miR‐373 regulates inflammatory cytokine‐mediated chondrocyte proliferation in osteoarthritis by targeting the P2X7 receptor

Inflammatory cytokines commonly initiate extreme changes in the synovium and cartilage microenvironment of osteoarthritis (OA) patients, which subsequently cause cellular dysfunction, especially in chondrocytes. It has been reported that induction of the purinergic P2X7 receptor (P2X7R) can regulate...

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Main Authors: Wei Zhang, Biao Zhong, Chi Zhang, Congfeng Luo, Yulin Zhan
Format: Article
Language:English
Published: Wiley 2018-03-01
Series:FEBS Open Bio
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Online Access:https://doi.org/10.1002/2211-5463.12345
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author Wei Zhang
Biao Zhong
Chi Zhang
Congfeng Luo
Yulin Zhan
author_facet Wei Zhang
Biao Zhong
Chi Zhang
Congfeng Luo
Yulin Zhan
author_sort Wei Zhang
collection DOAJ
description Inflammatory cytokines commonly initiate extreme changes in the synovium and cartilage microenvironment of osteoarthritis (OA) patients, which subsequently cause cellular dysfunction, especially in chondrocytes. It has been reported that induction of the purinergic P2X7 receptor (P2X7R) can regulate the expression of a variety of inflammatory factors, including interleukin (IL)‐6 and ‐8, leading to OA pathogenesis. However, knowledge of the mechanism of upregulation of P2X7R in OA is still incomplete, and its role in chondrocyte proliferation is also not clear. It was reported previously that the expression of P2X7R was controlled by certain microRNAs, and so we tested the expression of several microRNAs and found that microRNA‐373 (miR‐373) was downregulated in the chondrocytes from OA patients. Regarding the mechanism of action, miR‐373 inhibited chondrocyte proliferation by suppressing the expression of P2X7R, as well as inflammatory factors such as IL‐6 and IL‐8. Furthermore, the proliferative and pro‐inflammatory effects of miR‐373 on the chondrocytes could be suppressed by a P2X7R antagonist, further suggesting that miR‐373 mediates chondrocyte proliferation and inflammation by targeting P2X7R. Generally, our results suggest a novel method for OA treatment by targeting the miR‐373–P2X7R pathway.
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spelling doaj-art-2e071e33763e46f688879514ffbffd8c2025-08-20T01:57:24ZengWileyFEBS Open Bio2211-54632018-03-018332533110.1002/2211-5463.12345miR‐373 regulates inflammatory cytokine‐mediated chondrocyte proliferation in osteoarthritis by targeting the P2X7 receptorWei Zhang0Biao Zhong1Chi Zhang2Congfeng Luo3Yulin Zhan4Department of Orthopaedics Shanghai Jiao Tong University Affiliated Sixth People's Hospital Shanghai ChinaDepartment of Orthopaedics Shanghai Jiao Tong University Affiliated Sixth People's Hospital Shanghai ChinaDepartment of Orthopaedics Shanghai Jiao Tong University Affiliated Sixth People's Hospital Shanghai ChinaDepartment of Orthopaedics Shanghai Jiao Tong University Affiliated Sixth People's Hospital Shanghai ChinaDepartment of Orthopaedics Shanghai Jiao Tong University Affiliated Sixth People's Hospital Shanghai ChinaInflammatory cytokines commonly initiate extreme changes in the synovium and cartilage microenvironment of osteoarthritis (OA) patients, which subsequently cause cellular dysfunction, especially in chondrocytes. It has been reported that induction of the purinergic P2X7 receptor (P2X7R) can regulate the expression of a variety of inflammatory factors, including interleukin (IL)‐6 and ‐8, leading to OA pathogenesis. However, knowledge of the mechanism of upregulation of P2X7R in OA is still incomplete, and its role in chondrocyte proliferation is also not clear. It was reported previously that the expression of P2X7R was controlled by certain microRNAs, and so we tested the expression of several microRNAs and found that microRNA‐373 (miR‐373) was downregulated in the chondrocytes from OA patients. Regarding the mechanism of action, miR‐373 inhibited chondrocyte proliferation by suppressing the expression of P2X7R, as well as inflammatory factors such as IL‐6 and IL‐8. Furthermore, the proliferative and pro‐inflammatory effects of miR‐373 on the chondrocytes could be suppressed by a P2X7R antagonist, further suggesting that miR‐373 mediates chondrocyte proliferation and inflammation by targeting P2X7R. Generally, our results suggest a novel method for OA treatment by targeting the miR‐373–P2X7R pathway.https://doi.org/10.1002/2211-5463.12345chondrocytemiR‐373osteoarthritispurinergic P2X7 receptor
spellingShingle Wei Zhang
Biao Zhong
Chi Zhang
Congfeng Luo
Yulin Zhan
miR‐373 regulates inflammatory cytokine‐mediated chondrocyte proliferation in osteoarthritis by targeting the P2X7 receptor
FEBS Open Bio
chondrocyte
miR‐373
osteoarthritis
purinergic P2X7 receptor
title miR‐373 regulates inflammatory cytokine‐mediated chondrocyte proliferation in osteoarthritis by targeting the P2X7 receptor
title_full miR‐373 regulates inflammatory cytokine‐mediated chondrocyte proliferation in osteoarthritis by targeting the P2X7 receptor
title_fullStr miR‐373 regulates inflammatory cytokine‐mediated chondrocyte proliferation in osteoarthritis by targeting the P2X7 receptor
title_full_unstemmed miR‐373 regulates inflammatory cytokine‐mediated chondrocyte proliferation in osteoarthritis by targeting the P2X7 receptor
title_short miR‐373 regulates inflammatory cytokine‐mediated chondrocyte proliferation in osteoarthritis by targeting the P2X7 receptor
title_sort mir 373 regulates inflammatory cytokine mediated chondrocyte proliferation in osteoarthritis by targeting the p2x7 receptor
topic chondrocyte
miR‐373
osteoarthritis
purinergic P2X7 receptor
url https://doi.org/10.1002/2211-5463.12345
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AT biaozhong mir373regulatesinflammatorycytokinemediatedchondrocyteproliferationinosteoarthritisbytargetingthep2x7receptor
AT chizhang mir373regulatesinflammatorycytokinemediatedchondrocyteproliferationinosteoarthritisbytargetingthep2x7receptor
AT congfengluo mir373regulatesinflammatorycytokinemediatedchondrocyteproliferationinosteoarthritisbytargetingthep2x7receptor
AT yulinzhan mir373regulatesinflammatorycytokinemediatedchondrocyteproliferationinosteoarthritisbytargetingthep2x7receptor