N-Acetyl Cysteine Protects against Methamphetamine-Induced Dopaminergic Neurodegeneration via Modulation of Redox Status and Autophagy in Dopaminergic Cells

Methamphetamine- (MA-) induced neurotoxicity is associated with mitochondrial dysfunction and enhanced oxidative stress. Our previous study demonstrated that MA induces autophagy in a dopaminergic neuronal cell model (N27 cells). The cellular mechanisms underlying MA-induced autophagy and apoptosis...

Full description

Saved in:
Bibliographic Details
Main Authors: Prashanth Chandramani Shivalingappa, Huajun Jin, Vellareddy Anantharam, Anumantha Kanthasamy, Arthi Kanthasamy
Format: Article
Language:English
Published: Wiley 2012-01-01
Series:Parkinson's Disease
Online Access:http://dx.doi.org/10.1155/2012/424285
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849306716204695552
author Prashanth Chandramani Shivalingappa
Huajun Jin
Vellareddy Anantharam
Anumantha Kanthasamy
Arthi Kanthasamy
author_facet Prashanth Chandramani Shivalingappa
Huajun Jin
Vellareddy Anantharam
Anumantha Kanthasamy
Arthi Kanthasamy
author_sort Prashanth Chandramani Shivalingappa
collection DOAJ
description Methamphetamine- (MA-) induced neurotoxicity is associated with mitochondrial dysfunction and enhanced oxidative stress. Our previous study demonstrated that MA induces autophagy in a dopaminergic neuronal cell model (N27 cells). The cellular mechanisms underlying MA-induced autophagy and apoptosis remain poorly characterized. In the present study we sought to investigate the importance of GSH redox status in MA-induced neurotoxicity using a thiol antioxidant, N-acetylcysteine (NAC). Morphological and biochemical analysis revealed that MA-induced autophagy in N27 dopaminergic cells was associated with pronounced depletion of GSH levels. Moreover, pretreatment with NAC reduced MA-induced GSH depletion and autophagy, while depletion of GSH using L-buthionine sulfoximine (L-BSO) enhanced autophagy. Furthermore, treatment with NAC significantly attenuated MA-induced apoptotic cell death as well as oxidative stress markers, namely, 3-nitrotyrosine (3-NT) and 4-hydroxynonenal (4-HNE). Together, these results suggest that NAC exhibits significant protective effects against MA-induced dopaminergic cell death, presumably via modulation of the GSH level and autophagy. Collectively, our data provide mechanistic insights into the role of cellular GSH redox status in MA-induced autophagy and apoptotic cell death, and additional studies are needed to determine the therapeutic effectiveness of cellular redox modifiers in attenuating dopaminergic neurodegeneration in vivo.
format Article
id doaj-art-2caf6b5ff76d45d78c07c7bc90274c82
institution Kabale University
issn 2090-8083
2042-0080
language English
publishDate 2012-01-01
publisher Wiley
record_format Article
series Parkinson's Disease
spelling doaj-art-2caf6b5ff76d45d78c07c7bc90274c822025-08-20T03:55:00ZengWileyParkinson's Disease2090-80832042-00802012-01-01201210.1155/2012/424285424285N-Acetyl Cysteine Protects against Methamphetamine-Induced Dopaminergic Neurodegeneration via Modulation of Redox Status and Autophagy in Dopaminergic CellsPrashanth Chandramani Shivalingappa0Huajun Jin1Vellareddy Anantharam2Anumantha Kanthasamy3Arthi Kanthasamy4Parkinson's Disorder Research Laboratory, Iowa Center for Advanced Neurotoxicology, Department of Biomedical Sciences, College of Veterinary Medicine, Iowa State University, Ames, IA 50011, USAParkinson's Disorder Research Laboratory, Iowa Center for Advanced Neurotoxicology, Department of Biomedical Sciences, College of Veterinary Medicine, Iowa State University, Ames, IA 50011, USAParkinson's Disorder Research Laboratory, Iowa Center for Advanced Neurotoxicology, Department of Biomedical Sciences, College of Veterinary Medicine, Iowa State University, Ames, IA 50011, USAParkinson's Disorder Research Laboratory, Iowa Center for Advanced Neurotoxicology, Department of Biomedical Sciences, College of Veterinary Medicine, Iowa State University, Ames, IA 50011, USAParkinson's Disorder Research Laboratory, Iowa Center for Advanced Neurotoxicology, Department of Biomedical Sciences, College of Veterinary Medicine, Iowa State University, Ames, IA 50011, USAMethamphetamine- (MA-) induced neurotoxicity is associated with mitochondrial dysfunction and enhanced oxidative stress. Our previous study demonstrated that MA induces autophagy in a dopaminergic neuronal cell model (N27 cells). The cellular mechanisms underlying MA-induced autophagy and apoptosis remain poorly characterized. In the present study we sought to investigate the importance of GSH redox status in MA-induced neurotoxicity using a thiol antioxidant, N-acetylcysteine (NAC). Morphological and biochemical analysis revealed that MA-induced autophagy in N27 dopaminergic cells was associated with pronounced depletion of GSH levels. Moreover, pretreatment with NAC reduced MA-induced GSH depletion and autophagy, while depletion of GSH using L-buthionine sulfoximine (L-BSO) enhanced autophagy. Furthermore, treatment with NAC significantly attenuated MA-induced apoptotic cell death as well as oxidative stress markers, namely, 3-nitrotyrosine (3-NT) and 4-hydroxynonenal (4-HNE). Together, these results suggest that NAC exhibits significant protective effects against MA-induced dopaminergic cell death, presumably via modulation of the GSH level and autophagy. Collectively, our data provide mechanistic insights into the role of cellular GSH redox status in MA-induced autophagy and apoptotic cell death, and additional studies are needed to determine the therapeutic effectiveness of cellular redox modifiers in attenuating dopaminergic neurodegeneration in vivo.http://dx.doi.org/10.1155/2012/424285
spellingShingle Prashanth Chandramani Shivalingappa
Huajun Jin
Vellareddy Anantharam
Anumantha Kanthasamy
Arthi Kanthasamy
N-Acetyl Cysteine Protects against Methamphetamine-Induced Dopaminergic Neurodegeneration via Modulation of Redox Status and Autophagy in Dopaminergic Cells
Parkinson's Disease
title N-Acetyl Cysteine Protects against Methamphetamine-Induced Dopaminergic Neurodegeneration via Modulation of Redox Status and Autophagy in Dopaminergic Cells
title_full N-Acetyl Cysteine Protects against Methamphetamine-Induced Dopaminergic Neurodegeneration via Modulation of Redox Status and Autophagy in Dopaminergic Cells
title_fullStr N-Acetyl Cysteine Protects against Methamphetamine-Induced Dopaminergic Neurodegeneration via Modulation of Redox Status and Autophagy in Dopaminergic Cells
title_full_unstemmed N-Acetyl Cysteine Protects against Methamphetamine-Induced Dopaminergic Neurodegeneration via Modulation of Redox Status and Autophagy in Dopaminergic Cells
title_short N-Acetyl Cysteine Protects against Methamphetamine-Induced Dopaminergic Neurodegeneration via Modulation of Redox Status and Autophagy in Dopaminergic Cells
title_sort n acetyl cysteine protects against methamphetamine induced dopaminergic neurodegeneration via modulation of redox status and autophagy in dopaminergic cells
url http://dx.doi.org/10.1155/2012/424285
work_keys_str_mv AT prashanthchandramanishivalingappa nacetylcysteineprotectsagainstmethamphetamineinduceddopaminergicneurodegenerationviamodulationofredoxstatusandautophagyindopaminergiccells
AT huajunjin nacetylcysteineprotectsagainstmethamphetamineinduceddopaminergicneurodegenerationviamodulationofredoxstatusandautophagyindopaminergiccells
AT vellareddyanantharam nacetylcysteineprotectsagainstmethamphetamineinduceddopaminergicneurodegenerationviamodulationofredoxstatusandautophagyindopaminergiccells
AT anumanthakanthasamy nacetylcysteineprotectsagainstmethamphetamineinduceddopaminergicneurodegenerationviamodulationofredoxstatusandautophagyindopaminergiccells
AT arthikanthasamy nacetylcysteineprotectsagainstmethamphetamineinduceddopaminergicneurodegenerationviamodulationofredoxstatusandautophagyindopaminergiccells