Evaluation of bioequivalence of two tablet forms of lisinopril in healthy volunteers

Under cross, single, open, randomized trial with 1 week washout period, with two sequences of 18 volunteers studied bioequivalence coated tablets, two manufacturers of lisinopril (20 mg dose). The concentration of lisinopril in the plasma samples was determined using HPLC with fluorimetric detection...

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Main Authors: S. A. Altynbekov, G. A. Dzholdygulov, V. N. Seryakov, Y. M. Budach, O. E. Kurilo, N. I. Kuznetsova
Format: Article
Language:Russian
Published: LLC “Publisher OKI” 2013-09-01
Series:Фармакокинетика и Фармакодинамика
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Online Access:https://www.pharmacokinetica.ru/jour/article/view/133
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author S. A. Altynbekov
G. A. Dzholdygulov
V. N. Seryakov
Y. M. Budach
O. E. Kurilo
N. I. Kuznetsova
author_facet S. A. Altynbekov
G. A. Dzholdygulov
V. N. Seryakov
Y. M. Budach
O. E. Kurilo
N. I. Kuznetsova
author_sort S. A. Altynbekov
collection DOAJ
description Under cross, single, open, randomized trial with 1 week washout period, with two sequences of 18 volunteers studied bioequivalence coated tablets, two manufacturers of lisinopril (20 mg dose). The concentration of lisinopril in the plasma samples was determined using HPLC with fluorimetric detection within 72 hours for the investigated preparations the following pharmacokinetic parameters were calculated:AUC0-∞, Cmax, tmax, Cmax/AUC. 90% confidence interval relations AUC0-∞ compared drugs totaled 0.8520 — 1.2102 for Cmax — 0,9288 — 1,1451. In addition to the 90% confidence intervals, analysis of variance revealed no statistically significant differences between the studied drugs. Concluded bioequivalence compared drugs lisinopril.
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institution DOAJ
issn 2587-7836
2686-8830
language Russian
publishDate 2013-09-01
publisher LLC “Publisher OKI”
record_format Article
series Фармакокинетика и Фармакодинамика
spelling doaj-art-27f4e88bf2c7447db6b423e07dd636422025-08-20T03:20:16ZrusLLC “Publisher OKI”Фармакокинетика и Фармакодинамика2587-78362686-88302013-09-01023336132Evaluation of bioequivalence of two tablet forms of lisinopril in healthy volunteersS. A. Altynbekov0G. A. Dzholdygulov1V. N. Seryakov2Y. M. Budach3O. E. Kurilo4N. I. Kuznetsova5Republican Scientific and Practical Centre for Psychiatry, Psychotherapy and Addiction, MoH, Republic of Kazakhstan, AlmatyRepublican Scientific and Practical Centre for Psychiatry, Psychotherapy and Addiction, MoH, Republic of Kazakhstan, AlmatyRepublican Scientific and Practical Centre for Psychiatry, Psychotherapy and Addiction, MoH, Republic of Kazakhstan, AlmatyJSC «Chimpharm», Republic of Kazakhstan, AlmatyJSC «Chimpharm», Republic of Kazakhstan, AlmatyMedical University «First Moscow State University, I.M. Sechenov»Under cross, single, open, randomized trial with 1 week washout period, with two sequences of 18 volunteers studied bioequivalence coated tablets, two manufacturers of lisinopril (20 mg dose). The concentration of lisinopril in the plasma samples was determined using HPLC with fluorimetric detection within 72 hours for the investigated preparations the following pharmacokinetic parameters were calculated:AUC0-∞, Cmax, tmax, Cmax/AUC. 90% confidence interval relations AUC0-∞ compared drugs totaled 0.8520 — 1.2102 for Cmax — 0,9288 — 1,1451. In addition to the 90% confidence intervals, analysis of variance revealed no statistically significant differences between the studied drugs. Concluded bioequivalence compared drugs lisinopril.https://www.pharmacokinetica.ru/jour/article/view/133лизиноприлвэжхфлуорометрическое детектированиебиоэквивалентностьlisinoprilhplcfluorometric detectionbioequivalence
spellingShingle S. A. Altynbekov
G. A. Dzholdygulov
V. N. Seryakov
Y. M. Budach
O. E. Kurilo
N. I. Kuznetsova
Evaluation of bioequivalence of two tablet forms of lisinopril in healthy volunteers
Фармакокинетика и Фармакодинамика
лизиноприл
вэжх
флуорометрическое детектирование
биоэквивалентность
lisinopril
hplc
fluorometric detection
bioequivalence
title Evaluation of bioequivalence of two tablet forms of lisinopril in healthy volunteers
title_full Evaluation of bioequivalence of two tablet forms of lisinopril in healthy volunteers
title_fullStr Evaluation of bioequivalence of two tablet forms of lisinopril in healthy volunteers
title_full_unstemmed Evaluation of bioequivalence of two tablet forms of lisinopril in healthy volunteers
title_short Evaluation of bioequivalence of two tablet forms of lisinopril in healthy volunteers
title_sort evaluation of bioequivalence of two tablet forms of lisinopril in healthy volunteers
topic лизиноприл
вэжх
флуорометрическое детектирование
биоэквивалентность
lisinopril
hplc
fluorometric detection
bioequivalence
url https://www.pharmacokinetica.ru/jour/article/view/133
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AT gadzholdygulov evaluationofbioequivalenceoftwotabletformsoflisinoprilinhealthyvolunteers
AT vnseryakov evaluationofbioequivalenceoftwotabletformsoflisinoprilinhealthyvolunteers
AT ymbudach evaluationofbioequivalenceoftwotabletformsoflisinoprilinhealthyvolunteers
AT oekurilo evaluationofbioequivalenceoftwotabletformsoflisinoprilinhealthyvolunteers
AT nikuznetsova evaluationofbioequivalenceoftwotabletformsoflisinoprilinhealthyvolunteers