3‐HKA Promotes Vascular Remodeling After Stroke by Modulating the Activation of A1/A2 Reactive Astrocytes

Abstract Ischemic stroke is the most common cerebrovascular disease and the leading cause of permanent disability worldwide. Recent studies have shown that stroke development and prognosis are closely related to abnormal tryptophan metabolism. Here, significant downregulation of 3‐hydroxy‐kynurenami...

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Main Authors: Jun‐Min Chen, Guang Shi, Lu‐Lu Yu, Wei Shan, Jing‐Yu Sun, An‐Chen Guo, Jian‐Ping Wu, Tie‐Shan Tang, Xiang‐Jian Zhang, Qun Wang
Format: Article
Language:English
Published: Wiley 2025-03-01
Series:Advanced Science
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Online Access:https://doi.org/10.1002/advs.202412667
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author Jun‐Min Chen
Guang Shi
Lu‐Lu Yu
Wei Shan
Jing‐Yu Sun
An‐Chen Guo
Jian‐Ping Wu
Tie‐Shan Tang
Xiang‐Jian Zhang
Qun Wang
author_facet Jun‐Min Chen
Guang Shi
Lu‐Lu Yu
Wei Shan
Jing‐Yu Sun
An‐Chen Guo
Jian‐Ping Wu
Tie‐Shan Tang
Xiang‐Jian Zhang
Qun Wang
author_sort Jun‐Min Chen
collection DOAJ
description Abstract Ischemic stroke is the most common cerebrovascular disease and the leading cause of permanent disability worldwide. Recent studies have shown that stroke development and prognosis are closely related to abnormal tryptophan metabolism. Here, significant downregulation of 3‐hydroxy‐kynurenamine (3‐HKA) in stroke patients and animal models is identified. Supplementation with 3‐HKA improved long‐term neurological recovery, reduced infarct volume, and increased ipsilateral cerebral blood flow after distal middle cerebral artery occlusion (MCAO). 3‐HKA promoted angiogenesis, functional blood vessel formation, and blood‐brain barrier (BBB) repair. Moreover, 3‐HKA inhibited A1‐like (neurotoxic) astrocyte activation but promoted A2‐like (neuroprotective) astrocyte polarization. Proteomic analysis revealed that 3‐HKA inhibited AIM2 inflammasome activation after stroke, and co‐labeling studies indicated that AIM2 expression typically increased in astrocytes at 7 and 14 days after stroke. Consistently, in co‐cultures of primary mouse brain microvascular endothelial cells and astrocytes, 3‐HKA promoted angiogenesis after oxygen‐glucose deprivation (OGD). AIM2 overexpression in astrocytes abrogated 3‐HKA‐driven vascular remodeling in vitro and in vivo, suggesting that 3‐HKA may regulate astrocyte‐mediated vascular remodeling by impeding AIM2 inflammasome activation. In conclusion, 3‐HKA may promote post‐stroke vascular remodeling by regulating A1/A2 astrocyte activation, thereby improving long‐term neurological recovery, suggesting that supplementation with 3‐HKA may be an efficient therapy for stroke.
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spelling doaj-art-275806d40c3348598451ba26bbc72e862025-08-20T02:24:47ZengWileyAdvanced Science2198-38442025-03-011211n/an/a10.1002/advs.2024126673‐HKA Promotes Vascular Remodeling After Stroke by Modulating the Activation of A1/A2 Reactive AstrocytesJun‐Min Chen0Guang Shi1Lu‐Lu Yu2Wei Shan3Jing‐Yu Sun4An‐Chen Guo5Jian‐Ping Wu6Tie‐Shan Tang7Xiang‐Jian Zhang8Qun Wang9Department of Neurology Beijing Tiantan Hospital Capital Medical University Beijing 100070 ChinaDepartment of Neurology Second Hospital of Hebei Medical University Shijiazhuang 050000 ChinaDepartment of Neurology Beijing Tiantan Hospital Capital Medical University Beijing 100070 ChinaDepartment of Neurology Beijing Tiantan Hospital Capital Medical University Beijing 100070 ChinaKey Laboratory of Organ Regeneration and Reconstruction State Key Laboratory of Membrane Biology Institute of Zoology Chinese Academy of Sciences Beijing 100101 ChinaChina National Clinical Research Center for Neurological Diseases Beijing 100070 ChinaDepartment of Neurology Beijing Tiantan Hospital Capital Medical University Beijing 100070 ChinaKey Laboratory of Organ Regeneration and Reconstruction State Key Laboratory of Membrane Biology Institute of Zoology Chinese Academy of Sciences Beijing 100101 ChinaDepartment of Neurology Second Hospital of Hebei Medical University Shijiazhuang 050000 ChinaDepartment of Neurology Beijing Tiantan Hospital Capital Medical University Beijing 100070 ChinaAbstract Ischemic stroke is the most common cerebrovascular disease and the leading cause of permanent disability worldwide. Recent studies have shown that stroke development and prognosis are closely related to abnormal tryptophan metabolism. Here, significant downregulation of 3‐hydroxy‐kynurenamine (3‐HKA) in stroke patients and animal models is identified. Supplementation with 3‐HKA improved long‐term neurological recovery, reduced infarct volume, and increased ipsilateral cerebral blood flow after distal middle cerebral artery occlusion (MCAO). 3‐HKA promoted angiogenesis, functional blood vessel formation, and blood‐brain barrier (BBB) repair. Moreover, 3‐HKA inhibited A1‐like (neurotoxic) astrocyte activation but promoted A2‐like (neuroprotective) astrocyte polarization. Proteomic analysis revealed that 3‐HKA inhibited AIM2 inflammasome activation after stroke, and co‐labeling studies indicated that AIM2 expression typically increased in astrocytes at 7 and 14 days after stroke. Consistently, in co‐cultures of primary mouse brain microvascular endothelial cells and astrocytes, 3‐HKA promoted angiogenesis after oxygen‐glucose deprivation (OGD). AIM2 overexpression in astrocytes abrogated 3‐HKA‐driven vascular remodeling in vitro and in vivo, suggesting that 3‐HKA may regulate astrocyte‐mediated vascular remodeling by impeding AIM2 inflammasome activation. In conclusion, 3‐HKA may promote post‐stroke vascular remodeling by regulating A1/A2 astrocyte activation, thereby improving long‐term neurological recovery, suggesting that supplementation with 3‐HKA may be an efficient therapy for stroke.https://doi.org/10.1002/advs.2024126673‐hydroxy‐kynurenamineAIM2 inflammasomesischemic strokereactive astrocytesvascular remodeling
spellingShingle Jun‐Min Chen
Guang Shi
Lu‐Lu Yu
Wei Shan
Jing‐Yu Sun
An‐Chen Guo
Jian‐Ping Wu
Tie‐Shan Tang
Xiang‐Jian Zhang
Qun Wang
3‐HKA Promotes Vascular Remodeling After Stroke by Modulating the Activation of A1/A2 Reactive Astrocytes
Advanced Science
3‐hydroxy‐kynurenamine
AIM2 inflammasomes
ischemic stroke
reactive astrocytes
vascular remodeling
title 3‐HKA Promotes Vascular Remodeling After Stroke by Modulating the Activation of A1/A2 Reactive Astrocytes
title_full 3‐HKA Promotes Vascular Remodeling After Stroke by Modulating the Activation of A1/A2 Reactive Astrocytes
title_fullStr 3‐HKA Promotes Vascular Remodeling After Stroke by Modulating the Activation of A1/A2 Reactive Astrocytes
title_full_unstemmed 3‐HKA Promotes Vascular Remodeling After Stroke by Modulating the Activation of A1/A2 Reactive Astrocytes
title_short 3‐HKA Promotes Vascular Remodeling After Stroke by Modulating the Activation of A1/A2 Reactive Astrocytes
title_sort 3 hka promotes vascular remodeling after stroke by modulating the activation of a1 a2 reactive astrocytes
topic 3‐hydroxy‐kynurenamine
AIM2 inflammasomes
ischemic stroke
reactive astrocytes
vascular remodeling
url https://doi.org/10.1002/advs.202412667
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