Photodynamic therapy of the experimental tumors of different morphological types with liposomal boronated chlorin е6

The article summarizes the results of studies of the effectiveness of photodynamic therapy using a new domestic photosensitizer liposomal borated chlorin e6 (LBC) after its parenteral administration (intraperitoneal and intravenous). Antitumor efficacy was evaluated in rats with M-1 sarcoma and PC-1...

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Main Authors: O. B. Abramova, V. V. Drozhzhina, T. P. Churikova, E. A. Kozlovtceva, L. M. Arkhipova, M. A. Kaplan, S. A. Ivanov, A. D. Kaprin
Format: Article
Language:Russian
Published: Non-profit partnership for development of domestic photodynamic therapy and photodiagnosis "Russian Photodynamic Association" 2021-10-01
Series:Biomedical Photonics
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Online Access:https://www.pdt-journal.com/jour/article/view/501
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author O. B. Abramova
V. V. Drozhzhina
T. P. Churikova
E. A. Kozlovtceva
L. M. Arkhipova
M. A. Kaplan
S. A. Ivanov
A. D. Kaprin
author_facet O. B. Abramova
V. V. Drozhzhina
T. P. Churikova
E. A. Kozlovtceva
L. M. Arkhipova
M. A. Kaplan
S. A. Ivanov
A. D. Kaprin
author_sort O. B. Abramova
collection DOAJ
description The article summarizes the results of studies of the effectiveness of photodynamic therapy using a new domestic photosensitizer liposomal borated chlorin e6 (LBC) after its parenteral administration (intraperitoneal and intravenous). Antitumor efficacy was evaluated in rats with M-1 sarcoma and PC-1 alveolar liver cancer and mice with B16 melanoma and Ehrlich’s carcinoma, which were transplanted subcutaneously into the thigh area of the animals. The aim of the study was to determine the optimal regimes of photodynamic therapy that would allow achieving the maximum antitumor effect up to 21 days after the photodynamic therapy. The therapy was carried out under the control of the accumulation of the photosensitizer in the tumor and surrounding tissues of the thigh by selecting the doses of the drug and the parameters of laser radiation (energy density and power density). The effectiveness of therapy was assessed by the inhibition of tumor growth, by the percentage of animals with complete tumor regression, by the absolute growth rate in animals with continued tumor growth compared to controls. The results of our studies have shown that the domestic photosensitizer liposomal borated chlorin e6 has high antitumor activity in vivo. In an experimental study of the photosensitizer under certain PDT modes, the maximum antitumor effect (complete tumor regression in 100% of animals) was obtained up to 21 days after PDT in all tumor models used.
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id doaj-art-1fe03d4fe4624ff3be758a2d09ef59ae
institution DOAJ
issn 2413-9432
language Russian
publishDate 2021-10-01
publisher Non-profit partnership for development of domestic photodynamic therapy and photodiagnosis "Russian Photodynamic Association"
record_format Article
series Biomedical Photonics
spelling doaj-art-1fe03d4fe4624ff3be758a2d09ef59ae2025-08-20T03:21:05ZrusNon-profit partnership for development of domestic photodynamic therapy and photodiagnosis "Russian Photodynamic Association"Biomedical Photonics2413-94322021-10-01103122210.24931/2413-9432-2021-10-3-12-22236Photodynamic therapy of the experimental tumors of different morphological types with liposomal boronated chlorin е6O. B. Abramova0V. V. Drozhzhina1T. P. Churikova2E. A. Kozlovtceva3L. M. Arkhipova4M. A. Kaplan5S. A. Ivanov6A. D. Kaprin7A.Tsyb Medical Radiological Research Center – branch of the National Medical Research Radiological CenterA.Tsyb Medical Radiological Research Center – branch of the National Medical Research Radiological CenterA.Tsyb Medical Radiological Research Center – branch of the National Medical Research Radiological CenterA.Tsyb Medical Radiological Research Center – branch of the National Medical Research Radiological CenterA.Tsyb Medical Radiological Research Center – branch of the National Medical Research Radiological CenterA.Tsyb Medical Radiological Research Center – branch of the National Medical Research Radiological CenterA.Tsyb Medical Radiological Research Center – branch of the National Medical Research Radiological CenterA.Tsyb Medical Radiological Research Center – branch of the National Medical Research Radiological CenterThe article summarizes the results of studies of the effectiveness of photodynamic therapy using a new domestic photosensitizer liposomal borated chlorin e6 (LBC) after its parenteral administration (intraperitoneal and intravenous). Antitumor efficacy was evaluated in rats with M-1 sarcoma and PC-1 alveolar liver cancer and mice with B16 melanoma and Ehrlich’s carcinoma, which were transplanted subcutaneously into the thigh area of the animals. The aim of the study was to determine the optimal regimes of photodynamic therapy that would allow achieving the maximum antitumor effect up to 21 days after the photodynamic therapy. The therapy was carried out under the control of the accumulation of the photosensitizer in the tumor and surrounding tissues of the thigh by selecting the doses of the drug and the parameters of laser radiation (energy density and power density). The effectiveness of therapy was assessed by the inhibition of tumor growth, by the percentage of animals with complete tumor regression, by the absolute growth rate in animals with continued tumor growth compared to controls. The results of our studies have shown that the domestic photosensitizer liposomal borated chlorin e6 has high antitumor activity in vivo. In an experimental study of the photosensitizer under certain PDT modes, the maximum antitumor effect (complete tumor regression in 100% of animals) was obtained up to 21 days after PDT in all tumor models used.https://www.pdt-journal.com/jour/article/view/501photodynamic therapypharmacokineticslaserliposomal borated chlorin e6rat sarcoma m-1rat alveolar cancer liver pc-1mouse melanoma в16mouse ehrlich’s carcinoma
spellingShingle O. B. Abramova
V. V. Drozhzhina
T. P. Churikova
E. A. Kozlovtceva
L. M. Arkhipova
M. A. Kaplan
S. A. Ivanov
A. D. Kaprin
Photodynamic therapy of the experimental tumors of different morphological types with liposomal boronated chlorin е6
Biomedical Photonics
photodynamic therapy
pharmacokinetics
laser
liposomal borated chlorin e6
rat sarcoma m-1
rat alveolar cancer liver pc-1
mouse melanoma в16
mouse ehrlich’s carcinoma
title Photodynamic therapy of the experimental tumors of different morphological types with liposomal boronated chlorin е6
title_full Photodynamic therapy of the experimental tumors of different morphological types with liposomal boronated chlorin е6
title_fullStr Photodynamic therapy of the experimental tumors of different morphological types with liposomal boronated chlorin е6
title_full_unstemmed Photodynamic therapy of the experimental tumors of different morphological types with liposomal boronated chlorin е6
title_short Photodynamic therapy of the experimental tumors of different morphological types with liposomal boronated chlorin е6
title_sort photodynamic therapy of the experimental tumors of different morphological types with liposomal boronated chlorin е6
topic photodynamic therapy
pharmacokinetics
laser
liposomal borated chlorin e6
rat sarcoma m-1
rat alveolar cancer liver pc-1
mouse melanoma в16
mouse ehrlich’s carcinoma
url https://www.pdt-journal.com/jour/article/view/501
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