothelial migration during metastasis formation.
title_full_unstemmed SDA, a DNA aptamer inhibiting E- and P-selectin mediated adhesion of cancer and leukemia cells, the first and pivotal step in transendothelial migration during metastasis formation.
title_short SDA, a DNA aptamer inhibiting E- and P-selectin mediated adhesion of cancer and leukemia cells, the first and pivotal step in transendothelial migration during metastasis formation.
title_sort sda a dna aptamer inhibiting e and p selectin mediated adhesion of cancer and leukemia cells the first and pivotal step in transendothelial migration during metastasis formation
url https://journals.plos.org/plosone/article/file?id=10.1371/journal.pone.0093173&type=printable
work_keys_str_mv AT rassafaryammanesh sdaadnaaptamerinhibitingeandpselectinmediatedadhesionofcancerandleukemiacellsthefirstandpivotalstepintransendothelialmigrationduringmetastasisformation
AT tobiaslange sdaadnaaptamerinhibitingeandpselectinmediatedadhesionofcancerandleukemiacellsthefirstandpivotalstepintransendothelialmigrationduringmetastasisformation
AT eileenmagbanua sdaadnaaptamerinhibitingeandpselectinmediatedadhesionofcancerandleukemiacellsthefirstandpivotalstepintransendothelialmigrationduringmetastasisformation
AT sinahaas sdaadnaaptamerinhibitingeandpselectinmediatedadhesionofcancerandleukemiacellsthefirstandpivotalstepintransendothelialmigrationduringmetastasisformation
AT cindymeyer sdaadnaaptamerinhibitingeandpselectinmediatedadhesionofcancerandleukemiacellsthefirstandpivotalstepintransendothelialmigrationduringmetastasisformation
AT danielwicklein sdaadnaaptamerinhibitingeandpselectinmediatedadhesionofcancerandleukemiacellsthefirstandpivotalstepintransendothelialmigrationduringmetastasisformation
AT udoschumacher sdaadnaaptamerinhibitingeandpselectinmediatedadhesionofcancerandleukemiacellsthefirstandpivotalstepintransendothelialmigrationduringmetastasisformation
AT ulrichhahn sdaadnaaptamerinhibitingeandpselectinmediatedadhesionofcancerandleukemiacellsthefirstandpivotalstepintransendothelialmigrationduringmetastasisformation