Microwave‐Assisted Tragacanth Gum–Based Grafted Silver Nanocomposite Hydrogel for Sustained Release Formulations of Diclofenac Sodium and Antibacterial Assay

ABSTRACT In this work, novel tragacanth gum‐graft‐poly(2‐acrylamido‐2‐methylpropanesulfonic acid) (TG‐g‐PAMPS) hydrogel was synthesized via free radical copolymerization of TG, 2‐acrylamido‐2‐methylpropanesulfonic acid by using ammonium peroxodisulfate and N,N‐methylene‐bis‐acrylamide under microwav...

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Main Authors: Sharanappa Chapi, Gangadhar Babaladimath, M. V. Murugendrappa, Anjanapura V. Raghu
Format: Article
Language:English
Published: Wiley-VCH 2024-12-01
Series:Nano Select
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Online Access:https://doi.org/10.1002/nano.202300200
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author Sharanappa Chapi
Gangadhar Babaladimath
M. V. Murugendrappa
Anjanapura V. Raghu
author_facet Sharanappa Chapi
Gangadhar Babaladimath
M. V. Murugendrappa
Anjanapura V. Raghu
author_sort Sharanappa Chapi
collection DOAJ
description ABSTRACT In this work, novel tragacanth gum‐graft‐poly(2‐acrylamido‐2‐methylpropanesulfonic acid) (TG‐g‐PAMPS) hydrogel was synthesized via free radical copolymerization of TG, 2‐acrylamido‐2‐methylpropanesulfonic acid by using ammonium peroxodisulfate and N,N‐methylene‐bis‐acrylamide under microwave radiation, resulting in the cross‐linked graft copolymer network. Silver nanoparticles (SNs) were formed and stabilized by the reduction of silver nitrate using tri‐sodium citrate. The TG‐g‐PAMPS gel and its nanocomposite were characterized and confirmed using FTIR, TGA, XRD, SEM, EDS, and TEM techniques. It is observed that the presence of SNs significantly improves the swelling ability of the TG‐g‐PAMPS gel. Degradation studies of both hydrogels were studied using the soil burial method and determining the respective weight loss. The presence of SNs is found to impart significant antibacterial properties to the gel against Pseudomonas aeruginosa and Escherichia coli bacteria. Further, the TG‐g‐PAMPS gel and TG‐g‐PAMPS‐SN were evaluated as matrix materials for the release of the drug (diclofenac sodium) and the effect of SNs on the release was examined. The in‐vitro released data were analyzed using empirical equations to understand the mechanism of release. Among the various models, the released data were well fitted into the Korsmeyer–Peppas equation and the released kinetics followed non‐Fickian diffusion.
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spelling doaj-art-29f2cc3d7a2a4e78b7516a92f9327fe92025-08-20T02:21:52ZengWiley-VCHNano Select2688-40112024-12-01512n/an/a10.1002/nano.202300200Microwave‐Assisted Tragacanth Gum–Based Grafted Silver Nanocomposite Hydrogel for Sustained Release Formulations of Diclofenac Sodium and Antibacterial AssaySharanappa Chapi0Gangadhar Babaladimath1M. V. Murugendrappa2Anjanapura V. Raghu3Department of Physics B.M.S. College of Engineering Bengaluru Karnataka IndiaPost‐Graduation Department of Chemistry KLE Society's Raja Lakhamagouda Science Institute Belagavi Karnataka IndiaDepartment of Physics B.M.S. College of Engineering Bengaluru Karnataka IndiaDepartment of Basic Sciences Faculty of Engineering and Technology CMR University Bangalore IndiaABSTRACT In this work, novel tragacanth gum‐graft‐poly(2‐acrylamido‐2‐methylpropanesulfonic acid) (TG‐g‐PAMPS) hydrogel was synthesized via free radical copolymerization of TG, 2‐acrylamido‐2‐methylpropanesulfonic acid by using ammonium peroxodisulfate and N,N‐methylene‐bis‐acrylamide under microwave radiation, resulting in the cross‐linked graft copolymer network. Silver nanoparticles (SNs) were formed and stabilized by the reduction of silver nitrate using tri‐sodium citrate. The TG‐g‐PAMPS gel and its nanocomposite were characterized and confirmed using FTIR, TGA, XRD, SEM, EDS, and TEM techniques. It is observed that the presence of SNs significantly improves the swelling ability of the TG‐g‐PAMPS gel. Degradation studies of both hydrogels were studied using the soil burial method and determining the respective weight loss. The presence of SNs is found to impart significant antibacterial properties to the gel against Pseudomonas aeruginosa and Escherichia coli bacteria. Further, the TG‐g‐PAMPS gel and TG‐g‐PAMPS‐SN were evaluated as matrix materials for the release of the drug (diclofenac sodium) and the effect of SNs on the release was examined. The in‐vitro released data were analyzed using empirical equations to understand the mechanism of release. Among the various models, the released data were well fitted into the Korsmeyer–Peppas equation and the released kinetics followed non‐Fickian diffusion.https://doi.org/10.1002/nano.202300200antibacterial activitydrug deliveryKorsmeyer–Peppas modelmicrowave radiationsilver nanoparticlestragacanth gum
spellingShingle Sharanappa Chapi
Gangadhar Babaladimath
M. V. Murugendrappa
Anjanapura V. Raghu
Microwave‐Assisted Tragacanth Gum–Based Grafted Silver Nanocomposite Hydrogel for Sustained Release Formulations of Diclofenac Sodium and Antibacterial Assay
Nano Select
antibacterial activity
drug delivery
Korsmeyer–Peppas model
microwave radiation
silver nanoparticles
tragacanth gum
title Microwave‐Assisted Tragacanth Gum–Based Grafted Silver Nanocomposite Hydrogel for Sustained Release Formulations of Diclofenac Sodium and Antibacterial Assay
title_full Microwave‐Assisted Tragacanth Gum–Based Grafted Silver Nanocomposite Hydrogel for Sustained Release Formulations of Diclofenac Sodium and Antibacterial Assay
title_fullStr Microwave‐Assisted Tragacanth Gum–Based Grafted Silver Nanocomposite Hydrogel for Sustained Release Formulations of Diclofenac Sodium and Antibacterial Assay
title_full_unstemmed Microwave‐Assisted Tragacanth Gum–Based Grafted Silver Nanocomposite Hydrogel for Sustained Release Formulations of Diclofenac Sodium and Antibacterial Assay
title_short Microwave‐Assisted Tragacanth Gum–Based Grafted Silver Nanocomposite Hydrogel for Sustained Release Formulations of Diclofenac Sodium and Antibacterial Assay
title_sort microwave assisted tragacanth gum based grafted silver nanocomposite hydrogel for sustained release formulations of diclofenac sodium and antibacterial assay
topic antibacterial activity
drug delivery
Korsmeyer–Peppas model
microwave radiation
silver nanoparticles
tragacanth gum
url https://doi.org/10.1002/nano.202300200
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